8V4M
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![BU of 8v4m by Molmil](/molmil-images/mine/8v4m) | CCP5 in complex with microtubules class3 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-29 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (3 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V4K
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![BU of 8v4k by Molmil](/molmil-images/mine/8v4k) | CCP5 in complex with microtubules class1 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-29 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3M
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![BU of 8v3m by Molmil](/molmil-images/mine/8v3m) | CCP5 apo structure | 分子名称: | Cytosolic carboxypeptidase-like protein 5, D-MALATE, IMIDAZOLE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3P
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![BU of 8v3p by Molmil](/molmil-images/mine/8v3p) | CCP5 in complex with Glu-P-peptide 2 transition state analog | 分子名称: | Cytosolic carboxypeptidase-like protein 5, Tubulin beta-2A chain, ZINC ION | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | X-RAY DIFFRACTION (2.36 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3R
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![BU of 8v3r by Molmil](/molmil-images/mine/8v3r) | Structure of CCP5 class2 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3Q
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![BU of 8v3q by Molmil](/molmil-images/mine/8v3q) | Structure of CCP5 class1 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V4L
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![BU of 8v4l by Molmil](/molmil-images/mine/8v4l) | CCP5 in complex with microtubules class2 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-29 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3N
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![BU of 8v3n by Molmil](/molmil-images/mine/8v3n) | CCP5 in complex with Glu-P-Glu transition state analog | 分子名称: | (2S)-2-{[(S)-[(3S)-3-acetamido-4-(ethylamino)-4-oxobutyl](hydroxy)phosphoryl]methyl}pentanedioic acid, Cytosolic carboxypeptidase-like protein 5, D-MALATE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3O
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![BU of 8v3o by Molmil](/molmil-images/mine/8v3o) | CCP5 in complex with Glu-P-peptide 1 transition state analog | 分子名称: | Cytosolic carboxypeptidase-like protein 5, D-MALATE, POTASSIUM ION, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8V3S
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![BU of 8v3s by Molmil](/molmil-images/mine/8v3s) | Structure of CCP5 class3 | 分子名称: | Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 最終更新日 | 2024-08-07 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation. Nature, 631, 2024
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8QVO
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![BU of 8qvo by Molmil](/molmil-images/mine/8qvo) | L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris | 分子名称: | CALCIUM ION, Carboxypeptidase T, SULFATE ION, ... | 著者 | Timofeev, V.I, Dorovatovskii, P.V, Lazarenko, V.A, Akparov, V.K, Kuranova, I.P. | 登録日 | 2023-10-18 | 公開日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris To Be Published
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7Q87
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![BU of 7q87 by Molmil](/molmil-images/mine/7q87) | Carboxypeptidase T with (S)-3-phenyllactic acid | 分子名称: | ALPHA-HYDROXY-BETA-PHENYL-PROPIONIC ACID, CALCIUM ION, Carboxypeptidase T, ... | 著者 | Timofeev, V.I, Akparov, V.K, Shevtsov, M.B, Kuranova, I.P. | 登録日 | 2021-11-10 | 公開日 | 2022-01-26 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Carboxypeptidase T with (S)-3-phenyllactic acid To Be Published
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7EQZ
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![BU of 7eqz by Molmil](/molmil-images/mine/7eqz) | Crystal structure of Carboxypeptidase B complexed with Potato Carboxypeptidase Inhibitor | 分子名称: | Carboxypeptidase B, GLYCINE, Metallocarboxypeptidase inhibitor, ... | 著者 | Choong, Y.K, Gavor, E, Jobichen, C, Sivaraman, J. | 登録日 | 2021-05-05 | 公開日 | 2021-11-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structure of Aedes aegypti carboxypeptidase B1-inhibitor complex uncover the disparity between mosquito and non-mosquito insect carboxypeptidase inhibition mechanism. Protein Sci., 30, 2021
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7EQX
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![BU of 7eqx by Molmil](/molmil-images/mine/7eqx) | Crystal structure of an Aedes aegypti procarboxypeptidase B1 | 分子名称: | Carboxypeptidase B, ZINC ION | 著者 | Choong, Y.K, Gavor, E, Jobichen, C, Sivaraman, J. | 登録日 | 2021-05-05 | 公開日 | 2021-11-10 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Structure of Aedes aegypti procarboxypeptidase B1 and its binding with Dengue virus for controlling infection. Life Sci Alliance, 5, 2022
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7NEE
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![BU of 7nee by Molmil](/molmil-images/mine/7nee) | Inhibitor Complex with Thrombin Activatable Fibrinolysis inhibitor (TAFIa) | 分子名称: | (1R,3S)-3-(4-ammoniobutyl)-1-benzyl-1,4-azaphosphinan-1-ium-3-carboxylate 4,4-dioxide, Carboxypeptidase B2, ZINC ION | 著者 | Brown, D.G, Schaffner, A.P, Gloanec, P, Raimbaud, E, Vuillard, L.M. | 登録日 | 2021-02-03 | 公開日 | 2021-04-07 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | Phosphinanes and Azaphosphinanes as Potent and Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor (TAFIa). J.Med.Chem., 64, 2021
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7NEU
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![BU of 7neu by Molmil](/molmil-images/mine/7neu) | Inhibitor Complex with Thrombin Activatable Fibrinolysis Inhibitor (TAFIa) | 分子名称: | (1R,3S)-3-(4-ammoniobutyl)-1-(4-fluoro-2-(1-methyl-1H-imidazol-5-yl)benzyl)-1,4-azaphosphinan-1-ium-3-carboxylate 4,4-dioxide, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Brown, D.G, Schaffner, A.P, Vuillard, L.M, Gloanec, P, Raimbauld, E. | 登録日 | 2021-02-04 | 公開日 | 2021-04-07 | 最終更新日 | 2021-04-21 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Phosphinanes and Azaphosphinanes as Potent and Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor (TAFIa). J.Med.Chem., 64, 2021
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7AQP
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![BU of 7aqp by Molmil](/molmil-images/mine/7aqp) | T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris | 分子名称: | CALCIUM ION, Carboxypeptidase T, SULFATE ION, ... | 著者 | Timofeev, V.I, Akparov, V.K, Kuranova, I.P. | 登録日 | 2020-10-22 | 公開日 | 2020-12-02 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris To Be Published
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7ARU
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![BU of 7aru by Molmil](/molmil-images/mine/7aru) | |
6Z28
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![BU of 6z28 by Molmil](/molmil-images/mine/6z28) | |
6TNK
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![BU of 6tnk by Molmil](/molmil-images/mine/6tnk) | |
6T9Y
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![BU of 6t9y by Molmil](/molmil-images/mine/6t9y) | |
6SN6
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![BU of 6sn6 by Molmil](/molmil-images/mine/6sn6) | |
6I6Z
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![BU of 6i6z by Molmil](/molmil-images/mine/6i6z) | |
6F6Q
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![BU of 6f6q by Molmil](/molmil-images/mine/6f6q) | |
6F79
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![BU of 6f79 by Molmil](/molmil-images/mine/6f79) | |