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8V4M
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BU of 8v4m by Molmil
CCP5 in complex with microtubules class3
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-29
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (3 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V4K
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BU of 8v4k by Molmil
CCP5 in complex with microtubules class1
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-29
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3M
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BU of 8v3m by Molmil
CCP5 apo structure
分子名称: Cytosolic carboxypeptidase-like protein 5, D-MALATE, IMIDAZOLE, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3P
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BU of 8v3p by Molmil
CCP5 in complex with Glu-P-peptide 2 transition state analog
分子名称: Cytosolic carboxypeptidase-like protein 5, Tubulin beta-2A chain, ZINC ION
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3R
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BU of 8v3r by Molmil
Structure of CCP5 class2
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (3.4 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3Q
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BU of 8v3q by Molmil
Structure of CCP5 class1
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V4L
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BU of 8v4l by Molmil
CCP5 in complex with microtubules class2
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, GUANOSINE-5'-TRIPHOSPHATE, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-29
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3N
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BU of 8v3n by Molmil
CCP5 in complex with Glu-P-Glu transition state analog
分子名称: (2S)-2-{[(S)-[(3S)-3-acetamido-4-(ethylamino)-4-oxobutyl](hydroxy)phosphoryl]methyl}pentanedioic acid, Cytosolic carboxypeptidase-like protein 5, D-MALATE, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3O
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BU of 8v3o by Molmil
CCP5 in complex with Glu-P-peptide 1 transition state analog
分子名称: Cytosolic carboxypeptidase-like protein 5, D-MALATE, POTASSIUM ION, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8V3S
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BU of 8v3s by Molmil
Structure of CCP5 class3
分子名称: Cytosolic carboxypeptidase-like protein 5, GLUTAMIC ACID, ZINC ION, ...
著者Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A.
登録日2023-11-28
公開日2024-07-17
最終更新日2024-08-07
実験手法ELECTRON MICROSCOPY (3.6 Å)
主引用文献Tubulin code eraser CCP5 binds branch glutamates by substrate deformation.
Nature, 631, 2024
8QVO
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BU of 8qvo by Molmil
L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris
分子名称: CALCIUM ION, Carboxypeptidase T, SULFATE ION, ...
著者Timofeev, V.I, Dorovatovskii, P.V, Lazarenko, V.A, Akparov, V.K, Kuranova, I.P.
登録日2023-10-18
公開日2024-01-17
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris
To Be Published
7Q87
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BU of 7q87 by Molmil
Carboxypeptidase T with (S)-3-phenyllactic acid
分子名称: ALPHA-HYDROXY-BETA-PHENYL-PROPIONIC ACID, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Shevtsov, M.B, Kuranova, I.P.
登録日2021-11-10
公開日2022-01-26
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Carboxypeptidase T with (S)-3-phenyllactic acid
To Be Published
7EQZ
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BU of 7eqz by Molmil
Crystal structure of Carboxypeptidase B complexed with Potato Carboxypeptidase Inhibitor
分子名称: Carboxypeptidase B, GLYCINE, Metallocarboxypeptidase inhibitor, ...
著者Choong, Y.K, Gavor, E, Jobichen, C, Sivaraman, J.
登録日2021-05-05
公開日2021-11-10
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Structure of Aedes aegypti carboxypeptidase B1-inhibitor complex uncover the disparity between mosquito and non-mosquito insect carboxypeptidase inhibition mechanism.
Protein Sci., 30, 2021
7EQX
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BU of 7eqx by Molmil
Crystal structure of an Aedes aegypti procarboxypeptidase B1
分子名称: Carboxypeptidase B, ZINC ION
著者Choong, Y.K, Gavor, E, Jobichen, C, Sivaraman, J.
登録日2021-05-05
公開日2021-11-10
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.08 Å)
主引用文献Structure of Aedes aegypti procarboxypeptidase B1 and its binding with Dengue virus for controlling infection.
Life Sci Alliance, 5, 2022
7NEE
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BU of 7nee by Molmil
Inhibitor Complex with Thrombin Activatable Fibrinolysis inhibitor (TAFIa)
分子名称: (1R,3S)-3-(4-ammoniobutyl)-1-benzyl-1,4-azaphosphinan-1-ium-3-carboxylate 4,4-dioxide, Carboxypeptidase B2, ZINC ION
著者Brown, D.G, Schaffner, A.P, Gloanec, P, Raimbaud, E, Vuillard, L.M.
登録日2021-02-03
公開日2021-04-07
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2.55 Å)
主引用文献Phosphinanes and Azaphosphinanes as Potent and Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor (TAFIa).
J.Med.Chem., 64, 2021
7NEU
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BU of 7neu by Molmil
Inhibitor Complex with Thrombin Activatable Fibrinolysis Inhibitor (TAFIa)
分子名称: (1R,3S)-3-(4-ammoniobutyl)-1-(4-fluoro-2-(1-methyl-1H-imidazol-5-yl)benzyl)-1,4-azaphosphinan-1-ium-3-carboxylate 4,4-dioxide, 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Brown, D.G, Schaffner, A.P, Vuillard, L.M, Gloanec, P, Raimbauld, E.
登録日2021-02-04
公開日2021-04-07
最終更新日2021-04-21
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Phosphinanes and Azaphosphinanes as Potent and Selective Inhibitors of Activated Thrombin-Activatable Fibrinolysis Inhibitor (TAFIa).
J.Med.Chem., 64, 2021
7AQP
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BU of 7aqp by Molmil
T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris
分子名称: CALCIUM ION, Carboxypeptidase T, SULFATE ION, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-10-22
公開日2020-12-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris
To Be Published
7ARU
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BU of 7aru by Molmil
L254N mutant of carboxypeptidase T from Thermoactinomyces vulgaris N-sulfamoyl-L-valine
分子名称: (2~{S})-3-methyl-2-(sulfamoylamino)butanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-10-26
公開日2020-11-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献L254N mutant of carboxypeptidase T from Thermoactinomyces vulgaris N-sulfamoyl-L-valine
To Be Published
6Z28
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BU of 6z28 by Molmil
Carboxypeptidase T mutant L254N with N-sulfamoyl-L-glutamic acid
分子名称: CALCIUM ION, Carboxypeptidase T, N-sulfamoyl-L-glutamic acid, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-05-15
公開日2020-05-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献CARBOXYPEPTIDASE T MUTANT L254N WITH WITH N-SULFAMOYL-L-GLUT
To Be Published
6TNK
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BU of 6tnk by Molmil
CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-VALINE
分子名称: (2~{S})-3-methyl-2-(sulfamoylamino)butanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-12-09
公開日2019-12-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-VALINE
To Be Published
6T9Y
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BU of 6t9y by Molmil
CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-LYSIN
分子名称: (2~{S})-6-azanyl-2-(sulfamoylamino)hexanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-10-29
公開日2019-12-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-LYSIN
To Be Published
6SN6
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BU of 6sn6 by Molmil
CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-GLUTAMIC ACID
分子名称: CALCIUM ION, Carboxypeptidase T, N-sulfamoyl-L-glutamic acid, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-08-23
公開日2019-10-09
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-GLUTAMIC ACID
To Be Published
6I6Z
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BU of 6i6z by Molmil
Crystal structure of the human CARBOXYPEPTIDASE A1 in complex with the PHOSPHINIC INHIBITOR Acetyl-Tyr-Ala-Y(PO2CH2)-homoPhe-OH
分子名称: (2S)-2-{[(S)-{(1R)-1-[(N-acetyl-L-tyrosyl)amino]ethyl}(hydroxy)phosphoryl]methyl}-4-phenylbutanoic acid, Carboxypeptidase A1, ZINC ION
著者Gallego, P, Reverter, D.
登録日2018-11-15
公開日2018-12-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Synthesis and Structural/Functional Characterization of Selective M14 Metallocarboxypeptidase Inhibitors Based on Phosphinic Pseudopeptide Scaffold: Implications on the Design of Specific Optical Probes.
J. Med. Chem., 62, 2019
6F6Q
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BU of 6f6q by Molmil
Carboxypeptidase T mutant L254N with Sulphamoil Arginine
分子名称: CALCIUM ION, Carboxypeptidase T, N~2~-sulfamoyl-L-arginine, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2017-12-06
公開日2018-08-15
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Carboxypeptidase T mutant L254N with Sulphamoil Arginine
To Be Published
6F79
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BU of 6f79 by Molmil
Carboxypeptidase T mutant L211Q with Sulphamoil Arginine
分子名称: CALCIUM ION, Carboxypeptidase T, N~2~-sulfamoyl-L-arginine, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2017-12-07
公開日2018-08-15
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Carboxypeptidase T mutant L211Q with Sulphamoil Arginine
To Be Published

223532

件を2024-08-07に公開中

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