6UJS
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![BU of 6ujs by Molmil](/molmil-images/mine/6ujs) | P-glycoprotein mutant-F728A and C952A-with BDE100 | Descriptor: | 2,4-dibromophenyl 2,4,6-tribromophenyl ether, ATP-dependent translocase ABCB1 | Authors: | Aller, S.G, Le, C.A. | Deposit date: | 2019-10-03 | Release date: | 2020-05-27 | Last modified: | 2023-10-11 | Method: | X-RAY DIFFRACTION (4.17 Å) | Cite: | Structural definition of polyspecific compensatory ligand recognition by P-glycoprotein. Iucrj, 7, 2020
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4L31
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![BU of 4l31 by Molmil](/molmil-images/mine/4l31) | Tankyrase 2 in complex with methyl 4-(4-oxochromen-2-yl)benzoate | Descriptor: | GLYCEROL, SULFATE ION, Tankyrase-2, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-06-05 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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4KZU
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![BU of 4kzu by Molmil](/molmil-images/mine/4kzu) | Crystal structure of human tankyrase 2 in complex with 4' -bromo flavone | Descriptor: | 2-(4-bromophenyl)-4H-chromen-4-one, GLYCEROL, SULFATE ION, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-05-30 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.1 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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4L32
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![BU of 4l32 by Molmil](/molmil-images/mine/4l32) | Tankyrase 2 in complex with 2-[4-(4-methylpiperazine-1-carbonyl)phenyl]chromen-4-one | Descriptor: | 2-{4-[(4-methylpiperazin-1-yl)carbonyl]phenyl}-4H-chromen-4-one, GLYCEROL, SULFATE ION, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-06-05 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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4PFC
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![BU of 4pfc by Molmil](/molmil-images/mine/4pfc) | Crystal structure of insulin degrading enzyme complexed with inhibitor | Descriptor: | Insulin-degrading enzyme, ZINC ION, methyl [(2S)-2-(5-{5-[4-({(2S)-2-[(3S)-3-amino-2-oxopiperidin-1-yl]-2-cyclohexylacetyl}amino)phenyl]pentyl}-2-fluorophenyl)-3-(quinolin-3-yl)propyl]carbamate | Authors: | Wang, Y, Guo, S. | Deposit date: | 2014-04-28 | Release date: | 2015-06-17 | Last modified: | 2023-09-27 | Method: | X-RAY DIFFRACTION (2.21 Å) | Cite: | Dual Exosite-binding Inhibitors of Insulin-degrading Enzyme Challenge Its Role as the Primary Mediator of Insulin Clearance in Vivo. J.Biol.Chem., 290, 2015
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4L09
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![BU of 4l09 by Molmil](/molmil-images/mine/4l09) | Crystal structure of human tankyrase 2 in complex with 4-(4-oxo-4H-chromen-2-yl)benzoic acid | Descriptor: | 4-(4-oxo-4H-chromen-2-yl)benzoic acid, GLYCEROL, SULFATE ION, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-05-31 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.05 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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4L34
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![BU of 4l34 by Molmil](/molmil-images/mine/4l34) | Tankyrase 2 in complex with 4'-tetrazole flavone | Descriptor: | 2-[4-(1H-tetrazol-5-yl)phenyl]-4H-chromen-4-one, GLYCEROL, SULFATE ION, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-06-05 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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4KZQ
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![BU of 4kzq by Molmil](/molmil-images/mine/4kzq) | Crystal structure of human tankyrase 2 in complex with 4' -hydroxy flavone | Descriptor: | 2-(4-HYDROXY-PHENYL)-CHROMAN-4-ONE, SULFATE ION, Tankyrase-2, ... | Authors: | Narwal, M, Haikarainen, T, Lehtio, L. | Deposit date: | 2013-05-30 | Release date: | 2013-10-30 | Last modified: | 2023-09-20 | Method: | X-RAY DIFFRACTION (2.25 Å) | Cite: | Discovery of tankyrase inhibiting flavones with increased potency and isoenzyme selectivity. J.Med.Chem., 56, 2013
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2FPP
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![BU of 2fpp by Molmil](/molmil-images/mine/2fpp) | Crystal structure of pig GTP-specific succinyl-CoA synthetase from polyethylene glycol with chloride ions | Descriptor: | CHLORIDE ION, SULFATE ION, Succinyl-CoA ligase [GDP-forming] alpha-chain, ... | Authors: | Fraser, M.E, Hayakawa, K, Hume, M.S, Ryan, D.G, Brownie, E.R. | Deposit date: | 2006-01-16 | Release date: | 2006-02-21 | Last modified: | 2017-10-18 | Method: | X-RAY DIFFRACTION (2.35 Å) | Cite: | Interactions of GTP with the ATP-grasp Domain of GTP-specific Succinyl-CoA Synthetase J.Biol.Chem., 281, 2006
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2FPG
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2FP4
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2FPI
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2YDM
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![BU of 2ydm by Molmil](/molmil-images/mine/2ydm) | Structural characterization of angiotensin-I converting enzyme in complex with a selenium analogue of captopril | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, ANGIOTENSIN CONVERTING ENZYME, CHLORIDE ION, ... | Authors: | Akif, M, Masuyer, G, Schwager, S.L.U, Bhuyan, B.J, Mugesh, G, Sturrock, E.D, Acharya, K.R. | Deposit date: | 2011-03-22 | Release date: | 2011-09-14 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.44 Å) | Cite: | Structural Characterization of Angiotensin-I Converting Enzyme in Complex with a Selenium Analogue of Captopril FEBS J., 278, 2011
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5XHZ
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![BU of 5xhz by Molmil](/molmil-images/mine/5xhz) | Crystal Structure Analysis of CIN85-SH3B in complex with ARAP1-P2 | Descriptor: | ACETATE ION, Arf-GAP with Rho-GAP domain, ANK repeat and PH domain-containing protein 1, ... | Authors: | Liu, W, Yang, W. | Deposit date: | 2017-04-25 | Release date: | 2018-04-11 | Last modified: | 2023-11-22 | Method: | X-RAY DIFFRACTION (1.319 Å) | Cite: | Biochemical and Structural Studies of the Interaction between ARAP1 and CIN85. Biochemistry, 57, 2018
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1LSM
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![BU of 1lsm by Molmil](/molmil-images/mine/1lsm) | |
1LSN
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![BU of 1lsn by Molmil](/molmil-images/mine/1lsn) | |
7ICF
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![BU of 7icf by Molmil](/molmil-images/mine/7icf) | |
7ICP
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7ICL
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![BU of 7icl by Molmil](/molmil-images/mine/7icl) | |
7ICV
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![BU of 7icv by Molmil](/molmil-images/mine/7icv) | |
7ICG
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![BU of 7icg by Molmil](/molmil-images/mine/7icg) | |
7ICQ
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![BU of 7icq by Molmil](/molmil-images/mine/7icq) | |
7ICK
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![BU of 7ick by Molmil](/molmil-images/mine/7ick) | |
7ICU
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![BU of 7icu by Molmil](/molmil-images/mine/7icu) | |
7ICJ
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![BU of 7icj by Molmil](/molmil-images/mine/7icj) | |