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7BA7
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Cys-42-tethered stabilizer 9 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-[3,5-bis(chloranyl)phenoxy]-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
5CHW
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BU of 5chw by Molmil
Structure of ISG15 in space group P212121
分子名称: GLYCEROL, SULFATE ION, Ubiquitin-like protein ISG15
著者Fritz, G, Basters, A.
登録日2015-07-10
公開日2016-09-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Structure of ISG15 in space group P212121
To Be Published
7BA5
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BU of 7ba5 by Molmil
Cys-42-tethered stabilizer 7 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(4-fluoranylphenoxy)-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
1I37
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BU of 1i37 by Molmil
CRYSTAL STRUCTURE OF THE RAT ANDROGEN RECEPTOR LIGAND BINDING DOMAIN COMPLEX WITH DIHYDROTESTOSTERONE
分子名称: 5-ALPHA-DIHYDROTESTOSTERONE, ANDROGEN RECEPTOR
著者Sack, J.S.
登録日2001-02-13
公開日2001-03-21
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystallographic structures of the ligand-binding domains of the androgen receptor and its T877A mutant complexed with the natural agonist dihydrotestosterone.
Proc.Natl.Acad.Sci.USA, 98, 2001
7BA9
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BU of 7ba9 by Molmil
Cys-42-tethered stabilizer 11 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-methyl-2-(4-methylphenoxy)-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.48 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
1IAW
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BU of 1iaw by Molmil
CRYSTAL STRUCTURE OF NAEI COMPLEXED WITH 17MER DNA
分子名称: 5'-D(*TP*GP*CP*CP*AP*CP*GP*CP*CP*GP*GP*CP*GP*TP*GP*GP*C)-3', TYPE II RESTRICTION ENZYME NAEI
著者Huai, Q, Colandene, J.D, Topal, M.D, Ke, H.
登録日2001-03-23
公開日2001-08-03
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structure of NaeI-DNA complex reveals dual-mode DNA recognition and complete dimer rearrangement.
Nat.Struct.Biol., 8, 2001
2IIE
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BU of 2iie by Molmil
single chain Integration Host Factor protein (scIHF2) in complex with DNA
分子名称: DNA (5'-D(*DGP*DCP*DTP*DTP*DAP*DTP*DCP*DAP*DAP*DTP*DTP*DTP*DGP*DTP*DTP*DGP*DCP*DAP*DCP*DC)-3'), DNA (5'-D(*DGP*DGP*DCP*DCP*DAP*DAP*DAP*DAP*DAP*DAP*DGP*DCP*DAP*DTP*DT)-3'), Integration host factor, ...
著者Bao, Q, Droege, P, Davey, C.A.
登録日2006-09-28
公開日2007-02-20
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.41 Å)
主引用文献A Divalent Metal-mediated Switch Controlling Protein-induced DNA Bending
J.Mol.Biol., 367, 2007
7BAA
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BU of 7baa by Molmil
Cys-42-tethered stabilizer 12 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(4-bromanyl-3-methoxy-phenoxy)-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
6YNU
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BU of 6ynu by Molmil
CaM-P458 complex (crystal form 1)
分子名称: Bifunctional adenylate cyclase toxin/hemolysin CyaA, CALCIUM ION, Calmodulin-1
著者Mechaly, A.E, Voegele, A, Haouz, A, Chenal, A.
登録日2020-04-14
公開日2021-03-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.12 Å)
主引用文献A High-Affinity Calmodulin-Binding Site in the CyaA Toxin Translocation Domain is Essential for Invasion of Eukaryotic Cells.
Adv Sci, 8, 2021
5JTH
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BU of 5jth by Molmil
Crystal structure of E67A calmodulin - CaM:RM20 analog complex
分子名称: CALCIUM ION, Calmodulin, Myosin light chain kinase, ...
著者Grum-Tokars, V.L, Minasov, G, Anderson, W.F, Watterson, D.M.
登録日2016-05-09
公開日2017-07-19
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Crystal structure of E67A calmodulin - CaM:RM20 analog complex
To Be Published
7BA8
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BU of 7ba8 by Molmil
Cys-42-tethered stabilizer 10 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-methyl-2-phenoxy-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
6YNS
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BU of 6yns by Molmil
CaM-P458 complex (crystal form 2)
分子名称: Bifunctional adenylate cyclase toxin/hemolysin CyaA, CALCIUM ION, Calmodulin-1
著者Mechaly, A.E, Voegele, A, Haouz, A, Chenal, A.
登録日2020-04-14
公開日2021-03-17
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (3.94 Å)
主引用文献A High-Affinity Calmodulin-Binding Site in the CyaA Toxin Translocation Domain is Essential for Invasion of Eukaryotic Cells.
Adv Sci, 8, 2021
6TDZ
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BU of 6tdz by Molmil
Cryo-EM structure of Euglena gracilis mitochondrial ATP synthase, OSCP/F1/c-ring, rotational state 2
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, FRAGMENT OF TRITON X-100, ...
著者Muhleip, A, Amunts, A.
登録日2019-11-10
公開日2019-11-27
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (3.14 Å)
主引用文献Structure of a mitochondrial ATP synthase with bound native cardiolipin.
Elife, 8, 2019
7B9T
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BU of 7b9t by Molmil
Cys-45-tethered stabilizer 5 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(4-chlorophenyl)sulfanyl-~{N}-(3-sulfanylpropyl)ethanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-14
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
7BA6
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BU of 7ba6 by Molmil
Cys-42-tethered stabilizer 8 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-[3,5-bis(fluoranyl)phenoxy]-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
6CSF
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BU of 6csf by Molmil
Crystal structure of sodium/alanine symporter AgcS with D-alanine bound
分子名称: D-ALANINE, Monoclonal antibody FAB heavy chain, Monoclonal antibody FAB light chain, ...
著者Ma, J, Reyes, F.E, Gonen, T.
登録日2018-03-20
公開日2019-01-30
最終更新日2019-02-20
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Structural basis for substrate binding and specificity of a sodium-alanine symporter AgcS.
Proc. Natl. Acad. Sci. U.S.A., 116, 2019
7BAB
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BU of 7bab by Molmil
Cys-42-tethered stabilizer 13 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-[2-chloranyl-4-[oxidanyl(oxidanylidene)-$l^{4}-azanyl]phenoxy]-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
2IO4
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BU of 2io4 by Molmil
Crystal structure of PCNA12 dimer from Sulfolobus solfataricus.
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, DNA polymerase sliding clamp B, ...
著者Hlinkova, V, Ling, H.
登録日2006-10-09
公開日2008-04-08
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Structures of monomeric, dimeric and trimeric PCNA: PCNA-ring assembly and opening.
Acta Crystallogr.,Sect.D, 64, 2008
7B9M
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BU of 7b9m by Molmil
Cys-45-tethered stabilizer 3 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(2-cyanophenyl)sulfanyl-~{N}-(2-sulfanylethyl)benzamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-14
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
7B9R
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BU of 7b9r by Molmil
Cys-45-tethered stabilizer 4 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(2-cyanophenyl)sulfanyl-~{N}-(3-sulfanylpropyl)benzamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-14
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
7BA3
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BU of 7ba3 by Molmil
Cys-42-tethered stabilizer 6 of 14-3-3(sigma)/ERa PPI
分子名称: 14-3-3 protein sigma, 2-(4-bromanylphenoxy)-2-methyl-~{N}-(2-sulfanylethyl)propanamide, Estrogen receptor, ...
著者Sijbesma, E, Ottmann, C.
登録日2020-12-15
公開日2021-07-07
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Exploration of a 14-3-3 PPI Pocket by Covalent Fragments as Stabilizers.
Acs Med.Chem.Lett., 12, 2021
2J5D
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BU of 2j5d by Molmil
NMR structure of BNIP3 transmembrane domain in lipid bicelles
分子名称: BCL2/ADENOVIRUS E1B 19 KDA PROTEIN-INTERACTING PROTEIN 3
著者Bocharov, E.V, Pustovalova, Y.E, Volynsky, P.E, Maslennikov, I.V, Goncharuk, M.V, Ermolyuk, Y.S, Arseniev, A.S.
登録日2006-09-14
公開日2007-04-17
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Unique dimeric structure of BNip3 transmembrane domain suggests membrane permeabilization as a cell death trigger.
J. Biol. Chem., 282, 2007
7KZ0
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BU of 7kz0 by Molmil
Human MBD4 glycosylase domain bound to DNA containing substrate analog 2'-deoxy-pseudouridine
分子名称: DNA (5'-D(*CP*CP*AP*GP*CP*GP*(P2U)P*GP*CP*AP*GP*C)-3'), DNA (5'-D(*GP*CP*TP*GP*CP*GP*CP*GP*CP*TP*GP*G)-3'), GLYCEROL, ...
著者Pidugu, L.S, Pozharski, E, Drohat, A.C.
登録日2020-12-09
公開日2021-11-10
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.57 Å)
主引用文献Structural Insights into the Mechanism of Base Excision by MBD4.
J.Mol.Biol., 433, 2021
7KZG
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BU of 7kzg by Molmil
Human MBD4 glycosylase domain bound to DNA containing oxacarbenium-ion analog 1-aza-2'-deoxyribose
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
著者Pidugu, L.S, Pozharski, E, Drohat, A.C.
登録日2020-12-10
公開日2021-11-10
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.68 Å)
主引用文献Structural Insights into the Mechanism of Base Excision by MBD4.
J.Mol.Biol., 433, 2021
5K9L
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BU of 5k9l by Molmil
Beclin 2 CCD N187L mutant homodimer
分子名称: Beclin-2
著者Su, M, Sinha, S.
登録日2016-06-01
公開日2017-03-08
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献BECN2 interacts with ATG14 through a metastable coiled-coil to mediate autophagy.
Protein Sci., 26, 2017

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