7FR8
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![BU of 7fr8 by Molmil](/molmil-images/mine/7fr8) | |
7FRC
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![BU of 7frc by Molmil](/molmil-images/mine/7frc) | |
7FR0
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![BU of 7fr0 by Molmil](/molmil-images/mine/7fr0) | |
7FR6
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![BU of 7fr6 by Molmil](/molmil-images/mine/7fr6) | |
7FR2
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![BU of 7fr2 by Molmil](/molmil-images/mine/7fr2) | |
7FR9
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![BU of 7fr9 by Molmil](/molmil-images/mine/7fr9) | |
7FRA
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![BU of 7fra by Molmil](/molmil-images/mine/7fra) | |
7FRD
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![BU of 7frd by Molmil](/molmil-images/mine/7frd) | |
7FR4
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![BU of 7fr4 by Molmil](/molmil-images/mine/7fr4) | |
7FRB
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![BU of 7frb by Molmil](/molmil-images/mine/7frb) | |
7FR1
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![BU of 7fr1 by Molmil](/molmil-images/mine/7fr1) | |
7FR3
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![BU of 7fr3 by Molmil](/molmil-images/mine/7fr3) | |
7FR5
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![BU of 7fr5 by Molmil](/molmil-images/mine/7fr5) | |
7FR7
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![BU of 7fr7 by Molmil](/molmil-images/mine/7fr7) | |
7WR6
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![BU of 7wr6 by Molmil](/molmil-images/mine/7wr6) | Crystal structure of ADP-riboxanated caspase-4 in complex with Af1521 | Descriptor: | ADP-ribose glycohydrolase AF_1521, Caspase-4, [[(3~{a}~{S},5~{R},6~{R},6~{a}~{R})-2-azanylidene-3-[(4~{R})-4-azanyl-5-oxidanylidene-pentyl]-6-oxidanyl-3~{a},5,6,6~{a}-tetrahydrofuro[2,3-d][1,3]oxazol-5-yl]methoxy-oxidanyl-phosphoryl] [(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl hydrogen phosphate | Authors: | Hou, Y.J, Zeng, H, Shao, F, Ding, J. | Deposit date: | 2022-01-26 | Release date: | 2023-01-25 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (1.96 Å) | Cite: | Structural mechanisms of calmodulin activation of Shigella effector OspC3 to ADP-riboxanate caspase-4/11 and block pyroptosis. Nat.Struct.Mol.Biol., 30, 2023
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8C1A
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![BU of 8c1a by Molmil](/molmil-images/mine/8c1a) | |
8C19
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![BU of 8c19 by Molmil](/molmil-images/mine/8c19) | SARS-CoV-2 NSP3 macrodomain in complex with 1-methyl-4-[5-(morpholin-4-ylcarbonyl)-2-furyl]-1H-pyrrolo[2,3-b]pyridine | Descriptor: | 1,2-ETHANEDIOL, Non-structural protein 3, [5-(1-methylpyrrolo[2,3-b]pyridin-4-yl)furan-2-yl]-morpholin-4-yl-methanone | Authors: | Schuller, M, Ahel, I. | Deposit date: | 2022-12-20 | Release date: | 2023-03-08 | Method: | X-RAY DIFFRACTION (1.95 Å) | Cite: | Discovery and Development Strategies for SARS-CoV-2 NSP3 Macrodomain Inhibitors. Pathogens, 12, 2023
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8GIA
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![BU of 8gia by Molmil](/molmil-images/mine/8gia) | Crystal structure of SARS-CoV-2 (Covid-19) Nsp3 macrodomain in complex with TFMU-ADPr | Descriptor: | Non-structural protein 3, [(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl [(2R,3S,4R,5R)-3,4-dihydroxy-5-{[2-oxo-4-(trifluoromethyl)-2H-1-benzopyran-7-yl]oxy}oxolan-2-yl]methyl dihydrogen diphosphate | Authors: | Wallace, S.D, Bagde, S.R, Fromme, J.C. | Deposit date: | 2023-03-13 | Release date: | 2023-05-17 | Last modified: | 2023-10-25 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | A Fluorescence Polarization Assay for Macrodomains Facilitates the Identification of Potent Inhibitors of the SARS-CoV-2 Macrodomain. Acs Chem.Biol., 18, 2023
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8AZD
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![BU of 8azd by Molmil](/molmil-images/mine/8azd) | |
8AZC
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![BU of 8azc by Molmil](/molmil-images/mine/8azc) | |
8P0C
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![BU of 8p0c by Molmil](/molmil-images/mine/8p0c) | Rubella virus p150 macro domain (apo) | Descriptor: | Non-structural polyprotein p200 | Authors: | Stoll, G.A, Modis, Y. | Deposit date: | 2023-05-10 | Release date: | 2024-01-17 | Last modified: | 2024-03-06 | Method: | X-RAY DIFFRACTION (1.72 Å) | Cite: | Crystal structure and biochemical activity of the macrodomain from rubella virus p150. J.Virol., 98, 2024
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8P0E
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![BU of 8p0e by Molmil](/molmil-images/mine/8p0e) | |
8CB3
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![BU of 8cb3 by Molmil](/molmil-images/mine/8cb3) | SARS-CoV Macro domain complexed with 3-(N-morpholino)propanesulfonic acid | Descriptor: | 3[N-MORPHOLINO]PROPANE SULFONIC ACID, GLYCEROL, Papain-like protease nsp3 | Authors: | Morin, B, Ferron, F, Coutard, B, Canard, B, Marseilles Structural Genomics Program @ AFMB (MSGP) | Deposit date: | 2023-01-25 | Release date: | 2024-02-07 | Method: | X-RAY DIFFRACTION (1.572 Å) | Cite: | SARS-CoV Macro domain complexed with 3-(N-morpholino)propanesulfonic acid To Be Published
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8AZM
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![BU of 8azm by Molmil](/molmil-images/mine/8azm) | |
8AZI
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![BU of 8azi by Molmil](/molmil-images/mine/8azi) | |