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PDB: 3 results
6LJK
Crystal structure of human Sirt5 in complex with an internally quenched fluorescent substrate GluIQF
Descriptor:
BE2-SER-ALA-ILE-LYS-SER-NIY-GLY-SET, GLUTARIC ACID, NAD-dependent protein deacylase sirtuin-5, ...
Authors:
Chen, Q
,
Yu, Y.
Deposit date:
2019-12-17
Release date:
2020-12-23
Last modified:
2023-11-22
Method:
X-RAY DIFFRACTION (1.394 Å)
Cite:
Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery.
Eur.J.Med.Chem., 192, 2020
6LJM
Crystal structure of human Sirt5 in complex with the fluorogenic tetrapeptide substrate P13
Descriptor:
7-AMINO-4-METHYL-CHROMEN-2-ONE, ACE-SER-LEU-GLY-SLL, NAD-dependent protein deacylase sirtuin-5, ...
Authors:
Chen, Q
,
Yu, Y.
Deposit date:
2019-12-17
Release date:
2020-10-28
Last modified:
2023-11-29
Method:
X-RAY DIFFRACTION (1.78 Å)
Cite:
Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery.
Eur.J.Med.Chem., 192, 2020
6LJN
Crystal structure of human Sirt5 in complex with the fluorogenic tetrapeptide substrate P15
Descriptor:
7-AMINO-4-METHYL-CHROMEN-2-ONE, ACE-HIS-PHE-SER-SLL, NAD-dependent protein deacylase sirtuin-5, ...
Authors:
Chen, Q
,
Yu, Y.
Deposit date:
2019-12-17
Release date:
2020-10-28
Last modified:
2023-11-29
Method:
X-RAY DIFFRACTION (1.8 Å)
Cite:
Sensitive fluorogenic substrates for sirtuin deacylase inhibitor discovery.
Eur.J.Med.Chem., 192, 2020
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건을2024-07-17부터공개중