8U69
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![BU of 8u69 by Molmil](/molmil-images/mine/8u69) | Crystal Structure of HIV-1 Reverse Transcriptase in Complex with 3-chloro-5-(4-chloro-2-(2-(5-chloro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)ethoxy)phenoxy)benzonitrile (JLJ334), a non-nucleoside inhibitor | Descriptor: | 3-chloro-5-{4-chloro-2-[2-(5-chloro-2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)ethoxy]phenoxy}benzonitrile, Reverse transcriptase/ribonuclease H, p51 RT | Authors: | Hollander, K, Carter, Z, Jorgensen, W.L, Anderson, K.S. | Deposit date: | 2023-09-13 | Release date: | 2023-11-08 | Method: | X-RAY DIFFRACTION (2.45 Å) | Cite: | Covalent and noncovalent strategies for targeting Lys102 in HIV-1 reverse transcriptase. Eur.J.Med.Chem., 262, 2023
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8U66
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![BU of 8u66 by Molmil](/molmil-images/mine/8u66) | Firmicutes Rubisco | Descriptor: | 2-CARBOXYARABINITOL-1,5-DIPHOSPHATE, MAGNESIUM ION, Rubisco | Authors: | Kaeser, B.P, Liu, A.K, Shih, P.M. | Deposit date: | 2023-09-13 | Release date: | 2023-11-22 | Last modified: | 2023-12-27 | Method: | ELECTRON MICROSCOPY (2.21 Å) | Cite: | Deep-branching evolutionary intermediates reveal structural origins of form I rubisco. Curr.Biol., 33, 2023
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8U61
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![BU of 8u61 by Molmil](/molmil-images/mine/8u61) | Human RADX tetramer bound to ssDNA | Descriptor: | RPA-related protein RADX, dT25 DNA (25-MER) | Authors: | Balakrishnan, S, Chazin, W.J. | Deposit date: | 2023-09-13 | Release date: | 2024-01-31 | Last modified: | 2024-03-27 | Method: | ELECTRON MICROSCOPY (4 Å) | Cite: | Structure of RADX and mechanism for regulation of RAD51 nucleofilaments. Proc.Natl.Acad.Sci.USA, 121, 2024
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8U60
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![BU of 8u60 by Molmil](/molmil-images/mine/8u60) | |
8U5Z
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![BU of 8u5z by Molmil](/molmil-images/mine/8u5z) | Structure of Mango II variant aptamer bound to T01-7M-B | Descriptor: | 2-[(E)-(1,7-dimethylquinolin-4(1H)-ylidene)methyl]-3-{2,16-dioxo-20-[(3aR,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-6,9,12-trioxa-3,15-diazaicosan-1-yl}-1,3-benzothiazol-3-ium, Mango II variant, POTASSIUM ION, ... | Authors: | Passalacqua, L.F.M, Ferre-D'Amare, A.R. | Deposit date: | 2023-09-13 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (2.5 Å) | Cite: | Structure of Mango II variant aptamer bound to T01-7M-B To Be Published
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8U5Y
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![BU of 8u5y by Molmil](/molmil-images/mine/8u5y) | human RADX trimer bound to ssDNA | Descriptor: | DNA (25-MER), RPA-related protein RADX | Authors: | Balakrishnan, S, Chazin, W.J. | Deposit date: | 2023-09-13 | Release date: | 2023-10-11 | Last modified: | 2023-10-18 | Method: | ELECTRON MICROSCOPY (3.01 Å) | Cite: | Structure of RADX and mechanism for regulation of RAD51 nucleofilaments. Biorxiv, 2023
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8U5T
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![BU of 8u5t by Molmil](/molmil-images/mine/8u5t) | Structure of Mango II variant aptamer bound to T01-6A-B | Descriptor: | 3-{2,16-dioxo-20-[(3aS,4R,6aS)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-6,9,12-trioxa-3,15-diazaicosan-1-yl}-2-{(E)-[6-(4-methoxyphenyl)-1-methylquinolin-4(1H)-ylidene]methyl}-1,3-benzothiazol-3-ium, Mango II variant, POTASSIUM ION, ... | Authors: | Passalacqua, L.F.M, Ferre-D'Amare, A.R. | Deposit date: | 2023-09-12 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (2.2 Å) | Cite: | Structure of Mango II variant aptamer bound to T01-6A-B To Be Published
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8U5R
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![BU of 8u5r by Molmil](/molmil-images/mine/8u5r) | |
8U5P
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![BU of 8u5p by Molmil](/molmil-images/mine/8u5p) | Structure of Mango II aptamer bound to T01-6A-B | Descriptor: | 3-[2,16-dioxo-20-(2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)-6,9,12-trioxa-3,15-diazaicosan-1-yl]-2-{(E)-[6-(4-methoxyphenyl)-1-methylquinolin-4(1H)-ylidene]methyl}-1,3-benzothiazol-3-ium, Mango II, POTASSIUM ION | Authors: | Passalacqua, L.F.M, Ferre-D'Amare, A.R. | Deposit date: | 2023-09-12 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (2.9 Å) | Cite: | Structure of Mango II aptamer bound to T01-6A-B To Be Published
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8U5M
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![BU of 8u5m by Molmil](/molmil-images/mine/8u5m) | Structure of Sts-1 HP domain with rebamipide | Descriptor: | Rebamipide, Ubiquitin-associated and SH3 domain-containing protein B | Authors: | Azia, F, Dey, R, French, J.B. | Deposit date: | 2023-09-12 | Release date: | 2024-02-07 | Last modified: | 2024-02-21 | Method: | X-RAY DIFFRACTION (2.46 Å) | Cite: | Rebamipide and Derivatives are Potent, Selective Inhibitors of Histidine Phosphatase Activity of the Suppressor of T Cell Receptor Signaling Proteins. J.Med.Chem., 67, 2024
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8U5K
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![BU of 8u5k by Molmil](/molmil-images/mine/8u5k) | |
8U5J
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![BU of 8u5j by Molmil](/molmil-images/mine/8u5j) | Structure of Mango III variant aptamer bound to T01-07M-B | Descriptor: | 2-[(E)-(1,7-dimethylquinolin-4(1H)-ylidene)methyl]-3-{2,16-dioxo-20-[(3aR,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]-6,9,12-trioxa-3,15-diazaicosan-1-yl}-1,3-benzothiazol-3-ium, DIMETHYL SULFOXIDE, Mango III variant, ... | Authors: | Passalacqua, L.F.M, Ferre-D'Amare, A.R. | Deposit date: | 2023-09-12 | Release date: | 2024-03-27 | Method: | X-RAY DIFFRACTION (1.7 Å) | Cite: | Structure of Mango III variant aptamer bound to T01-07M-B To Be Published
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8U5H
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![BU of 8u5h by Molmil](/molmil-images/mine/8u5h) | |
8U5G
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![BU of 8u5g by Molmil](/molmil-images/mine/8u5g) | Crystal structure of the co-expressed SDS22:PP1:I3 complex | Descriptor: | E3 ubiquitin-protein ligase PPP1R11, FE (III) ION, PHOSPHATE ION, ... | Authors: | Choy, M.S, Peti, W, Page, R. | Deposit date: | 2023-09-12 | Release date: | 2023-12-06 | Last modified: | 2024-01-03 | Method: | X-RAY DIFFRACTION (3.2 Å) | Cite: | The SDS22:PP1:I3 complex: SDS22 binding to PP1 loosens the active site metal to prime metal exchange. J.Biol.Chem., 300, 2023
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8U5F
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![BU of 8u5f by Molmil](/molmil-images/mine/8u5f) | Crystal Structure of Trypsinized Clostridium perfringens Enterotoxin | Descriptor: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLYCEROL, Heat-labile enterotoxin B chain, ... | Authors: | Kapoor, S, Ogbu, C.P, Vecchio, A.J. | Deposit date: | 2023-09-12 | Release date: | 2023-09-27 | Last modified: | 2023-12-20 | Method: | X-RAY DIFFRACTION (2.32 Å) | Cite: | Structural Basis of Clostridium perfringens Enterotoxin Activation and Oligomerization by Trypsin. Toxins, 15, 2023
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8U5E
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![BU of 8u5e by Molmil](/molmil-images/mine/8u5e) | |
8U5D
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![BU of 8u5d by Molmil](/molmil-images/mine/8u5d) | |
8U5B
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![BU of 8u5b by Molmil](/molmil-images/mine/8u5b) | |
8U5A
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![BU of 8u5a by Molmil](/molmil-images/mine/8u5a) | Improving protein expression, stability, and function with ProteinMPNN | Descriptor: | Designed myoglobin, PROTOPORPHYRIN IX CONTAINING FE | Authors: | Kalvet, I, Bera, A.K, Baker, D. | Deposit date: | 2023-09-12 | Release date: | 2024-01-17 | Last modified: | 2024-01-31 | Method: | X-RAY DIFFRACTION (2 Å) | Cite: | Improving Protein Expression, Stability, and Function with ProteinMPNN. J.Am.Chem.Soc., 146, 2024
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8U55
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![BU of 8u55 by Molmil](/molmil-images/mine/8u55) | |
8U53
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![BU of 8u53 by Molmil](/molmil-images/mine/8u53) | Mechanically activated ion channel OSCA3.1 in nanodiscs | Descriptor: | 1-PALMITOYL-2-LINOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, CSC1-like protein ERD4, PALMITIC ACID, ... | Authors: | Jojoa-Cruz, S, Lee, W.H, Ward, A.B. | Deposit date: | 2023-09-12 | Release date: | 2024-06-05 | Method: | ELECTRON MICROSCOPY (2.6 Å) | Cite: | Structure-guided mutagenesis of OSCAs reveals differential activation to mechanical stimuli. Elife, 12, 2024
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8U51
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![BU of 8u51 by Molmil](/molmil-images/mine/8u51) | |
8U50
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![BU of 8u50 by Molmil](/molmil-images/mine/8u50) | |
8U4Z
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![BU of 8u4z by Molmil](/molmil-images/mine/8u4z) | |
8U4W
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![BU of 8u4w by Molmil](/molmil-images/mine/8u4w) | |