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PDB: 3 results

6CQE
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BU of 6cqe by Molmil
Crystal structure of HPK1 kinase domain S171A mutant
Descriptor: Mitogen-activated protein kinase kinase kinase kinase 1
Authors:Wu, P, Lehoux, I, Mortara, K, Franke, Y, Wang, W.
Deposit date:2018-03-15
Release date:2018-12-19
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (1.886 Å)
Cite:Hematopoietic Progenitor Kinase-1 Structure in a Domain-Swapped Dimer.
Structure, 27, 2019
6CQF
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BU of 6cqf by Molmil
Crystal structure of HPK1 in complex an inhibitor G1858
Descriptor: Mitogen-activated protein kinase kinase kinase kinase 1, N-{2-(3,3-difluoropyrrolidin-1-yl)-6-[(3R)-pyrrolidin-3-yl]pyrimidin-4-yl}-1-(propan-2-yl)-1H-pyrazolo[4,3-c]pyridin-6-amine
Authors:Wu, P, Lehoux, I, Mortara, K, Franke, Y, Chan, B.K, Wang, W.
Deposit date:2018-03-15
Release date:2018-12-19
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.246 Å)
Cite:Hematopoietic Progenitor Kinase-1 Structure in a Domain-Swapped Dimer.
Structure, 27, 2019
6CQD
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BU of 6cqd by Molmil
Crystal structure of HPK1 in complex with ATP analogue (AMPPNP)
Descriptor: MAGNESIUM ION, Mitogen-activated protein kinase kinase kinase kinase 1, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
Authors:Wu, P, Lehoux, I, Franke, Y, Mortara, K, Wang, W.
Deposit date:2018-03-14
Release date:2018-12-19
Last modified:2024-03-13
Method:X-RAY DIFFRACTION (2.12 Å)
Cite:Hematopoietic Progenitor Kinase-1 Structure in a Domain-Swapped Dimer.
Structure, 27, 2019

222624

数据于2024-07-17公开中

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