1HXD
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![BU of 1hxd by Molmil](/molmil-images/mine/1hxd) | CRYSTAL STRUCTURE OF E. COLI BIOTIN REPRESSOR WITH BOUND BIOTIN | 分子名称: | BIOTIN, BIRA BIFUNCTIONAL PROTEIN | 著者 | Kwon, K, Streaker, E.D, Ruparelia, S, Beckett, D. | 登録日 | 2001-01-12 | 公開日 | 2001-05-30 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Corepressor-induced organization and assembly of the biotin repressor: a model for allosteric activation of a transcriptional regulator. Proc.Natl.Acad.Sci.USA, 98, 2001
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3FJP
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![BU of 3fjp by Molmil](/molmil-images/mine/3fjp) | Apo structure of Biotin protein ligase from Aquifex aeolicus | 分子名称: | Biotin [acetyl-CoA-carboxylase] ligase, SULFATE ION | 著者 | McNae, I.W, Tron, C.M, Baxter, R.L, Walkinshaw, M.D, Campopiano, D.J. | 登録日 | 2008-12-15 | 公開日 | 2009-06-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural and functional studies of the biotin protein ligase from Aquifex aeolicus reveal a critical role for a conserved residue in target specificity. J.Mol.Biol., 387, 2009
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4WF2
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![BU of 4wf2 by Molmil](/molmil-images/mine/4wf2) | Structure of E. coli BirA G142A bound to biotinol-5'-AMP | 分子名称: | ((2R,3S,4R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-3,4-DIHYDROXY-TETRAHYDROFURAN-2-YL)METHYL 5-((3AS,4S,6AR)-2-OXO-HEXAHYDRO-1H-THIENO[3,4-D]IMIDAZOL-4-YL)PENTYL HYDROGEN PHOSPHATE, Bifunctional ligase/repressor BirA | 著者 | Eginton, C, Beckett, D, Wade, H. | 登録日 | 2014-09-11 | 公開日 | 2014-10-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.31 Å) | 主引用文献 | Allosteric Coupling via Distant Disorder-to-Order Transitions. J.Mol.Biol., 427, 2015
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4OP0
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![BU of 4op0 by Molmil](/molmil-images/mine/4op0) | Crystal structure of biotin protein ligase (RV3279C) of Mycobacterium tuberculosis, complexed with biotinyl-5'-AMP | 分子名称: | BIOTINYL-5-AMP, BirA bifunctional protein, SULFATE ION | 著者 | Ma, Q, Wilmanns, M, Akhter, Y. | 登録日 | 2014-02-04 | 公開日 | 2014-04-30 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Active site conformational changes upon reaction intermediate biotinyl-5'-AMP binding in biotin protein ligase from Mycobacterium tuberculosis. Protein Sci., 23, 2014
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8FI3
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![BU of 8fi3 by Molmil](/molmil-images/mine/8fi3) | |
2ZGW
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![BU of 2zgw by Molmil](/molmil-images/mine/2zgw) | Crystal Structure Of Biotin Protein Ligase From Pyrococcus Horikoshii Complexed with Adenosine and Biotin, Mutations R48A and K111A | 分子名称: | ADENOSINE, BIOTIN, biotin--[acetyl-CoA-carboxylase] ligase | 著者 | Bagautdinov, B, Matsuura, Y, Bagautdinova, S, Kunishima, N, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2008-01-28 | 公開日 | 2008-02-05 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Protein biotinylation visualized by a complex structure of biotin protein ligase with a substrate J.Biol.Chem., 283, 2008
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3RUX
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![BU of 3rux by Molmil](/molmil-images/mine/3rux) | |
6NDL
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![BU of 6ndl by Molmil](/molmil-images/mine/6ndl) | Crystal structure of Staphylococcus aureus biotin protein ligase in complex with a sulfonamide inhibitor | 分子名称: | 1-[4-(6-aminopurin-9-yl)butylsulfamoyl]-3-[4-[(4~{S})-2-oxidanylidene-1,3,3~{a},4,6,6~{a}-hexahydrothieno[3,4-d]imidazol-4-yl]butyl]urea, Biotin Protein Ligase, GLYCEROL | 著者 | Marshall, A.C, Polyak, S.W, Bruning, J.B, Lee, K. | 登録日 | 2018-12-13 | 公開日 | 2019-12-18 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Sulfonamide-Based Inhibitors of Biotin Protein Ligase as New Antibiotic Leads. Acs Chem.Biol., 14, 2019
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6ORU
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![BU of 6oru by Molmil](/molmil-images/mine/6oru) | |
1BIA
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![BU of 1bia by Molmil](/molmil-images/mine/1bia) | |
1BIB
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![BU of 1bib by Molmil](/molmil-images/mine/1bib) | |
3EFR
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![BU of 3efr by Molmil](/molmil-images/mine/3efr) | Biotin protein ligase R40G mutant from Aquifex aeolicus in complex with biotin | 分子名称: | BIOTIN, Biotin [acetyl-CoA-carboxylase] ligase, SULFATE ION | 著者 | Tron, C.M, McNae, I.W, Walkinshaw, M.D, Baxter, R.L, Campopiano, D.J. | 登録日 | 2008-09-10 | 公開日 | 2009-06-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Structural and functional studies of the biotin protein ligase from Aquifex aeolicus reveal a critical role for a conserved residue in target specificity. J.Mol.Biol., 387, 2009
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8ENI
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![BU of 8eni by Molmil](/molmil-images/mine/8eni) | Crystal structure of Staphylococcus aureus biotin protein ligase in complex with inhibitor | 分子名称: | 3-[4-(5-fluoro-4-{5-[(3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentyl}-1H-1,2,3-triazol-1-yl)butyl]-5-methyl-1,3-benzoxazol-2(3H)-one, Bifunctional ligase/repressor BirA | 著者 | Wilce, M.C.J, Cini, D.A. | 登録日 | 2022-09-30 | 公開日 | 2022-11-30 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Halogenation of Biotin Protein Ligase Inhibitors Improves Whole Cell Activity against Staphylococcus aureus. ACS Infect Dis, 4, 2018
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8F8U
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![BU of 8f8u by Molmil](/molmil-images/mine/8f8u) | |
3EFS
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![BU of 3efs by Molmil](/molmil-images/mine/3efs) | Biotin protein ligase from Aquifex aeolicus in complex with biotin and ATP | 分子名称: | ADENOSINE-5'-TRIPHOSPHATE, BIOTIN, Biotin [acetyl-CoA-carboxylase] ligase, ... | 著者 | Tron, C.M, McNae, I.W, Walkinshaw, M.D, Baxter, R.L, Campopiano, D.J. | 登録日 | 2008-09-10 | 公開日 | 2009-06-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural and functional studies of the biotin protein ligase from Aquifex aeolicus reveal a critical role for a conserved residue in target specificity. J.Mol.Biol., 387, 2009
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3L2Z
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![BU of 3l2z by Molmil](/molmil-images/mine/3l2z) | Crystal structure of hydrated Biotin Protein Ligase from M. tuberculosis | 分子名称: | BirA bifunctional protein | 著者 | Gupta, V, Gupta, R.K, Khare, G, Salunke, D.M, Tyagi, A.K. | 登録日 | 2009-12-16 | 公開日 | 2010-03-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Structural ordering of disordered ligand-binding loops of biotin protein ligase into active conformations as a consequence of dehydration. Plos One, 5, 2010
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3L1A
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![BU of 3l1a by Molmil](/molmil-images/mine/3l1a) | |
2HNI
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![BU of 2hni by Molmil](/molmil-images/mine/2hni) | |
2EWN
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![BU of 2ewn by Molmil](/molmil-images/mine/2ewn) | Ecoli Biotin Repressor with co-repressor analog | 分子名称: | ((2R,3S,4R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-3,4-DIHYDROXY-TETRAHYDROFURAN-2-YL)METHYL 5-((3AS,4S,6AR)-2-OXO-HEXAHYDRO-1H-THIENO[3,4-D]IMIDAZOL-4-YL)PENTYL HYDROGEN PHOSPHATE, BirA bifunctional protein | 著者 | Wood, Z.A, Weaver, L.H, Matthews, B.W. | 登録日 | 2005-11-04 | 公開日 | 2006-02-21 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Co-repressor Induced Order and Biotin Repressor Dimerization: A Case for Divergent Followed by Convergent Evolution. J.Mol.Biol., 357, 2006
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2FYK
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1WNL
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![BU of 1wnl by Molmil](/molmil-images/mine/1wnl) | |
1WQW
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1WQ7
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![BU of 1wq7 by Molmil](/molmil-images/mine/1wq7) | |
1X01
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![BU of 1x01 by Molmil](/molmil-images/mine/1x01) | |
1WPY
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![BU of 1wpy by Molmil](/molmil-images/mine/1wpy) | |