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PDB: 1 results

5K9R
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BU of 5k9r by Molmil
PDE10a with imidazopyrazine inhibitor
Descriptor: 4-[5-[1-(2-methoxyethyl)pyrazol-4-yl]-2-(quinolin-2-yloxymethyl)imidazo[1,2-a]pyrazin-8-yl]morpholine, MAGNESIUM ION, ZINC ION, ...
Authors:Gibbs, A.G, Schubert, C.
Deposit date:2016-06-01
Release date:2016-08-24
Method:X-RAY DIFFRACTION (2.7 Å)
Cite:Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitors.
Bioorg.Med.Chem.Lett., 26, 2016

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