English
日本語
简体中文
繁體中文
한국어
✖
Menu
RCSB PDB
PDBe
BMRB
Adv. Search
Search help
PDB: 2 results
5LMB
HUMAN SPLEEN TYROSINE KINASE KINASE DOMAIN IN COMPLEX WITH AZANAPHTHYRIDINE INHIBITOR
Descriptor:
7-[6-(dimethylamino)pyridin-3-yl]-~{N}-[[(3~{S})-piperidin-3-yl]methyl]pyrido[3,4-b]pyrazin-5-amine, GLYCEROL, Tyrosine-protein kinase SYK
Authors:
Somers, D.O
,
Neu, M.
Deposit date:
2016-07-29
Release date:
2016-09-14
Last modified:
2024-05-01
Method:
X-RAY DIFFRACTION (1.95 Å)
Cite:
Optimisation of a novel series of potent and orally bioavailable azanaphthyridine SYK inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
5LMA
HUMAN SPLEEN TYROSINE KINASE KINASE DOMAIN IN COMPLEX WITH AZANAPHTHYRIDINE INHIBITOR
Descriptor:
DIMETHYL SULFOXIDE, GLYCEROL, Tyrosine-protein kinase SYK, ...
Authors:
Somers, D.O
,
Neu, M.
Deposit date:
2016-07-29
Release date:
2016-09-14
Last modified:
2024-05-01
Method:
X-RAY DIFFRACTION (1.43 Å)
Cite:
Optimisation of a novel series of potent and orally bioavailable azanaphthyridine SYK inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016
Home
Top Page
Statistics
Help
FAQ
Contact Us
Cite Us / Terms and Conditions
Links
Settings
Data deposition (OneDep)
Help
Deposition to PDB, EMDB or BMRB
Download
Download PDB archive / snapshot archive
Standard format
PDBx/mmCIF Resources
Format Conversion
PDBx/mmCIF editor
Quick links
Help
non-PDB format compatible
Group Depositions
Chemical Component entries
Latest entries
Search services
Help
Search PDB (PDBj Mine)
Search PDBj RDB
Chemie search
Search BMRB
Sequence-Navigator
DASH
EM Navigator
Omokage search
SeSAW
wwPDB/RDF
RDF Portal
Status search
Molecular Viewers
Help
jV: Graphic Viewer
Molmil: WebGL Mol. Viewer
Services & Softwares
Help
Yorodumi
ASH
MAFFTash
NMRToolBox
gmfit
CRNPRED
Spanner
SFAS
HOMCOS
Derived databases
Help
eF-site
eF-seek
eF-surf
ProMode Elastic
hGTOP
Educational service
Help
eProtS
Molecule of the Month
Previous workshop
Games
Papermodels
About PDBj
Help
Publications
Newsletters / Public Relations Resources
PDBj Members
PDBj Advisory Committee
Privacy Policy
222415
PDB entries from 2024-07-10