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PDB: 1 results

5ONE
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BU of 5one by Molmil
Crystal structure of Aurora-A in complex with FMF-03-145-1 (compound 2)
Descriptor: 4-(propanoylamino)-~{N}-[4-[(5,8,11-trimethyl-6-oxidanylidene-pyrimido[4,5-b][1,4]benzodiazepin-2-yl)amino]phenyl]benzamide, Aurora kinase A
Authors:Chaikuad, A, Ferguson, F.M, Gray, N.S, Knapp, S.
Deposit date:2017-08-03
Release date:2017-09-06
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Characterization of a highly selective inhibitor of the Aurora kinases.
Bioorg. Med. Chem. Lett., 27, 2017

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