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PDB: 5 results

5L1H
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BU of 5l1h by Molmil
AMPA subtype ionotropic glutamate receptor GluA2 in complex with noncompetitive inhibitor GYKI53655
Descriptor: (8R)-5-(4-aminophenyl)-N,8-dimethyl-8,9-dihydro-2H,7H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-7-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2
Authors:Yelshanskaya, M.V, Singh, A.K, Sampson, J.M, Sobolevsky, A.I.
Deposit date:2016-07-29
Release date:2016-10-19
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (3.801 Å)
Cite:Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Neuron, 91, 2016
5L1B
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BU of 5l1b by Molmil
AMPA subtype ionotropic glutamate receptor GluA2 in Apo state
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2,Glutamate receptor 2
Authors:Yelshanskaya, M.V, Singh, A.K, Sampson, J.M, Sobolevsky, A.I.
Deposit date:2016-07-28
Release date:2016-10-19
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (4 Å)
Cite:Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Neuron, 91, 2016
5L1G
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BU of 5l1g by Molmil
AMPA subtype ionotropic glutamate receptor GluA2 in complex with GYKI-Br
Descriptor: (8R)-5-(4-amino-3-bromophenyl)-N,8-dimethyl-8,9-dihydro-2H,7H-[1,3]dioxolo[4,5-h][2,3]benzodiazepine-7-carboxamide, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2
Authors:Yelshanskaya, M.V, Singh, A.K, Sampson, J.M, Sobolevsky, A.I.
Deposit date:2016-07-29
Release date:2016-10-19
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (4.507 Å)
Cite:Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Neuron, 91, 2016
5L1F
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BU of 5l1f by Molmil
AMPA subtype ionotropic glutamate receptor GluA2 in complex with noncompetitive inhibitor Perampanel
Descriptor: 2-(6'-oxo-1'-phenyl[1',6'-dihydro[2,3'-bipyridine]]-5'-yl)benzonitrile, 2-acetamido-2-deoxy-beta-D-glucopyranose, Glutamate receptor 2
Authors:Yelshanskaya, M.V, Singh, A.K, Sampson, J.M, Sobolevsky, A.I.
Deposit date:2016-07-29
Release date:2016-10-19
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (4 Å)
Cite:Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Neuron, 91, 2016
5L1E
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BU of 5l1e by Molmil
AMPA subtype ionotropic glutamate receptor GluA2 in complex with noncompetitive inhibitor CP465022
Descriptor: 2-acetamido-2-deoxy-beta-D-glucopyranose, 3-(2-chlorophenyl)-2-(2-{6-[(diethylamino)methyl]pyridin-2-yl}ethyl)-6-fluoroquinazolin-4(3H)-one, Glutamate receptor 2
Authors:Yelshanskaya, M.V, Singh, A.K, Sampson, J.M, Sobolevsky, A.I.
Deposit date:2016-07-29
Release date:2016-10-19
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (4.37 Å)
Cite:Structural Bases of Noncompetitive Inhibition of AMPA-Subtype Ionotropic Glutamate Receptors by Antiepileptic Drugs.
Neuron, 91, 2016

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건을2024-06-26부터공개중

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