Loading
PDBj
メニューPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

2CLD
DownloadVisualize
BU of 2cld by Molmil
CRYSTAL STRUCTURE ANALYSIS OF A FLUORESCENT FORM OF H-RAS P21 IN COMPLEX WITH GDP (2)
分子名称: GTPASE HRAS, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION
著者Klink, B.U, Goody, R.S, Scheidig, A.J.
登録日2006-04-27
公開日2006-05-31
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.22 Å)
主引用文献A Newly Designed Microspectrofluorometer for Kinetic Studies on Protein Crystals in Combination with X-Ray Diffraction
Biophys.J., 91, 2006
1J8A
DownloadVisualize
BU of 1j8a by Molmil
CRYSTAL STRUCTURE OF BENZAMIDINE INHIBITED BOVINE PANCREATIC TRYPSIN AT 105K TO 1.21A RESOLUTION FROM LABORATORY SOURCE WITH HIGH NUMBER OF WATERS MODELLED
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, BENZAMIDINE, CALCIUM ION, ...
著者Cuesta-Seijo, J.A, Garcia-Granda, S.
登録日2001-05-21
公開日2001-09-12
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.21 Å)
主引用文献Trypsin as a model for high resolution X-ray diffraction in proteins.
BOL.R.SOC.HIST.NAT.SEC.GEOL., 97, 2002
2CN8
DownloadVisualize
BU of 2cn8 by Molmil
Crystal structure of human Chk2 in complex with debromohymenialdisine
分子名称: DEBROMOHYMENIALDISINE, MAGNESIUM ION, NITRATE ION, ...
著者Oliver, A.W, Pearl, L.H.
登録日2006-05-18
公開日2006-06-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Trans-Activation of the DNA-Damage Signalling Protein Kinase Chk2 by T-Loop Exchange
Embo J., 25, 2006
1J8K
DownloadVisualize
BU of 1j8k by Molmil
NMR STRUCTURE OF THE FIBRONECTIN EDA DOMAIN, NMR, 20 STRUCTURES
分子名称: FIBRONECTIN
著者Niimi, T, Osawa, M, Yamaji, N, Yasunaga, K, Sakashita, H, Mase, T, Tanaka, A, Fujita, S.
登録日2001-05-22
公開日2002-02-06
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献NMR structure of human fibronectin EDA.
J.Biomol.NMR, 21, 2001
1WTN
DownloadVisualize
BU of 1wtn by Molmil
The structure of HEW Lysozyme Orthorhombic Crystal Growth under a High Magnetic Field
分子名称: CHLORIDE ION, Lysozyme C
著者Saijo, S, Yamada, Y, Sato, T, Tanaka, N, Matsui, T, Sazaki, G, Nakajima, K, Matsuura, Y.
登録日2004-11-25
公開日2004-12-14
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.13 Å)
主引用文献Structural consequences of hen egg-white lysozyme orthorhombic crystal growth in a high magnetic field: validation of X-ray diffraction intensity, conformational energy searching and quantitative analysis of B factors and mosaicity.
Acta Crystallogr.,Sect.D, 61, 2005
1WHW
DownloadVisualize
BU of 1whw by Molmil
Solution structure of the N-terminal RNA binding domain from hypothetical protein BAB23448
分子名称: hypothetical protein RIKEN CDNA 1200009A02
著者Nagata, T, Muto, Y, Inoue, M, Kigawa, T, Terada, T, Shirouzu, M, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2004-05-28
公開日2004-11-28
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the N-terminal RNA binding domain from hypothetical protein BAB23448
To be Published
2C8Q
DownloadVisualize
BU of 2c8q by Molmil
insuline(1sec) and UV laser excited fluorescence
分子名称: INSULIN A CHAIN, INSULIN B CHAIN
著者Vernede, X, Lavault, B, Ohana, J, Nurizzo, D, Joly, J, Jacquamet, L, Felisaz, F, Cipriani, F, Bourgeois, D.
登録日2005-12-06
公開日2006-03-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Uv Laser-Excited Fluorescence as a Tool for the Visualization of Protein Crystals Mounted in Loops.
Acta Crystallogr.,Sect.D, 62, 2006
2CL7
DownloadVisualize
BU of 2cl7 by Molmil
CRYSTAL STRUCTURE ANALYSIS OF A FLUORESCENT FORM OF H-RAS P21 IN COMPLEX WITH GTP
分子名称: GTPASE HRAS, GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ...
著者Klink, B.U, Goody, R.S, Scheidig, A.J.
登録日2006-04-26
公開日2006-05-24
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献A Newly Designed Microspectrofluorometer for Kinetic Studies on Protein Crystals in Combination with X-Ray Diffraction.
Biophys.J., 91, 2006
1IFC
DownloadVisualize
BU of 1ifc by Molmil
REFINEMENT OF THE STRUCTURE OF RECOMBINANT RAT INTESTINAL FATTY ACID-BINDING APOPROTEIN AT 1.2 ANGSTROMS RESOLUTION
分子名称: INTESTINAL FATTY ACID BINDING PROTEIN
著者Scapin, G, Gordon, J.I, Sacchettini, J.C.
登録日1991-12-19
公開日1994-01-31
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.19 Å)
主引用文献Refinement of the structure of recombinant rat intestinal fatty acid-binding apoprotein at 1.2-A resolution.
J.Biol.Chem., 267, 1992
1IOQ
DownloadVisualize
BU of 1ioq by Molmil
STABILIZATION OF HEN EGG WHITE LYSOZYME BY A CAVITY-FILLING MUTATION
分子名称: LYSOZYME C
著者Ohmura, T, Ueda, T, Ootsuka, K, Saito, M, Imoto, T.
登録日2001-03-28
公開日2001-04-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.79 Å)
主引用文献Stabilization of hen egg white lysozyme by a cavity-filling mutation.
Protein Sci., 10, 2001
1IOS
DownloadVisualize
BU of 1ios by Molmil
STABILIZATION OF HEN EGG WHITE LYSOZYME BY A CAVITY-FILLING MUTATION
分子名称: LYSOZYME C
著者Ohmura, T, Ueda, T, Ootsuka, K, Saito, M, Imoto, T.
登録日2001-03-28
公開日2001-04-11
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.76 Å)
主引用文献Stabilization of hen egg white lysozyme by a cavity-filling mutation.
Protein Sci., 10, 2001
2CN5
DownloadVisualize
BU of 2cn5 by Molmil
Crystal structure of human Chk2 in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MAGNESIUM ION, ...
著者Oliver, A.W, Pearl, L.H.
登録日2006-05-18
公開日2006-06-28
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献Trans-Activation of the DNA-Damage Signalling Protein Kinase Chk2 by T-Loop Exchange
Embo J., 25, 2006
2CGX
DownloadVisualize
BU of 2cgx by Molmil
Identification of chemically diverse Chk1 inhibitors by receptor- based virtual screening
分子名称: 2-[(6-AMINO-7H-PURIN-8-YL)THIO]ACETAMIDE, SERINE/THREONINE-PROTEIN KINASE CHK1
著者Foloppe, N, Fisher, L.M, Howes, R, Potter, A, Robertson, A.G.S, Surgenor, A.E.
登録日2006-03-09
公開日2006-04-05
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Identification of Chemically Diverse Chk1 Inhibitors by Receptor-Based Virtual Screening.
Bioorg.Med.Chem., 14, 2006
1WWD
DownloadVisualize
BU of 1wwd by Molmil
NMR structure determined for MLV NC complex with RNA sequence AACAGU
分子名称: 5'-R(P*AP*AP*CP*AP*GP*U)-3', Nucleoprotein p10, ZINC ION
著者Dey, A, York, D, Smalls-Mantey, A, Summers, M.F.
登録日2005-01-05
公開日2005-03-22
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Composition and sequence-dependent binding of RNA to the nucleocapsid protein of Moloney murine leukemia virus(,)
Biochemistry, 44, 2005
2CLX
DownloadVisualize
BU of 2clx by Molmil
4-Arylazo-3,5-diamino-1H-pyrazole CDK Inhibitors: SAR Study, Crystal Structure in Complex with CDK2, Selectivity, and Cellular Effects
分子名称: 4-[(E)-(3,5-DIAMINO-1H-PYRAZOL-4-YL)DIAZENYL]PHENOL, CELL DIVISION PROTEIN KINASE 2
著者Krystof, V, Cankar, P, Frysova, I, Slouka, J, Kontopidis, G, Dzubak, P, Hajduch, M, Deazevedo, W.F, Paprskarova, M, Orsag, M, Rolcik, J, Latr, A, Fischer, P.M, Strnad, M.
登録日2006-05-02
公開日2006-11-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献4-Arylazo-3,5-Diamino-1H-Pyrazole Cdk Inhibitors: Sar Study, Crystal Structure in Complex with Cdk2, Selectivity, and Cellular Effects
J.Med.Chem., 49, 2006
2YCQ
DownloadVisualize
BU of 2ycq by Molmil
Crystal structure of checkpoint kinase 2 in complex with inhibitor PV1115
分子名称: N-{4-[(1E)-N-1H-IMIDAZOL-2-YLETHANEHYDRAZONOYL]PHENYL}-7-NITRO-1H-INDOLE-2-CARBOXAMIDE, NITRATE ION, SERINE/THREONINE-PROTEIN KINASE CHK2
著者Lountos, G.T, Jobson, A.G, Tropea, J.E, Self, C.R, Pommier, Y, Shoemaker, R.H, Zhang, G, Waugh, D.S.
登録日2011-03-16
公開日2011-11-16
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献Structural Characterization of Inhibitor Complexes with Checkpoint Kinase 2 (Chk2), a Drug Target for Cancer Therapy.
J.Struct.Biol., 176, 2011
2CKE
DownloadVisualize
BU of 2cke by Molmil
Human death-associated DRP-1 kinase in complex with inhibitor
分子名称: DEATH-ASSOCIATED PROTEIN KINASE 2, N-(2-AMINOETHYL)ISOQUINOLINE-5-SULFONAMIDE
著者Kursula, P, Wilmanns, M.
登録日2006-04-18
公開日2007-05-15
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Crystal Structure of Human Drp-1 Complexed with an Inhibitor
To be Published
2CMY
DownloadVisualize
BU of 2cmy by Molmil
Crystal complex between bovine trypsin and Veronica hederifolia trypsin inhibitor
分子名称: CALCIUM ION, CATIONIC TRYPSIN, GLYCEROL, ...
著者Conners, R, Yardley, J.L, Konarev, A, Shewry, P, Brady, R.L.
登録日2006-05-16
公開日2007-05-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献An Unusual Helix-Turn-Helix Protease Inhibitory Motif in a Novel Trypsin Inhibitor from Seeds of Veronica (Veronica Hederifolia L.).
J.Biol.Chem., 282, 2007
2YM4
DownloadVisualize
BU of 2ym4 by Molmil
Crystal structure of checkpoint kinase 1 (Chk1) in complex with inhibitors
分子名称: 1,2-ETHANEDIOL, SERINE/THREONINE-PROTEIN KINASE CHK1, ethyl 4-[(2R)-2-(aminomethyl)morpholin-4-yl]-3-(3-cyanophenyl)-1H-pyrazolo[3,4-b]pyridine-5-carboxylate
著者Reader, J.C, Matthews, T.P, Klair, S, Cheung, K.M.J, Scanlon, J, Proisy, N, Addison, G, Ellard, J, Piton, N, Taylor, S, Cherry, M, Fisher, M, Boxall, K, Burns, S, Walton, M.I, Westwood, I.M, Hayes, A, Eve, P, Valenti, M, Brandon, A.H, Box, G, vanMontfort, R.L.M, Williams, D.H, Aherne, G.W, Raynaud, F.I, Eccles, S.A, Garrett, M.D, Collins, I.
登録日2011-06-06
公開日2012-01-11
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structure-Guided Evolution of Potent and Selective Chk1 Inhibitors Through Scaffold Morphing.
J.Med.Chem., 54, 2011
1IWK
DownloadVisualize
BU of 1iwk by Molmil
Putidaredoxin-Binding Stablilizes an Active Conformer of Cytochrome P450cam in its Reduced State; Crystal Structure of Mutant(112K) Cytochrome P450cam
分子名称: CYTOCHROME P450-CAM, PROTOPORPHYRIN IX CONTAINING FE
著者Nagano, S, Shimada, H, Tarumi, A, Hishiki, T, Kimata-Ariga, Y, Egawa, T, Park, S.-Y, Adachi, S, Shiro, Y, Ishimura, Y, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2002-05-15
公開日2002-06-05
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Infrared spectroscopic and mutational studies on putidaredoxin-induced conformational changes in ferrous CO-P450cam
Biochemistry, 42, 2003
1IWY
DownloadVisualize
BU of 1iwy by Molmil
Crystal Structure Analysis of Human lysozyme at 170K.
分子名称: CHLORIDE ION, LYSOZYME C
著者Joti, Y, Nakasako, M, Kidera, A, Go, N.
登録日2002-06-03
公開日2002-09-04
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Nonlinear temperature dependence of the crystal structure of lysozyme: correlation between coordinate shifts and thermal factors.
Acta Crystallogr.,Sect.D, 58, 2002
2BD5
DownloadVisualize
BU of 2bd5 by Molmil
Porcine pancreatic elastase complexed with beta-casomorphin-7 and Lys-Ser at pH 5 and immersed in pH 9 buffer for 30 seconds
分子名称: CALCIUM ION, Elastase-1, LYSINE, ...
著者Liu, B, Schofield, C.J, Wilmouth, R.C.
登録日2005-10-20
公開日2006-05-30
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structural analyses on intermediates in serine protease catalysis
J.Biol.Chem., 281, 2006
1WVY
DownloadVisualize
BU of 1wvy by Molmil
Crystal structures of kinase domain of DAP kinase in complex with small molecular inhibitors
分子名称: Death-associated protein kinase 1, STAUROSPORINE
著者Ueda, Y, Ogata, H, Yamakawa, A, Higuchi, Y.
登録日2004-12-27
公開日2006-04-11
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Complex structure of kinase domain of DAP kinase with Staurosporine
To be Published
1J7Y
DownloadVisualize
BU of 1j7y by Molmil
Crystal structure of partially ligated mutant of HbA
分子名称: CARBON MONOXIDE, Hemoglobin, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Miele, A.E, Draghi, F, Arcovito, A, Bellelli, A, Brunori, M, Travaglini-Allocatelli, C, Vallone, B.
登録日2001-05-19
公開日2002-02-27
最終更新日2023-08-16
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Control of heme reactivity by diffusion: structural basis and functional characterization in hemoglobin mutants.
Biochemistry, 40, 2001
8JPF
DownloadVisualize
BU of 8jpf by Molmil
Focused refiment structure of NTSR1 in NTSR1-GRK2-Galpha(q) complexes
分子名称: 2-[{2-(1-fluorocyclopropyl)-4-[4-(2-methoxyphenyl)piperidin-1-yl]quinazolin-6-yl}(methyl)amino]ethan-1-ol, NTS, Neurotensin receptor type 1
著者Duan, J, Liu, H, Zhao, F, Yuan, Q, Ji, Y, Xu, H.E.
登録日2023-06-11
公開日2023-08-09
最終更新日2023-08-30
実験手法ELECTRON MICROSCOPY (3.02 Å)
主引用文献GPCR activation and GRK2 assembly by a biased intracellular agonist.
Nature, 620, 2023

223532

件を2024-08-07に公開中

PDB statisticsPDBj update infoContact PDBjnumon