Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

6GDL
DownloadVisualize
BU of 6gdl by Molmil
Calmodulin mutant - F141L apo-form Unstructured C-domain
Descriptor: Calmodulin-1
Authors:Holt, C, Overgaard, M.T, Wimmer, R.
Deposit date:2018-04-23
Release date:2018-10-17
Last modified:2024-05-15
Method:SOLUTION NMR
Cite:Arrhythmia mutations in calmodulin cause conformational changes that affect interactions with the cardiac voltage-gated calcium channel.
Proc. Natl. Acad. Sci. U.S.A., 115, 2018
6XCX
DownloadVisualize
BU of 6xcx by Molmil
Nitric Oxide Synthase from Bacillus subtilis in complex with N2-((3-((2-aminoquinolin-7-yl)methoxy)phenoxy)methyl)pyridine-2,6-diamine
Descriptor: 7-{[3-(2-{[(6-aminopyridin-2-yl)methyl]amino}ethoxy)phenoxy]methyl}quinolin-2-amine, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Lewis, M.C, Poulos, T.L.
Deposit date:2020-06-09
Release date:2021-06-16
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.2520268 Å)
Cite:Selective Anti-MRSA inhibitors targeting Nitric Oxide Synthase
To Be Published
1DJW
DownloadVisualize
BU of 1djw by Molmil
PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-2-METHYLENE-1,2-CYCLIC-MONOPHOSPHONATE
Descriptor: ACETATE ION, CALCIUM ION, INOSITOL-2-METHYLENE-1,2-CYCLIC-MONOPHOSPHATE, ...
Authors:Essen, L.-O, Perisic, O, Williams, R.L.
Deposit date:1996-08-24
Release date:1997-07-23
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.45 Å)
Cite:Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
1DJX
DownloadVisualize
BU of 1djx by Molmil
PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-1,4,5-TRISPHOSPHATE
Descriptor: ACETATE ION, CALCIUM ION, D-MYO-INOSITOL-1,4,5-TRIPHOSPHATE, ...
Authors:Essen, L.-O, Perisic, O, Williams, R.L.
Deposit date:1996-08-24
Release date:1997-07-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
1DSO
DownloadVisualize
BU of 1dso by Molmil
CYTOCHROME C PEROXIDASE H175G MUTANT, IMIDAZOLE COMPLEX AT PH 6, ROOM TEMPERATURE.
Descriptor: CYTOCHROME C PEROXIDASE, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE
Authors:Hirst, J, Wilcox, S.K, Williams, P.A, McRee, D.E, Goodin, D.B.
Deposit date:2000-01-07
Release date:2001-03-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Replacement of the axial histidine ligand with imidazole in cytochrome c peroxidase. 1. Effects on structure.
Biochemistry, 40, 2001
1DSE
DownloadVisualize
BU of 1dse by Molmil
CYTOCHROME C PEROXIDASE H175G MUTANT, IMIDAZOLE COMPLEX, WITH PHOSPHATE BOUND, PH 6, 100K
Descriptor: CYTOCHROME C PEROXIDASE, IMIDAZOLE, PHOSPHATE ION, ...
Authors:Hirst, J, Wilcox, S.K, Williams, P.A, McRee, D.E, Goodin, D.B.
Deposit date:2000-01-07
Release date:2001-03-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2 Å)
Cite:Replacement of the axial histidine ligand with imidazole in cytochrome c peroxidase. 1. Effects on structure.
Biochemistry, 40, 2001
6Y3J
DownloadVisualize
BU of 6y3j by Molmil
RING-DTC domains of Deltex 2, bound to ADP-ribose
Descriptor: ADENOSINE-5-DIPHOSPHORIBOSE, Probable E3 ubiquitin-protein ligase DTX2, ZINC ION
Authors:Gabrielssen, M, Buetow, L, Huang, D.T.
Deposit date:2020-02-18
Release date:2020-09-02
Last modified:2024-01-24
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:DELTEX2 C-terminal domain recognizes and recruits ADP-ribosylated proteins for ubiquitination.
Sci Adv, 6, 2020
1DSL
DownloadVisualize
BU of 1dsl by Molmil
GAMMA B CRYSTALLIN C-TERMINAL DOMAIN
Descriptor: GAMMA B CRYSTALLIN
Authors:Norledge, B.V, Mayr, E.-M, Glockshuber, R, Bateman, O.A, Slingsby, C, Jaenicke, R, Driessen, H.P.C.
Deposit date:1996-02-01
Release date:1996-07-11
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (1.55 Å)
Cite:The X-ray structures of two mutant crystallin domains shed light on the evolution of multi-domain proteins.
Nat.Struct.Biol., 3, 1996
1DW2
DownloadVisualize
BU of 1dw2 by Molmil
STRUCTURE OF THE NITRIC OXIDE COMPLEX OF REDUCED SHP, AN OXYGEN BINDING CYTOCHROME C
Descriptor: CYTOCHROME C, NITRIC OXIDE, PROTOPORPHYRIN IX CONTAINING FE
Authors:Leys, D, Backers, K, Meyer, T.E, Hagen, W.R, Cusanovich, M.A, Van Beeumen, J.J.
Deposit date:2000-01-24
Release date:2000-06-28
Last modified:2024-11-06
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal structures of an oxygen-binding cytochrome c from Rhodobacter sphaeroides.
J.Biol.Chem., 275, 2000
1DS4
DownloadVisualize
BU of 1ds4 by Molmil
CYTOCHROME C PEROXIDASE H175G MUTANT, IMIDAZOLE COMPLEX, PH 6, 100K
Descriptor: CYTOCHROME C PEROXIDASE, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE
Authors:Hirst, J, Wilcox, S.K, Williams, P.A, McRee, D.E, Goodin, D.B.
Deposit date:2000-01-07
Release date:2001-03-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.02 Å)
Cite:Replacement of the axial histidine ligand with imidazole in cytochrome c peroxidase. 1. Effects on structure.
Biochemistry, 40, 2001
6H7Z
DownloadVisualize
BU of 6h7z by Molmil
X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a inhibitor RNA 2-65-1
Descriptor: (2~{S})-2-[[(2~{S})-6-[(6-fluoranylpyridin-3-yl)-methyl-amino]-1-oxidanyl-1,6-bis(oxidanylidene)hexan-2-yl]carbamoylamino]pentanedioic acid, 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ...
Authors:Motlova, L, Novakova, Z, Barinka, C.
Deposit date:2018-07-31
Release date:2018-12-05
Last modified:2024-11-20
Method:X-RAY DIFFRACTION (2 Å)
Cite:2-Aminoadipic Acid-C(O)-Glutamate Based Prostate-Specific Membrane Antigen Ligands for Potential Use as Theranostics.
ACS Med Chem Lett, 9, 2018
1DSP
DownloadVisualize
BU of 1dsp by Molmil
CYTOCHROME C PEROXIDASE H175G MUTANT, IMIDAZOLE COMPLEX AT PH 7, ROOM TEMPERATURE.
Descriptor: CYTOCHROME C PEROXIDASE, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE
Authors:Hirst, J, Wilcox, S.K, Williams, P.A, McRee, D.E, Goodin, D.B.
Deposit date:2000-01-07
Release date:2001-03-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Replacement of the axial histidine ligand with imidazole in cytochrome c peroxidase. 1. Effects on structure.
Biochemistry, 40, 2001
1DSG
DownloadVisualize
BU of 1dsg by Molmil
CYTOCHROME C PEROXIDASE H175G MUTANT, IMIDAZOLE COMPLEX AT PH 5, ROOM TEMPERATURE.
Descriptor: CYTOCHROME C PEROXIDASE, IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE
Authors:Hirst, J, Wilcox, S.K, Williams, P.A, McRee, D.E, Goodin, D.B.
Deposit date:2000-01-07
Release date:2001-03-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.56 Å)
Cite:Replacement of the axial histidine ligand with imidazole in cytochrome c peroxidase. 1. Effects on structure.
Biochemistry, 40, 2001
6NMJ
DownloadVisualize
BU of 6nmj by Molmil
Crystal Structure of Rat Ric-8A G alpha binding domain, "Paratone-N Immersed"
Descriptor: Resistance to inhibitors of cholinesterase 8 homolog A (C. elegans)
Authors:Zeng, B, Mou, T.C, Sprang, S.R.
Deposit date:2019-01-11
Release date:2019-06-26
Last modified:2023-10-11
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Structure, Function, and Dynamics of the G alpha Binding Domain of Ric-8A.
Structure, 27, 2019
5L3M
DownloadVisualize
BU of 5l3m by Molmil
D11 bound [S39_PQ]-IGF-II
Descriptor: Insulin-like growth factor II
Authors:Hexnerova, R.
Deposit date:2016-05-23
Release date:2016-08-10
Last modified:2024-10-23
Method:SOLUTION NMR
Cite:Probing Receptor Specificity by Sampling the Conformational Space of the Insulin-like Growth Factor II C-domain.
J.Biol.Chem., 291, 2016
5L3N
DownloadVisualize
BU of 5l3n by Molmil
D11 bound [N29, S39_PQ]-IGF-II
Descriptor: Insulin-like growth factor II
Authors:Hexnerova, R.
Deposit date:2016-05-23
Release date:2016-08-10
Last modified:2024-11-06
Method:SOLUTION NMR
Cite:Probing Receptor Specificity by Sampling the Conformational Space of the Insulin-like Growth Factor II C-domain.
J.Biol.Chem., 291, 2016
1DJY
DownloadVisualize
BU of 1djy by Molmil
PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-2,4,5-TRISPHOSPHATE
Descriptor: ACETATE ION, CALCIUM ION, D-MYO-INOSITOL-2,4,5-TRIPHOSPHATE, ...
Authors:Essen, L.-O, Perisic, O, Williams, R.L.
Deposit date:1996-08-24
Release date:1997-07-07
Last modified:2024-05-22
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
1DJZ
DownloadVisualize
BU of 1djz by Molmil
PHOSPHOINOSITIDE-SPECIFIC PHOSPHOLIPASE C-DELTA1 FROM RAT COMPLEXED WITH INOSITOL-4,5-BISPHOSPHATE
Descriptor: ACETATE ION, CALCIUM ION, D-MYO-INOSITOL-4,5-BISPHOSPHATE, ...
Authors:Essen, L.-O, Perisic, O, Williams, R.L.
Deposit date:1996-08-24
Release date:1997-07-07
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.95 Å)
Cite:Structural mapping of the catalytic mechanism for a mammalian phosphoinositide-specific phospholipase C.
Biochemistry, 36, 1997
6H6G
DownloadVisualize
BU of 6h6g by Molmil
Crystal Structure of TcdB2-TccC3 without hypervariable C-terminal region
Descriptor: TcdB2,TccC3
Authors:Gatsogiannis, C, Merino, F, Roderer, D, Balchin, D, Schubert, E, Kuhlee, A, Hayer-Hartl, M, Raunser, S.
Deposit date:2018-07-27
Release date:2018-10-03
Last modified:2024-01-17
Method:X-RAY DIFFRACTION (3.004 Å)
Cite:Tc toxin activation requires unfolding and refolding of a beta-propeller.
Nature, 563, 2018
7AG5
DownloadVisualize
BU of 7ag5 by Molmil
Structure of the Laspartomycin C double mutant G4D D-allo-Thr9D-Dap in complex with Geranyl phosphate
Descriptor: (~{E})-13-methyltetradec-2-enoic acid, CALCIUM ION, Geranyl phosphate, ...
Authors:Zeronian, M.R, Pearce, N.M, Wood, T.M, Martin, N.I, Janssen, B.J.C.
Deposit date:2020-09-21
Release date:2022-02-02
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.04 Å)
Cite:Mechanistic insights into the C55-P targeting lipopeptide antibiotics revealed by structure-activity studies and high-resolution crystal structures
Chem Sci, 13, 2022
6HKJ
DownloadVisualize
BU of 6hkj by Molmil
X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a inhibitor RNA 2-19-1
Descriptor: (2~{S})-2-[[(2~{S})-6-[(6-fluoranylpyridin-3-yl)amino]-1-oxidanyl-1,6-bis(oxidanylidene)hexan-2-yl]carbamoylamino]pentanedioic acid, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
Authors:Motlova, L, Novakova, Z, Barinka, C.
Deposit date:2018-09-06
Release date:2018-12-05
Last modified:2024-10-23
Method:X-RAY DIFFRACTION (2.09 Å)
Cite:2-Aminoadipic Acid-C(O)-Glutamate Based Prostate-Specific Membrane Antigen Ligands for Potential Use as Theranostics.
ACS Med Chem Lett, 9, 2018
6OGH
DownloadVisualize
BU of 6ogh by Molmil
Structure of Aedes aegypti OBP22 in the complex with linoleic acid
Descriptor: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, AAEL005772-PA, CADMIUM ION, ...
Authors:Jones, D.N, Wang, J.
Deposit date:2019-04-02
Release date:2019-04-24
Last modified:2024-11-13
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Aedes aegypti Odorant Binding Protein 22 selectively binds fatty acids through a conformational change in its C-terminal tail.
Sci Rep, 10, 2020
8ENJ
DownloadVisualize
BU of 8enj by Molmil
Design, synthesis, biological evaluation, and X-ray crystallography of diarylpyrazole derivatives possessing terminal arylsulfonamide moieties as anti-proliferative agents targeting c-Jun N-terminal kinase (JNK)
Descriptor: Mitogen-activated protein kinase 10, N-[3-({(4P)-4-[(3M)-1-tert-butyl-3-(3-hydroxyphenyl)-1H-pyrazol-4-yl]pyridin-2-yl}amino)propyl]-4-hydroxybenzene-1-sulfonamide
Authors:Park, H, Mersal, K.I.
Deposit date:2022-09-30
Release date:2023-10-18
Method:X-RAY DIFFRACTION (2.81 Å)
Cite:Evaluation of novel pyrazol-4-yl pyridine derivatives possessing arylsulfonamide tethers as c-Jun N-terminal kinase (JNK) inhibitors in leukemia cells.
Eur.J.Med.Chem., 261, 2023
8V80
DownloadVisualize
BU of 8v80 by Molmil
Alpha7-nicotinic acetylcholine receptor bound to epibatidine and (-)-TQS
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, (3aR,4S,9bS)-4-(naphthalen-1-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide, (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, ...
Authors:Burke, S.M, Noviello, C.M, Hibbs, R.E.
Deposit date:2023-12-04
Release date:2024-02-21
Last modified:2025-05-21
Method:ELECTRON MICROSCOPY (2.34 Å)
Cite:Structural mechanisms of alpha 7 nicotinic receptor allosteric modulation and activation.
Cell, 187, 2024
8V88
DownloadVisualize
BU of 8v88 by Molmil
Alpha7-nicotinic acetylcholine receptor bound to epibatidine and GAT107
Descriptor: (2S)-3-(hexadecanoyloxy)-2-[(9Z)-octadec-9-enoyloxy]propyl 2-(trimethylammonio)ethyl phosphate, (3aR,4S,9bS)-4-(4-bromophenyl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinoline-8-sulfonamide, (3beta,14beta,17beta,25R)-3-[4-methoxy-3-(methoxymethyl)butoxy]spirost-5-en, ...
Authors:Burke, S.M, Noviello, C.M, Hibbs, R.E.
Deposit date:2023-12-05
Release date:2024-02-21
Last modified:2025-05-14
Method:ELECTRON MICROSCOPY (2.3 Å)
Cite:Structural mechanisms of alpha 7 nicotinic receptor allosteric modulation and activation.
Cell, 187, 2024

238895

數據於2025-07-16公開中

PDB statisticsPDBj update infoContact PDBjnumon