7E3U
| Crystal structure of the Pseudomonas aeruginosa dihydropyrimidinase complexed with 5-AU | 分子名称: | 5-AMINO-1H-PYRIMIDINE-2,4-DIONE, D-hydantoinase/dihydropyrimidinase, ZINC ION | 著者 | Yang, Y.C, Luo, R.H, Huang, Y.H, Huang, C.Y, Lin, E.S. | 登録日 | 2021-02-09 | 公開日 | 2022-02-16 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (2.159 Å) | 主引用文献 | Molecular Insights into How the Dimetal Center in Dihydropyrimidinase Can Bind the Thymine Antagonist 5-Aminouracil: A Different Binding Mode from the Anticancer Drug 5-Fluorouracil. Bioinorg Chem Appl, 2022, 2022
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3NUC
| STAPHLOCOCCAL NUCLEASE, 1-N-PROPANE THIOL DISULFIDE TO V23C VARIANT | 分子名称: | CALCIUM ION, STAPHYLOCOCCAL NUCLEASE, THYMIDINE-3',5'-DIPHOSPHATE | 著者 | Wynn, R, Harkins, P.C, Richards, F.M, Fox, R.O. | 登録日 | 1997-12-06 | 公開日 | 1998-03-18 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Mobile unnatural amino acid side chains in the core of staphylococcal nuclease. Protein Sci., 5, 1996
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4BP9
| Oligopeptidase B from Trypanosoma brucei with covalently bound antipain - closed form | 分子名称: | ANTIPAIN, OLIGOPEPTIDASSE B | 著者 | Canning, P, Rea, D, Morty, R, Fulop, V. | 登録日 | 2013-05-23 | 公開日 | 2014-02-12 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2.85 Å) | 主引用文献 | Crystal Structures of Trypanosoma Brucei Oligopeptidase B Broaden the Paradigm of Catalytic Regulation in Prolyl Oligopeptidase Family Enzymes. Plos One, 8, 2013
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3PPM
| Crystal Structure of a Noncovalently Bound alpha-Ketoheterocycle Inhibitor (Phenhexyl/Oxadiazole/Pyridine) to a Humanized Variant of Fatty Acid Amide Hydrolase | 分子名称: | 1-DODECANOL, 7-phenyl-1-[5-(pyridin-2-yl)-1,3,4-oxadiazol-2-yl]heptan-1-one, CHLORIDE ION, ... | 著者 | Mileni, M, Han, G.W, Boger, D.L, Stevens, R.C. | 登録日 | 2010-11-24 | 公開日 | 2011-11-09 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Fluoride-mediated capture of a noncovalent bound state of a reversible covalent enzyme inhibitor: X-ray crystallographic analysis of an exceptionally potent alpha-ketoheterocycle inhibitor of fatty acid amide hydrolase. J.Am.Chem.Soc., 133, 2011
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3Q2D
| Optimization of the in silico designed Kemp eliminase KE70 by computational design and directed evolution | 分子名称: | 5-nitro-1H-benzotriazole, Deoxyribose phosphate aldolase | 著者 | Khersonsky, O, Rothlisberge, D, Wollacott, A.M, Murphy, P, Dym, O, Albeck, S, Kiss, G, Houk, K.N, Baker, D, Tawfik, D.S, Israel Structural Proteomics Center (ISPC) | 登録日 | 2010-12-20 | 公開日 | 2011-02-09 | 最終更新日 | 2023-11-01 | 実験手法 | X-RAY DIFFRACTION (2.19 Å) | 主引用文献 | Optimization of the in-silico-designed kemp eliminase KE70 by computational design and directed evolution J.Mol.Biol., 407, 2011
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3PTE
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3P5S
| Structural insights into the catalytic mechanism of CD38: Evidence for a conformationally flexible covalent enzyme-substrate complex | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CD38 molecule, SULFATE ION, ... | 著者 | Egea, P.F, Muller-Stauffler, H, Kohn, I, Cakou-Kefir, C, Stroud, R.M, Kellenberburger, E, Schuber, F. | 登録日 | 2010-10-10 | 公開日 | 2011-10-19 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Insights into the mechanism of bovine CD38/NAD+glycohydrolase from the X-ray structures of its Michaelis complex and covalently-trapped intermediates. Plos One, 7, 2012
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3PCD
| PROTOCATECHUATE 3,4-DIOXYGENASE Y447H MUTANT | 分子名称: | BETA-MERCAPTOETHANOL, CARBONATE ION, FE (III) ION, ... | 著者 | Orville, A.M, Lipscomb, J.D, Ohlendorf, D.H. | 登録日 | 1997-11-24 | 公開日 | 1998-05-27 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The axial tyrosinate Fe3+ ligand in protocatechuate 3,4-dioxygenase influences substrate binding and product release: evidence for new reaction cycle intermediates. Biochemistry, 37, 1998
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4FO2
| Heat-labile enterotoxin LT-IIb-B5(T13I) mutant | 分子名称: | ACETATE ION, Heat-labile enterotoxin IIB, B chain, ... | 著者 | Cody, V, Pace, J, Nawar, H, Liang, S, Connell, T, Hajishengallis, G. | 登録日 | 2012-06-20 | 公開日 | 2012-11-21 | 最終更新日 | 2023-09-13 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structure-activity correlations of variant forms of the B pentamer of Escherichia coli type II heat-labile enterotoxin LT-IIb with Toll-like receptor 2 binding. Acta Crystallogr.,Sect.D, 68, 2012
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3M9Z
| Crystal Structure of extracellular domain of mouse NKR-P1A | 分子名称: | Killer cell lectin-like receptor subfamily B member 1A, PHOSPHATE ION | 著者 | Kolenko, P, Rozbesky, D, Bezouska, K, Hasek, J, Dohnalek, J. | 登録日 | 2010-03-23 | 公開日 | 2011-04-06 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Molecular architecture of mouse activating NKR-P1 receptors. J.Struct.Biol., 175, 2011
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3MAT
| E.COLI METHIONINE AMINOPEPTIDASE TRANSITION-STATE INHIBITOR COMPLEX | 分子名称: | COBALT (II) ION, METHIONINE AMINOPEPTIDASE, SODIUM ION, ... | 著者 | Lowther, W.T, Orville, A.M, Madden, D.T, Lim, S, Rich, D.H, Matthews, B.W. | 登録日 | 1999-03-29 | 公開日 | 1999-06-18 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Escherichia coli methionine aminopeptidase: implications of crystallographic analyses of the native, mutant, and inhibited enzymes for the mechanism of catalysis. Biochemistry, 38, 1999
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4ER2
| The active site of aspartic proteinases | 分子名称: | ENDOTHIAPEPSIN, PEPSTATIN, SULFATE ION | 著者 | Bailey, D, Veerapandian, B, Cooper, J.B, Blundell, T.L. | 登録日 | 1990-10-20 | 公開日 | 1991-01-15 | 最終更新日 | 2017-11-29 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | The active site of aspartic proteinases FEBS Lett., 174, 1984
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4FIT
| FHIT-APO | 分子名称: | FRAGILE HISTIDINE TRIAD PROTEIN | 著者 | Lima, C.D, Klein, M.G, Hendrickson, W.A. | 登録日 | 1997-09-25 | 公開日 | 1998-03-25 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structure-based analysis of catalysis and substrate definition in the HIT protein family. Science, 278, 1997
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4GEP
| SULFITE REDUCTASE HEMOPROTEIN CYANIDE COMPLEX REDUCED WITH CRII EDTA | 分子名称: | CYANIDE ION, IRON/SULFUR CLUSTER, POTASSIUM ION, ... | 著者 | Crane, B.R, Getzoff, E.D. | 登録日 | 1997-07-10 | 公開日 | 1998-01-14 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Probing the catalytic mechanism of sulfite reductase by X-ray crystallography: structures of the Escherichia coli hemoprotein in complex with substrates, inhibitors, intermediates, and products. Biochemistry, 36, 1997
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4G93
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2VKA
| Site-Directed Mutagenesis of the Catalytic Tryptophan Environment in Pleurotus eryngii Versatile Peroxidase | 分子名称: | CALCIUM ION, GLYCEROL, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Ruiz-Duenas, F.J, Morales, M, Mate, M.J, Romero, A, Martinez, M.J, Smith, A, Martinez, A.T. | 登録日 | 2007-12-18 | 公開日 | 2008-01-29 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Site-Directed Mutagenesis of the Catalytic Tryptophan Environment in Pleurotus Eryngii Versatile Peroxidase Biochemistry, 47, 2008
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2V7E
| Crystal structure of coactivator-associated arginine methyltransferase 1 (CARM1), unliganded | 分子名称: | HISTONE-ARGININE METHYLTRANSFERASE CARM1, MERCURY (II) ION | 著者 | Yue, W.W, Hassler, M, Roe, S.M, Thompson-Vale, V, Pearl, L.H. | 登録日 | 2007-07-30 | 公開日 | 2007-10-02 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Insights Into Histone Code Syntax from Structural and Biochemical Studies of Carm1 Methyltransferase Embo J., 26, 2007
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2V74
| Crystal structure of coactivator-associated arginine methyltransferase 1 (CARM1), in complex with S-adenosyl-homocysteine | 分子名称: | HISTONE-ARGININE METHYLTRANSFERASE CARM1, S-ADENOSYL-L-HOMOCYSTEINE | 著者 | Yue, W.W, Hassler, M, Roe, S.M, Thompson-Vale, V, Pearl, L.H. | 登録日 | 2007-07-26 | 公開日 | 2007-10-02 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Insights Into Histone Code Syntax from Structural and Biochemical Studies of Carm1 Methyltransferase Embo J., 26, 2007
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7WG7
| Acidic Omicron Spike Trimer | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein, ... | 著者 | Cui, Z. | 登録日 | 2021-12-28 | 公開日 | 2022-06-22 | 実験手法 | ELECTRON MICROSCOPY (4 Å) | 主引用文献 | Structural and functional characterizations of infectivity and immune evasion of SARS-CoV-2 Omicron. Cell, 185, 2022
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7WGC
| Neutral Omicron Spike Trimer in complex with ACE2. | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, Processed angiotensin-converting enzyme 2, Spike glycoprotein | 著者 | Cui, Z. | 登録日 | 2021-12-28 | 公開日 | 2022-06-22 | 最終更新日 | 2022-07-13 | 実験手法 | ELECTRON MICROSCOPY (3.6 Å) | 主引用文献 | Structural and functional characterizations of infectivity and immune evasion of SARS-CoV-2 Omicron. Cell, 185, 2022
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7WG9
| Delta Spike Trimer(1 RBD Up) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Cui, Z. | 登録日 | 2021-12-28 | 公開日 | 2022-06-22 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural and functional characterizations of infectivity and immune evasion of SARS-CoV-2 Omicron. Cell, 185, 2022
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1E60
| OXIDIZED DMSO REDUCTASE EXPOSED TO HEPES - Structure II BUFFER | 分子名称: | 2-AMINO-5,6-DIMERCAPTO-7-METHYL-3,7,8A,9-TETRAHYDRO-8-OXA-1,3,9,10-TETRAAZA-ANTHRACEN-4-ONE GUANOSINE DINUCLEOTIDE, Dimethyl sulfoxide/trimethylamine N-oxide reductase, MOLYBDENUM (IV)OXIDE, ... | 著者 | Bailey, S, Bennett, B, Adams, B, Smith, A.T, Bray, R.C. | 登録日 | 2000-08-06 | 公開日 | 2000-08-25 | 最終更新日 | 2024-05-01 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Reversible Dissociation of Thiolate Ligands from Molybdenum in an Enzyme of the Dimethyl Sulfoxide Reductase Family Biochemistry, 39, 2000
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7WGB
| Neutral Omicron Spike Trimer in complex with ACE2 | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Processed angiotensin-converting enzyme 2, ... | 著者 | Cui, Z. | 登録日 | 2021-12-28 | 公開日 | 2022-06-22 | 実験手法 | ELECTRON MICROSCOPY (3.5 Å) | 主引用文献 | Structural and functional characterizations of infectivity and immune evasion of SARS-CoV-2 Omicron. Cell, 185, 2022
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2VKL
| X-ray crystal structure of the intracellular Chorismate mutase from Mycobactrerium Tuberculosis in complex with malate | 分子名称: | D-MALATE, RV0948C/MT0975 | 著者 | Okvist, M, Roderer, K, Sasso, S, Kast, P, Krengel, U. | 登録日 | 2007-12-20 | 公開日 | 2008-01-15 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Structure and Function of a Complex between Chorismate Mutase and Dahp Synthase: Efficiency Boost for the Junior Partner. Embo J., 28, 2009
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7WG8
| Delta Spike Trimer(3 RBD Down) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Spike glycoprotein | 著者 | Cui, Z. | 登録日 | 2021-12-28 | 公開日 | 2022-06-22 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | Structural and functional characterizations of infectivity and immune evasion of SARS-CoV-2 Omicron. Cell, 185, 2022
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