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PDB: 1 results
6YIZ
Crystal structure of PqsR (MvfR) ligand-binding domain in complex with triazolo-pyridine inverse agonist A
Descriptor:
7-oxidanylidene-8-[2-(4-sulfonaphthalen-1-yl)hydrazinyl]-8~{H}-naphthalene-1,3-disulfonic acid, MAGNESIUM ION, Transcriptional regulator MvfR, ...
Authors:
Schmelz, S
,
Blankenfeldt, W.
Deposit date:
2020-04-01
Release date:
2021-04-14
Last modified:
2024-01-24
Method:
X-RAY DIFFRACTION (2.163 Å)
Cite:
A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate Pseudomonas aeruginosa Biofilms.
Adv Sci, 8, 2021
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PDB entries from 2025-07-09