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PDB: 2 results

4LL3
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BU of 4ll3 by Molmil
Structure of wild-type HIV protease in complex with darunavir
Descriptor: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, Protease
Authors:Grantz Saskova, K, Rezacova, P, Brynda, J, Kozisek, M, Konvalinka, J.
Deposit date:2013-07-09
Release date:2014-04-16
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Thermodynamic and structural analysis of HIV protease resistance to darunavir - analysis of heavily mutated patient-derived HIV-1 proteases.
Febs J., 281, 2014
3TTP
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BU of 3ttp by Molmil
Structure of multiresistant HIV-1 protease in complex with darunavir
Descriptor: (3R,3AS,6AR)-HEXAHYDROFURO[2,3-B]FURAN-3-YL(1S,2R)-3-[[(4-AMINOPHENYL)SULFONYL](ISOBUTYL)AMINO]-1-BENZYL-2-HYDROXYPROPYLCARBAMATE, BETA-MERCAPTOETHANOL, CHLORIDE ION, ...
Authors:Saskova, K.G, Brynda, J, Kozisek, M, Konvalinka, J, Rezacova, P.
Deposit date:2011-09-15
Release date:2012-09-26
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.23 Å)
Cite:Thermodynamic and structural analysis of HIV protease resistance to darunavir - analysis of heavily mutated patient-derived HIV-1 proteases.
Febs J., 281, 2014

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數據於2024-07-17公開中

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