8X37
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![BU of 8x37 by Molmil](/molmil-images/mine/8x37) | Neryl diphosphate synthase from Solanum lycopersicum complexed with DMSAPP | 分子名称: | DIMETHYLALLYL S-THIOLODIPHOSPHATE, MAGNESIUM ION, Neryl-diphosphate synthase 1 | 著者 | Imaizumi, R, Matsuura, H, Yanai, T, Takeshita, K, Misawa, S, Yamaguchi, H, Sakai, N, Miyagi-Inoue, Y, Suenaga-Hiromori, M, Kataoka, K, Nakayama, T, Yamamoto, M, Takahashi, S, Yamashita, S. | 登録日 | 2023-11-12 | 公開日 | 2024-02-07 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Structural-Functional Correlations between Unique N-terminal Region and C-terminal Conserved Motif in Short-chain cis-Prenyltransferase from Tomato. Chembiochem, 25, 2024
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1KAR
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![BU of 1kar by Molmil](/molmil-images/mine/1kar) | L-HISTIDINOL DEHYDROGENASE (HISD) STRUCTURE COMPLEXED WITH HISTAMINE (INHIBITOR), ZINC AND NAD (COFACTOR) | 分子名称: | HISTAMINE, Histidinol dehydrogenase, ZINC ION | 著者 | Barbosa, J.A.R.G, Sivaraman, J, Li, Y, Larocque, R, Matte, A, Schrag, J.D, Cygler, M. | 登録日 | 2001-11-02 | 公開日 | 2002-06-12 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Mechanism of action and NAD+-binding mode revealed by the crystal structure of L-histidinol dehydrogenase. Proc.Natl.Acad.Sci.USA, 99, 2002
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3DU0
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![BU of 3du0 by Molmil](/molmil-images/mine/3du0) | E. coli dihydrodipicolinate synthase with first substrate, pyruvate, bound in active site | 分子名称: | CHLORIDE ION, Dihydrodipicolinate synthase, GLYCEROL, ... | 著者 | Dobson, R.C.J, Devenish, S.R.A, Gerrard, J.A, Jameson, G.B. | 登録日 | 2008-07-16 | 公開日 | 2008-11-18 | 最終更新日 | 2019-12-18 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The high-resolution structure of dihydrodipicolinate synthase from Escherichia coli bound to its first substrate, pyruvate. Acta Crystallogr.,Sect.F, 64, 2008
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5N61
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![BU of 5n61 by Molmil](/molmil-images/mine/5n61) | RNA polymerase I initially transcribing complex | 分子名称: | DNA-directed RNA polymerase I subunit RPA12, DNA-directed RNA polymerase I subunit RPA135, DNA-directed RNA polymerase I subunit RPA14, ... | 著者 | Engel, C, Gubbey, T, Neyer, S, Sainsbury, S, Oberthuer, C, Baejen, C, Bernecky, C, Cramer, P. | 登録日 | 2017-02-14 | 公開日 | 2017-04-05 | 最終更新日 | 2019-10-02 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Structural Basis of RNA Polymerase I Transcription Initiation. Cell, 169, 2017
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1DHP
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![BU of 1dhp by Molmil](/molmil-images/mine/1dhp) | DIHYDRODIPICOLINATE SYNTHASE | 分子名称: | DIHYDRODIPICOLINATE SYNTHASE, POTASSIUM ION | 著者 | Mirwaldt, C, Korndoerfer, I, Huber, R. | 登録日 | 1995-02-09 | 公開日 | 1997-02-12 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | The crystal structure of dihydrodipicolinate synthase from Escherichia coli at 2.5 A resolution. J.Mol.Biol., 246, 1995
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8UN8
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8XPZ
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![BU of 8xpz by Molmil](/molmil-images/mine/8xpz) | The Crystal Structure of TTBK1 from Biortus. | 分子名称: | 1,2-ETHANEDIOL, Tau-tubulin kinase 1 | 著者 | Wang, F, Cheng, W, Yuan, Z, Lin, D, Ni, C. | 登録日 | 2024-01-04 | 公開日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | The Crystal Structure of TTBK1 from Biortus. To Be Published
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5M64
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![BU of 5m64 by Molmil](/molmil-images/mine/5m64) | RNA Polymerase I elongation complex with A49 tandem winged helix domain | 分子名称: | DNA-directed RNA polymerase I subunit RPA12, DNA-directed RNA polymerase I subunit RPA135, DNA-directed RNA polymerase I subunit RPA14, ... | 著者 | Tafur, L, Sadian, Y, Hoffmann, N.A, Jakobi, A.J, Wetzel, R, Hagen, W.J.H, Sachse, C, Muller, C.W. | 登録日 | 2016-10-24 | 公開日 | 2016-12-21 | 最終更新日 | 2019-12-11 | 実験手法 | ELECTRON MICROSCOPY (4.6 Å) | 主引用文献 | Molecular Structures of Transcribing RNA Polymerase I. Mol. Cell, 64, 2016
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5N5Y
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![BU of 5n5y by Molmil](/molmil-images/mine/5n5y) | Cryo-EM structure of RNA polymerase I in complex with Rrn3 and Core Factor (Orientation III) | 分子名称: | DNA-directed RNA polymerase I subunit RPA12, DNA-directed RNA polymerase I subunit RPA135, DNA-directed RNA polymerase I subunit RPA14, ... | 著者 | Engel, C, Gubbey, T, Neyer, S, Sainsbury, S, Oberthuer, C, Baejen, C, Bernecky, C, Cramer, P. | 登録日 | 2017-02-14 | 公開日 | 2017-04-05 | 最終更新日 | 2018-10-03 | 実験手法 | ELECTRON MICROSCOPY (7.7 Å) | 主引用文献 | Structural Basis of RNA Polymerase I Transcription Initiation. Cell, 169, 2017
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5N5Z
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![BU of 5n5z by Molmil](/molmil-images/mine/5n5z) | Cryo-EM structure of RNA polymerase I in complex with Rrn3 and Core Factor (Orientation II) | 分子名称: | DNA-directed RNA polymerase I subunit RPA12, DNA-directed RNA polymerase I subunit RPA135, DNA-directed RNA polymerase I subunit RPA14, ... | 著者 | Engel, C, Gubbey, T, Neyer, S, Sainsbury, S, Oberthuer, C, Baejen, C, Bernecky, C, Cramer, P. | 登録日 | 2017-02-14 | 公開日 | 2017-04-05 | 最終更新日 | 2018-10-03 | 実験手法 | ELECTRON MICROSCOPY (7.7 Å) | 主引用文献 | Structural Basis of RNA Polymerase I Transcription Initiation. Cell, 169, 2017
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6HLQ
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![BU of 6hlq by Molmil](/molmil-images/mine/6hlq) | Yeast RNA polymerase I* elongation complex bound to nucleotide analog GMPCPP | 分子名称: | DNA-directed RNA polymerase I subunit RPA12, DNA-directed RNA polymerase I subunit RPA135, DNA-directed RNA polymerase I subunit RPA14, ... | 著者 | Tafur, L, Sadian, Y, Weis, F, Muller, C.W. | 登録日 | 2018-09-11 | 公開日 | 2019-04-03 | 最終更新日 | 2024-05-15 | 実験手法 | ELECTRON MICROSCOPY (3.18 Å) | 主引用文献 | The cryo-EM structure of a 12-subunit variant of RNA polymerase I reveals dissociation of the A49-A34.5 heterodimer and rearrangement of subunit A12.2. Elife, 8, 2019
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5ENJ
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![BU of 5enj by Molmil](/molmil-images/mine/5enj) | Crystal structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in complex with compound-14 N11530 (SGC - Diamond I04-1 fragment screening) | 分子名称: | MAGNESIUM ION, PH-interacting protein, ~{N}-[[2,6-bis(chloranyl)phenyl]methyl]-~{N}-methyl-ethanamide | 著者 | Krojer, T, Talon, R, Collins, P, Bradley, A, Cox, O, Szykowska, A, Burgess-Brown, N, Brennan, P, Bountra, C, Arrowsmith, C.H, Edwards, A, von Delft, F, Structural Genomics Consortium (SGC) | 登録日 | 2015-11-09 | 公開日 | 2016-04-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Chem Sci, 7, 2016
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5ENE
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![BU of 5ene by Molmil](/molmil-images/mine/5ene) | Crystal structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in complex with 5-Amino-2-benzyl-1,3-oxazole-4-carbonitrile (SGC - Diamond I04-1 fragment screening) | 分子名称: | 5-azanyl-2-(phenylmethyl)-1,3-oxazole-4-carbonitrile, PH-interacting protein | 著者 | Krojer, T, Talon, R, Collins, P, Bradley, A, Cox, O, Amin, J, Szykowska, A, Burgess-Brown, N, Spencer, J, Brennan, P, Bountra, C, Arrowsmith, C.H, Edwards, A, von Delft, F, Structural Genomics Consortium (SGC) | 登録日 | 2015-11-09 | 公開日 | 2016-04-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.49 Å) | 主引用文献 | A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Chem Sci, 7, 2016
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7JZB
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7JZC
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7JZD
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7JZG
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7JZF
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7AV9
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![BU of 7av9 by Molmil](/molmil-images/mine/7av9) | Crystal Structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 | 分子名称: | 1,2-ETHANEDIOL, PH-interacting protein | 著者 | Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F. | 登録日 | 2020-11-04 | 公開日 | 2021-01-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.23 Å) | 主引用文献 | Crystal Structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group C2 To Be Published
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7JZ9
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7JZE
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7JZA
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7JZ7
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![BU of 7jz7 by Molmil](/molmil-images/mine/7jz7) | Dihydrodipicolinate synthase mutant S48F | 分子名称: | 4-hydroxy-tetrahydrodipicolinate synthase, GLYCEROL, POTASSIUM ION | 著者 | Board, A.J, Dobson, R.C.J. | 登録日 | 2020-09-01 | 公開日 | 2021-10-06 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Mapping the unchartered waters of dihydrodipicolinate synthase: a novel mechanism of allosteric inhibition. To Be Published
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7JZ8
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7AV8
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![BU of 7av8 by Molmil](/molmil-images/mine/7av8) | Crystal Structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group P21212 | 分子名称: | PH-interacting protein | 著者 | Krojer, T, Talon, R, Fairhead, M, Szykowska, A, Burgess-Brown, N.A, Brennan, P.E, Arrowsmith, C.H, Edwards, A.M, Bountra, C, von Delft, F, Structural Genomics Consortium (SGC) | 登録日 | 2020-11-04 | 公開日 | 2021-01-13 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.63 Å) | 主引用文献 | Crystal Structure of the second bromodomain of Pleckstrin homology domain interacting protein (PHIP) in space group P21212 To Be Published
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