7Q1C
| Crystal structure of Trypanosoma cruzi histone deacetylase DAC2 complexed with a hydroxamate inhibitor | 分子名称: | (E)-3-dibenzofuran-4-yl-N-oxidanyl-prop-2-enamide, Histone deacetylase DAC2, POTASSIUM ION, ... | 著者 | Ramos-Morales, E, Marek, M, Romier, C. | 登録日 | 2021-10-18 | 公開日 | 2021-12-15 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Species-selective targeting of pathogens revealed by the atypical structure and active site of Trypanosoma cruzi histone deacetylase DAC2. Cell Rep, 37, 2021
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8AP8
| Peripheral stalk of Trypanosoma brucei mitochondrial ATP synthase | 分子名称: | ATPTB3, ATPTB4, OSCP, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8AP9
| rotor of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | ATP synthase gamma subunit, ATP synthase subunit epsilon, mitochondrial, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 最終更新日 | 2024-07-24 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8AP7
| membrane region of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (2.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APC
| rotational state 1c of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APF
| rotational state 2a of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (4.3 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APJ
| rotational state 2d of Trypanosoma brucei mitochondrial ATP synthase | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APD
| rotational state 1d of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APB
| rotational state 1b of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APH
| rotational state 2c of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.8 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APE
| rotational state 1e of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APA
| rotational state 1a of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APG
| rotational state 2b of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-dioleoyl-sn-glycero-3-phosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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8APK
| rotational state 3 of the Trypanosoma brucei mitochondrial ATP synthase dimer | 分子名称: | 1,2-DIACYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, 2-{[(4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranosyl)oxy]methyl}-4-{[(3beta,9beta,14beta,17beta,25R)-spirost-5-en-3-yl]oxy}butyl 4-O-alpha-D-glucopyranosyl-alpha-D-glucopyranoside, ... | 著者 | Muehleip, A, Gahura, O, Zikova, A, Amunts, A. | 登録日 | 2022-08-09 | 公開日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | An ancestral interaction module promotes oligomerization in divergent mitochondrial ATP synthases. Nat Commun, 13, 2022
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6UJ5
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8STX
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5FUW
| catalytic domain of Thymidine kinase from Trypanosoma brucei with dTMP or dThd | 分子名称: | PHOSPHATE ION, THYMDINE KINASE, THYMIDINE, ... | 著者 | Timm, J, Valente, M, Castillo-Acosta, V, Balzarini, T, Nettleship, J.E, Rada, H, Wilson, K.S, Gonzalez-Pacanowska, D. | 登録日 | 2016-01-31 | 公開日 | 2016-07-27 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Cell Cycle Regulation and Novel Structural Features of Thymidine Kinase, an Essential Enzyme in Trypanosoma Brucei. Mol.Microbiol., 102, 2016
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4I70
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8S9Y
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5N8V
| Targeting the PEX14-PEX5 interaction by small molecules provides novel therapeutic routes to treat trypanosomiases. | 分子名称: | 1-(2-azanylethyl)-5-[(4-methoxynaphthalen-1-yl)methyl]-~{N}-(naphthalen-1-ylmethyl)-6,7-dihydro-4~{H}-pyrazolo[4,3-c]pyridine-3-carboxamide, BETA-MERCAPTOETHANOL, CHLORIDE ION, ... | 著者 | Dawidowski, M, Emmanouilidis, L, Sattler, M, Popowicz, G.M. | 登録日 | 2017-02-24 | 公開日 | 2017-03-15 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | Inhibitors of PEX14 disrupt protein import into glycosomes and kill Trypanosoma parasites. Science, 355, 2017
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2K11
| Solution structure of human pancreatic ribonuclease | 分子名称: | Pancreatic Ribonuclease | 著者 | Kover, K.E, Bruix, M, Santoro, J, Batta, G, Laurents, D.V, Rico, M. | 登録日 | 2008-02-20 | 公開日 | 2008-06-03 | 最終更新日 | 2022-03-16 | 実験手法 | SOLUTION NMR | 主引用文献 | The solution structure and dynamics of human pancreatic ribonuclease determined by NMR spectroscopy provide insight into its remarkable biological activities and inhibition. J.Mol.Biol., 379, 2008
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3QTT
| Crystal Structure of Pantoate-beta-alanine Ligase from Francisella tularensis Complexed with Beta-gamma ATP and Beta-alanine | 分子名称: | BETA-ALANINE, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, ... | 著者 | Maltseva, N, Kim, Y, Kwon, K, Anderson, W.F, Joachimiak, A, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2011-02-23 | 公開日 | 2011-03-23 | 最終更新日 | 2017-11-08 | 実験手法 | X-RAY DIFFRACTION (2.599 Å) | 主引用文献 | Crystal Structure of Pantoate-beta-alanine Ligase from Francisella tularensis Complexed with Beta-gamma ATP and Beta-alanine. To be Published
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4MYL
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4MYF
| Crystal structure of Trypanosoma cruzi formiminoglutamase(oxidized) with Mn2+2 at pH 6.0 | 分子名称: | Formiminoglutamase, MANGANESE (II) ION | 著者 | Hai, Y, Dugery, R.J, Healy, D, Christianson, D.W. | 登録日 | 2013-09-27 | 公開日 | 2013-11-27 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.799 Å) | 主引用文献 | Formiminoglutamase from trypanosoma cruzi is an arginase-like manganese metalloenzyme. Biochemistry, 52, 2013
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4I73
| Crystal structure of the Trypanosoma brucei Inosine-Adenosine-Guanosine nucleoside hydrolase in complex with compound UAMC-00312 | 分子名称: | (2R,3R,4S)-2-(hydroxymethyl)-1-[(4-hydroxythieno[3,2-d]pyrimidin-7-yl)methyl]pyrrolidine-3,4-diol, CALCIUM ION, Inosine-adenosine-guanosine-nucleoside hydrolase, ... | 著者 | Giannese, F, Degano, M. | 登録日 | 2012-11-30 | 公開日 | 2013-08-07 | 最終更新日 | 2013-12-18 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Structures of purine nucleosidase from Trypanosoma brucei bound to isozyme-specific trypanocidals and a novel metalorganic inhibitor Acta Crystallogr.,Sect.D, 69, 2013
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