PDB: 663 件ウェブページステータス検索Chemie searchBIRD

---

3BKI	Crystal Structure of the GluR2 ligand binding core (S1S2J) in complex with FQX at 1.87 Angstroms 分子名称: Glutamate receptor 2, [1,2,5]oxadiazolo[3,4-g]quinoxaline-6,7(5H,8H)-dione 1-oxide 著者 Cruz, L, Estebanez-Perpina, E, Pfaff, S, Borngraeber, S, Bao, N, Fletterick, R, England, P. 登録日 2007-12-06 公開日 2008-09-16 最終更新日 2019-09-04 実験手法 X-RAY DIFFRACTION (1.87 Å) 主引用文献 6-Azido-7-nitro-1,4-dihydroquinoxaline-2,3-dione (ANQX) forms an irreversible bond to the active site of the GluR2 AMPA receptor. J.Med.Chem., 51, 2008
3C31	Crystal structure of GluR5 ligand-binding core in complex with lithium at 1.49 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.49 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
3C34	Crystal structure of GluR5 ligand-binding core in complex with rubidium at 1.82 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.82 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
3C36	Crystal structure of GluR5 ligand-binding core in complex with ammonium ions at 1.68 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, AMMONIUM ION, CHLORIDE ION, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.68 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
3C33	Crystal structure of GluR5 ligand-binding core in complex with potassium at 1.78 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.72 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
3C32	Crystal structure of GluR5 ligand-binding core in complex with sodium at 1.72 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CHLORIDE ION, GLUTAMATE RECEPTOR, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.72 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
3C35	Crystal structure of GluR5 ligand-binding core in complex with cesium at 1.97 Angstrom resolution 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, CESIUM ION, CHLORIDE ION, ... 著者 Mayer, M.L. 登録日 2008-01-27 公開日 2008-06-17 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.97 Å) 主引用文献 Molecular basis of kainate receptor modulation by sodium. Neuron, 58, 2008
2ZNU	Crystal structure of the ligand-binding core of the human ionotropic glutamate receptor, GluR5, in complex with a novel selective agonist, neodysiherbaine A 分子名称: (2R,3aR,6R,7R,7aR)-2-[(2S)-2-amino-2-carboxyethyl]-6,7-dihydroxyhexahydro-2H-furo[3,2-b]pyran-2-carboxylic acid, BETA-MERCAPTOETHANOL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2008-05-01 公開日 2009-05-05 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.8 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
2ZNT	Crystal structure of the ligand-binding core of the human ionotropic glutamate receptor, GluR5, in complex with a novel selective agonist, dysiherbaine 分子名称: (2R,3aR,6S,7R,7aR)-2-[(2S)-2-amino-2-carboxyethyl]-6-hydroxy-7-(methylamino)hexahydro-2H-furo[3,2-b]pyran-2-carboxylic acid, BETA-MERCAPTOETHANOL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2008-05-01 公開日 2009-05-05 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.6 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
2ZNS	Crystal structure of the ligand-binding core of the human ionotropic glutamate receptor, GluR5, in complex with glutamate 分子名称: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 1 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2008-05-01 公開日 2009-05-05 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (2 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3DLN	Crystal structure of the binding domain of the AMPA subunit GluR3 bound to glutamate 分子名称: GLUTAMIC ACID, Glutamate receptor 3, ZINC ION 著者 Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. 登録日 2008-06-27 公開日 2008-11-25 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.91 Å) 主引用文献 Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
3DP6	Crystal structure of the binding domain of the AMPA subunit GluR2 bound to glutamate 分子名称: GLUTAMIC ACID, Glutamate receptor 2, ZINC ION 著者 Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. 登録日 2008-07-07 公開日 2008-11-25 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (1.55 Å) 主引用文献 Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
3DP4	Crystal structure of the binding domain of the AMPA subunit GluR3 bound to AMPA 分子名称: (S)-ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID, Glutamate receptor 3, ZINC ION 著者 Ahmed, A.H, Wang, Q, Sondermann, H, Oswald, R.E. 登録日 2008-07-07 公開日 2008-11-25 最終更新日 2023-08-30 実験手法 X-RAY DIFFRACTION (2.11 Å) 主引用文献 Structure of the S1S2 glutamate binding domain of GLuR3. Proteins, 75, 2008
3EN3	Crystal Structure of the GluR4 Ligand-Binding domain in complex with kainate 分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, Glutamate receptor 4,Glutamate receptor 著者 Gill, A, Madden, D.R. 登録日 2008-09-25 公開日 2009-05-19 最終更新日 2017-07-26 実験手法 X-RAY DIFFRACTION (2.43 Å) 主引用文献 Correlating AMPA receptor activation and cleft closure across subunits: crystal structures of the GluR4 ligand-binding domain in complex with full and partial agonists Biochemistry, 47, 2008
3EPE	Crystal Structure of the GluR4 Ligand-Binding domain in complex with glutamate 分子名称: GLUTAMIC ACID, Glutamate receptor 4,Glutamate receptor 著者 Gill, A, Madden, D.R. 登録日 2008-09-29 公開日 2009-05-19 最終更新日 2023-09-06 実験手法 X-RAY DIFFRACTION (1.85 Å) 主引用文献 Correlating AMPA receptor activation and cleft closure across subunits: crystal structures of the GluR4 ligand-binding domain in complex with full and partial agonists Biochemistry, 47, 2008
3FAS	X-ray structure of iGluR4 flip ligand-binding core (S1S2) in complex with (S)-glutamate at 1.40A resolution 分子名称: GLUTAMIC ACID, GLYCEROL, Glutamate receptor 4, ... 著者 Kasper, C, Frydenvang, K, Naur, P, Gajhede, M, Kastrup, J.S. 登録日 2008-11-18 公開日 2008-12-09 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.4 Å) 主引用文献 Molecular mechanism of agonist recognition by the ligand-binding core of the ionotropic glutamate receptor 4 Febs Lett., 582, 2008
3FAT	X-ray structure of iGluR4 flip ligand-binding core (S1S2) in complex with (S)-AMPA at 1.90A resolution 分子名称: (S)-ALPHA-AMINO-3-HYDROXY-5-METHYL-4-ISOXAZOLEPROPIONIC ACID, ACETIC ACID, GLYCEROL, ... 著者 Kasper, C, Frydenvang, K, Naur, P, Gajhede, M, Kastrup, J.S. 登録日 2008-11-18 公開日 2008-12-09 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.9 Å) 主引用文献 Molecular mechanism of agonist recognition by the ligand-binding core of the ionotropic glutamate receptor 4 Febs Lett., 582, 2008
3FVG	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with MSVIII-19 in space group P1 分子名称: (2R,3aR,7aR)-2-[(2S)-2-amino-3-hydroxy-3-oxo-propyl]-3,3a,5,6,7,7a-hexahydrofuro[4,5-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-15 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3FUZ	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with L-glutamate in space group P1 分子名称: GLUTAMIC ACID, Glutamate receptor, ionotropic kainate 1, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-15 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.65 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3FVK	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with 8-deoxy-neodysiherbaine A in space group P1 分子名称: (2R,3aR,6S,7aR)-2-[(2S)-2-amino-3-hydroxy-3-oxo-propyl]-6-hydroxy-3,3a,5,6,7,7a-hexahydrofuro[4,5-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-15 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3FV1	Crystal Structure of the human glutamate receptor, GluR5, ligand-binding core in complex with dysiherbaine in space group P1 分子名称: (2R,3aR,6S,7R,7aR)-2-[(2S)-2-amino-2-carboxyethyl]-6-hydroxy-7-(methylamino)hexahydro-2H-furo[3,2-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-15 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3FV2	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with neodysiherbaine A in space group P1 分子名称: (2R,3aR,6R,7R,7aR)-2-[(2S)-2-amino-2-carboxyethyl]-6,7-dihydroxyhexahydro-2H-furo[3,2-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-15 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3FVO	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with 8-epi-neodysiherbaine A in space group P1 分子名称: (2R,3aR,6R,7S,7aR)-2-[(2S)-2-amino-3-hydroxy-3-oxo-propyl]-6,7-dihydroxy-3,3a,5,6,7,7a-hexahydrofuro[4,5-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-16 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Crystal Structures of Human GluR5 Ligand-Binding Core in Complexes with Novel Marine-Derived Toxins, Dysiherbaine and Neodysiherbaine A, and Their Analogues To be Published
3FVN	Crystal structure of the human glutamate receptor, GluR5, ligand-binding core in complex with 9-deoxy-neodysiherbaine A in space group P1 分子名称: (2R,3aR,7R,7aR)-2-[(2S)-2-amino-3-hydroxy-3-oxo-propyl]-7-hydroxy-3,3a,5,6,7,7a-hexahydrofuro[4,5-b]pyran-2-carboxylic acid, GLYCEROL, Glutamate receptor, ... 著者 Unno, M, Sasaki, M, Ikeda-Saito, M. 登録日 2009-01-16 公開日 2010-01-19 最終更新日 2023-11-01 実験手法 X-RAY DIFFRACTION (1.5 Å) 主引用文献 Binding and Selectivity of the Marine Toxin Neodysiherbaine A and Its Synthetic Analogues to GluK1 and GluK2 Kainate Receptors. J.Mol.Biol., 413, 2011
3G3G	Crystal structure of the GluR6 ligand binding domain dimer K665R mutant with glutamate and NaCl at 1.3 Angstrom resolution 分子名称: CHLORIDE ION, GLUTAMIC ACID, Glutamate receptor, ... 著者 Chaudhry, C, Mayer, M.L. 登録日 2009-02-02 公開日 2009-06-02 最終更新日 2021-10-20 実験手法 X-RAY DIFFRACTION (1.303 Å) 主引用文献 Stability of ligand-binding domain dimer assembly controls kainate receptor desensitization. Embo J., 28, 2009

<12345678910111213141516>