8INR
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![BU of 8inr by Molmil](/molmil-images/mine/8inr) | Cryo-EM structure of the alpha-MSH-bound human melanocortin receptor 5 (MC5R)-Gs complex | Descriptor: | CALCIUM ION, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, Guanine nucleotide-binding protein G(I)/G(S)/G(T) subunit beta-1,HiBiT, ... | Authors: | Feng, W.B, Zhou, Q.T, Chen, X.Y, Dai, A.T, Cai, X.Q, Liu, X, Zhao, F.H, Chen, Y, Ye, C.Y, Xu, Y.N, Cong, Z.T, Li, H, Lin, S, Yang, D.H, Wang, M.W. | Deposit date: | 2023-03-10 | Release date: | 2023-09-20 | Method: | ELECTRON MICROSCOPY (2.73 Å) | Cite: | Structural insights into ligand recognition and subtype selectivity of the human melanocortin-3 and melanocortin-5 receptors. Cell Discov, 9, 2023
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8INP
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![BU of 8inp by Molmil](/molmil-images/mine/8inp) | A reversible glycosyltransferase of tectorigenin - Bc7OUGT | Descriptor: | Bc7OUGT, URIDINE-5'-DIPHOSPHATE, beta-D-glucopyranose | Authors: | Zhang, Z.Y, Lu, L, Guan, Z.F, Cheng, W.J. | Deposit date: | 2023-03-10 | Release date: | 2023-08-23 | Last modified: | 2023-11-29 | Method: | X-RAY DIFFRACTION (2.12 Å) | Cite: | Functional characterization and structural basis of a reversible glycosyltransferase involves in plant chemical defence. Plant Biotechnol J, 21, 2023
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8INO
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![BU of 8ino by Molmil](/molmil-images/mine/8ino) | Crystal structure of UGT74AN3 in complex UDP and PER | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3-[(3S,5S,8S,9S,10R,13R,14S,17R)-10,13-dimethyl-3,5,14-tris(oxidanyl)-2,3,4,6,7,8,9,11,12,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]-2H-furan-5-one, Glycosyltransferase, ... | Authors: | Long, F, Huang, W. | Deposit date: | 2023-03-10 | Release date: | 2024-01-24 | Method: | X-RAY DIFFRACTION (2.3 Å) | Cite: | Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3 Acs Catalysis, 14, 2024
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8INL
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![BU of 8inl by Molmil](/molmil-images/mine/8inl) | LSD1 in complex with S2172 | Descriptor: | 3-[3,5-bis(fluoranyl)-2-phenylmethoxy-phenyl]propanal, FLAVIN-ADENINE DINUCLEOTIDE, GLYCEROL, ... | Authors: | Niwa, H, Sato, S, Umehara, T. | Deposit date: | 2023-03-10 | Release date: | 2024-03-13 | Method: | X-RAY DIFFRACTION (2.62 Å) | Cite: | LSD1 in complex with S2172 To Be Published
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8INJ
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![BU of 8inj by Molmil](/molmil-images/mine/8inj) | Crystal structure of UGT74AN3-UDP-DIG | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, DIGITOXIGENIN, Glycosyltransferase, ... | Authors: | Feng, L, Wei, H. | Deposit date: | 2023-03-10 | Release date: | 2024-02-14 | Method: | X-RAY DIFFRACTION (1.76 Å) | Cite: | Crystal structure of UGT74AN3-UDP-DIG To Be Published
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8IND
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![BU of 8ind by Molmil](/molmil-images/mine/8ind) | Crystal structure of UGT74AN3-UDP-RES | Descriptor: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 5-[(1R,2S,4R,6R,7R,10S,11S,14S,16R)-14-hydroxy-7,11-dimethyl-3-oxapentacyclo[8.8.0.02,4.02,7.011,16]octadecan-6-yl]pyran-2-one, Glycosyltransferase, ... | Authors: | Huang, W. | Deposit date: | 2023-03-09 | Release date: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.85 Å) | Cite: | Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3 Acs Catalysis, 14, 2024
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8INA
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![BU of 8ina by Molmil](/molmil-images/mine/8ina) | Crystal structure of UGT74AN3-UDP | Descriptor: | GLYCEROL, Glycosyltransferase, URIDINE-5'-DIPHOSPHATE | Authors: | Long, F, Huang, W. | Deposit date: | 2023-03-09 | Release date: | 2024-01-24 | Method: | X-RAY DIFFRACTION (1.86 Å) | Cite: | Substrate Promiscuity, Crystal Structure, and Application of a Plant UDP-Glycosyltransferase UGT74AN3 Acs Catalysis, 14, 2024
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8IN9
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![BU of 8in9 by Molmil](/molmil-images/mine/8in9) | The structure of the GfsA KSQ-AT didomain in complex with the GfsA ACP domain | Descriptor: | N-[2-(acetylamino)ethyl]-N~3~-[(2R)-2-hydroxy-3,3-dimethyl-4-(phosphonooxy)butanoyl]-beta-alaninamide, Polyketide synthase | Authors: | Chisuga, T, Murakami, S, Miyanaga, A, Kudo, F, Eguchi, T. | Deposit date: | 2023-03-09 | Release date: | 2023-05-31 | Last modified: | 2023-06-28 | Method: | X-RAY DIFFRACTION (3.4 Å) | Cite: | Structure-Based Analysis of Transient Interactions between Ketosynthase-like Decarboxylase and Acyl Carrier Protein in a Loading Module of Modular Polyketide Synthase. Acs Chem.Biol., 18, 2023
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8IN6
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![BU of 8in6 by Molmil](/molmil-images/mine/8in6) | Eisenia hydrolysis-enhancing protein from Aplysia kurodai complex with tannic acid | Descriptor: | 25 kDa polyphenol-binding protein, BETA-1,2,3,4,6-PENTA-O-GALLOYL-D-GLUCOPYRANOSE | Authors: | Sun, X.M, Ye, Y.X, Kato, K, Yu, J, Yao, M. | Deposit date: | 2023-03-08 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.9 Å) | Cite: | Structural basis of EHEP-mediated offense against phlorotannin-induced defense from brown algae to protect aku BGL activity. Elife, 12, 2023
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8IN4
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![BU of 8in4 by Molmil](/molmil-images/mine/8in4) | Eisenia hydrolysis-enhancing protein from Aplysia kurodai | Descriptor: | 25 kDa polyphenol-binding protein, ACETYL GROUP, GLYCEROL | Authors: | Sun, X.M, Ye, Y.X, Kato, K, Yu, J, Yao, M. | Deposit date: | 2023-03-08 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.4 Å) | Cite: | Structural basis of EHEP-mediated offense against phlorotannin-induced defense from brown algae to protect aku BGL activity. Elife, 12, 2023
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8IN3
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![BU of 8in3 by Molmil](/molmil-images/mine/8in3) | Eisenia hydrolysis-enhancing protein from Aplysia kurodai | Descriptor: | 25 kDa polyphenol-binding protein, GLYCEROL | Authors: | Sun, X.M, Ye, Y.X, Kato, K, Yu, J, Yao, M. | Deposit date: | 2023-03-08 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (1.15 Å) | Cite: | Structural basis of EHEP-mediated offense against phlorotannin-induced defense from brown algae to protect aku BGL activity. Elife, 12, 2023
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8IN1
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![BU of 8in1 by Molmil](/molmil-images/mine/8in1) | beta-glucosidase protein from Aplysia kurodai | Descriptor: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Beta-Glucosidase, alpha-L-fucopyranose-(1-3)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Sun, X.M, Ye, Y.X, Kato, K, Yu, J, Yao, M. | Deposit date: | 2023-03-08 | Release date: | 2023-11-15 | Method: | X-RAY DIFFRACTION (2.7 Å) | Cite: | Structural basis of EHEP-mediated offense against phlorotannin-induced defense from brown algae to protect aku BGL activity. Elife, 12, 2023
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8IMY
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![BU of 8imy by Molmil](/molmil-images/mine/8imy) | Cryo-EM structure of GPI-T (inactive mutant) with GPI and proULBP2, a proprotein substrate | Descriptor: | 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Li, T, Xu, Y, Qu, Q, Li, D. | Deposit date: | 2023-03-07 | Release date: | 2023-08-16 | Last modified: | 2023-11-01 | Method: | ELECTRON MICROSCOPY (3.22 Å) | Cite: | Structures of liganded glycosylphosphatidylinositol transamidase illuminate GPI-AP biogenesis. Nat Commun, 14, 2023
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8IMX
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![BU of 8imx by Molmil](/molmil-images/mine/8imx) | Cryo-EM structure of GPI-T with a chimeric GPI-anchored protein | Descriptor: | 1-palmitoyl-2-oleoyl-sn-glycero-3-phosphocholine, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | Authors: | Xu, Y, Li, T, Qu, Q, Li, D. | Deposit date: | 2023-03-07 | Release date: | 2023-08-16 | Last modified: | 2023-11-01 | Method: | ELECTRON MICROSCOPY (2.85 Å) | Cite: | Structures of liganded glycosylphosphatidylinositol transamidase illuminate GPI-AP biogenesis. Nat Commun, 14, 2023
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8IMU
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![BU of 8imu by Molmil](/molmil-images/mine/8imu) | Dihydroxyacid dehydratase (DHAD) mutant-V497F | Descriptor: | ACETATE ION, Dihydroxy-acid dehydratase, chloroplastic, ... | Authors: | Zhou, J, Zang, X, Tang, Y, Yan, Y. | Deposit date: | 2023-03-07 | Release date: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.93 Å) | Cite: | Dihydroxyacid dehydratase (DHAD) mutant-V497F To Be Published
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8IMR
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![BU of 8imr by Molmil](/molmil-images/mine/8imr) | Structure of ligand-free human macrophage migration inhibitory factor | Descriptor: | 1,2-ETHANEDIOL, ISOPROPYL ALCOHOL, Macrophage migration inhibitory factor, ... | Authors: | Sugishima, K, Noguchi, K, Yohda, M, Odaka, M, Matsumura, H. | Deposit date: | 2023-03-07 | Release date: | 2024-03-13 | Method: | X-RAY DIFFRACTION (1.3 Å) | Cite: | Identification of methotrexate as an inhibitor of macrophage migration inhibitory factor by high-resolution crystal structure analysis To Be Published
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8IMO
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![BU of 8imo by Molmil](/molmil-images/mine/8imo) | Rt1'I-Rt1'II, Rt2I-Rt2II, Rt3'I-Rt3'II cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster G) | Descriptor: | CpcA, CpcB, CpcD, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (3.08 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMN
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![BU of 8imn by Molmil](/molmil-images/mine/8imn) | Rt1I-Rt1II, Rt2'I-Rt2'II, Rt3I-Rt3II cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster F) | Descriptor: | CpcA, CpcB, CpcD, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (3.07 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMM
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![BU of 8imm by Molmil](/molmil-images/mine/8imm) | Rs2'I-Rs2'II, Rs1'I-Rs1'II, Rb'I-Rb'II cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster E) | Descriptor: | CpcA, CpcB, CpcD, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.76 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IML
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![BU of 8iml by Molmil](/molmil-images/mine/8iml) | Rs2I-Rs2II, Rs1I-Rs1II, RbI-RbII cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster D) | Descriptor: | CpcA, CpcB, CpcD, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.74 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMK
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![BU of 8imk by Molmil](/molmil-images/mine/8imk) | D3-D4, D1-D2, D'3-D'4, D'1-D'2 cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster C) | Descriptor: | ApcA1, ApcA2, ApcB1, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.48 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMJ
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![BU of 8imj by Molmil](/molmil-images/mine/8imj) | A'1-A'2, A'3-A'4, B1-B2, C1-C2 cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster B) | Descriptor: | ApcA2, ApcB2, ApcB3, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.59 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMI
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![BU of 8imi by Molmil](/molmil-images/mine/8imi) | A1-A2, A3-A4, B'1-B'2, C'1-C'2 cylinder in cyanobacterial phycobilisome from Anthocerotibacter panamensis (Cluster A) | Descriptor: | ApcA2, ApcB2, ApcB3, ... | Authors: | Wang, C.H, Yang, C.H, Wu, H.Y, Jiang, H.W, Ho, M.C, Ho, M.Y. | Deposit date: | 2023-03-07 | Release date: | 2023-10-25 | Last modified: | 2024-05-08 | Method: | ELECTRON MICROSCOPY (2.59 Å) | Cite: | A structure of the relict phycobilisome from a thylakoid-free cyanobacterium. Nat Commun, 14, 2023
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8IMG
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![BU of 8img by Molmil](/molmil-images/mine/8img) | Human cGAS catalytic domain bound with C20 | Descriptor: | 2-[2-hydroxy-2-oxoethyl-[3-(7-methoxy-4-methyl-2-oxidanylidene-chromen-3-yl)propanoyl]amino]ethanoic acid, Cyclic GMP-AMP synthase, ZINC ION | Authors: | Zhao, W.F, Li, J.M, Xu, Y.C. | Deposit date: | 2023-03-06 | Release date: | 2024-01-03 | Method: | X-RAY DIFFRACTION (1.8 Å) | Cite: | Discovery of novel cGAS inhibitors based on natural flavonoids. Bioorg.Chem., 140, 2023
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8IMD
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![BU of 8imd by Molmil](/molmil-images/mine/8imd) | Crystal structure of Cu/Zn Superoxide dismutase from Paenibacillus lautus | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, COPPER (II) ION, Cu/Zn-Superoxide dismutase, ... | Authors: | Narikiyo, S, Furukawa, Y, Akutsu, M. | Deposit date: | 2023-03-06 | Release date: | 2024-01-17 | Method: | X-RAY DIFFRACTION (1.45 Å) | Cite: | Characterization of a novel cysteine-less Cu/Zn-superoxide dismutase in Paenibacillus lautus missing a conserved disulfide bond. J.Biol.Chem., 299, 2023
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