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PDB: 1 results
5M2B
Yeast 20S proteasome with human beta5i (1-138) and human beta6 (97-111; 118-133) in complex with thiazole based inhibitor Ro19
Descriptor:
(2~{S})-2-cyclohexyl-4-oxidanylidene-4-[[7-(4-phenyl-1,3-thiazol-2-yl)quinolin-2-yl]amino]butanoic acid, CHLORIDE ION, MAGNESIUM ION, ...
Authors:
Groll, M.
Deposit date:
2016-10-12
Release date:
2017-01-25
Last modified:
2024-01-17
Method:
X-RAY DIFFRACTION (2.7 Å)
Cite:
Structural Elucidation of a Nonpeptidic Inhibitor Specific for the Human Immunoproteasome.
Chembiochem, 18, 2017
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PDB entries from 2024-07-10