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1M3C
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Solution structure of a circular form of the N-terminal SH3 domain (E132C, E133G, R191G mutant) from oncogene protein c-Crk
分子名称: Proto-oncogene C-crk
著者Schumann, F.H, Varadan, R, Tayakuniyil, P.P, Hall, J.B, Camarero, J.A, Fushman, D.
登録日2002-06-27
公開日2003-08-05
最終更新日2021-10-27
実験手法SOLUTION NMR
主引用文献Changing protein backbone topology: Structural and dynamic consequences of the backbone cyclization in SH3 domain
To be Published
1LYY
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BU of 1lyy by Molmil
AMYLOIDOGENIC VARIANT (ASP67HIS) OF HUMAN LYSOZYME
分子名称: LYSOZYME
著者Sunde, M, Blake, C.C.F.
登録日1997-01-16
公開日1997-04-01
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Instability, unfolding and aggregation of human lysozyme variants underlying amyloid fibrillogenesis.
Nature, 385, 1997
1LZ8
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LYSOZYME PHASED ON ANOMALOUS SIGNAL OF SULFURS AND CHLORINES
分子名称: CHLORIDE ION, PROTEIN (LYSOZYME), SODIUM ION
著者Dauter, Z, Dauter, M, De La Fortelle, E, Bricogne, G, Sheldrick, G.M.
登録日1999-03-14
公開日1999-05-26
最終更新日2023-12-27
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Can anomalous signal of sulfur become a tool for solving protein crystal structures?
J.Mol.Biol., 289, 1999
1M7Q
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Crystal structure of p38 MAP kinase in complex with a dihydroquinazolinone inhibitor
分子名称: 1-(2,6-DICHLOROPHENYL)-5-(2,4-DIFLUOROPHENYL)-7-PIPERAZIN-1-YL-3,4-DIHYDROQUINAZOLIN-2(1H)-ONE, Mitogen-activated protein kinase 14, SULFATE ION
著者Stelmach, J.E, Liu, L, Patel, S.B, Pivnichny, J.V, Scapin, G, Singh, S, Hop, C.E.C.A, Wang, Z, Cameron, P.M, Nichols, E.A, O'Keefe, S.J, O'Neill, E.A, Schmatz, D.M, Schwartz, C.D, Thompson, C.M, Zaller, D.M, Doherty, J.B.
登録日2002-07-22
公開日2002-12-11
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase.
Bioorg.Med.Chem.Lett., 13, 2003
2FJW
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d(CTTGAATGCATTCAAG) in complex with MMLV RT catalytic fragment
分子名称: 5'-D(*CP*TP*TP*GP*AP*AP*TP*G)-3', 5'-D(P*CP*AP*TP*TP*CP*AP*AP*G)-3', Reverse transcriptase
著者Goodwin, K.D, Georgiadis, M.M.
登録日2006-01-03
公開日2006-06-27
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献A High-Throughput, High-Resolution Strategy for the Study of Site-Selective DNA Binding Agents: Analysis of a "Highly Twisted" Benzimidazole-Diamidine.
J.Am.Chem.Soc., 128, 2006
1M5V
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Transition State Stabilization by a Catalytic RNA
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, RNA HAIRPIN RIBOZYME, ...
著者Rupert, P.B, Massey, A.P, Sigurdsson, S.T, Ferre-D'Amare, A.R.
登録日2002-07-09
公開日2002-10-12
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Transition state stabilization by a catalytic RNA
Science, 298, 2002
2FLE
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Structural analysis of asymmetric inhibitor bound to the HIV-1 Protease V82A mutant
分子名称: (2S,2'S)-N,N'-[(2S,3S,4S,5S)-1-CYCLOHEXYL-3,4-DIHYDROXY-6-PHENYLHEXANE-2,5-DIYL]BIS[3-METHYL-2-({[METHYL(PYRIDIN-2-YLMETHYL)AMINO]CARBONYL}AMINO)BUTANAMIDE], GLYCEROL, pol protein
著者Clemente, J.C, Robbins, A, Dunn, B.M, Sussman, F.
登録日2006-01-05
公開日2007-01-16
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Design, synthesis, evaluation, and crystallographic-based structural studies of HIV-1 protease inhibitors with reduced response to the V82A mutation.
J.Med.Chem., 51, 2008
2FLJ
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BU of 2flj by Molmil
Fatty acid binding protein from locust flight muscle in complex with oleate
分子名称: Fatty acid-binding protein, OLEIC ACID
著者Luecke, C, Qiao, Y, van Moerkerk, H.T.B, Veerkamp, J.H, Hamilton, J.A.
登録日2006-01-06
公開日2006-05-23
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Fatty-acid-binding protein from the flight muscle of Locusta migratoria: evolutionary variations in fatty acid binding.
Biochemistry, 45, 2006
1M6C
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V68N MYOGLOBIN WITH CO
分子名称: CARBON MONOXIDE, PROTEIN (MYOGLOBIN), PROTOPORPHYRIN IX CONTAINING FE
著者Murshudov, G.N, Krzywda, S, Brzozowski, A.M, Jaskolski, M, Scott, E.E, Klizas, S.A, Gibson, Q.H, Olson, J.S, Wilkinson, A.J.
登録日1998-08-12
公開日1998-08-19
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Stabilizing bound O2 in myoglobin by valine68 (E11) to asparagine substitution.
Biochemistry, 37, 1998
1LVY
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PORCINE ELASTASE
分子名称: CALCIUM ION, ELASTASE, SULFATE ION
著者Schiltz, M, Prange, T.
登録日1996-07-20
公開日1997-01-27
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (1.87 Å)
主引用文献High-pressure krypton gas and statistical heavy-atom refinement: a successful combination of tools for macromolecular structure determination.
Acta Crystallogr.,Sect.D, 53, 1997
1MEU
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HIV-1 MUTANT (V82F, I84V) PROTEASE COMPLEXED WITH DMP323
分子名称: HIV-1 PROTEASE, [4-R-(-4-ALPHA,5-ALPHA,6-BETA,7-BETA)]-HEXAHYDRO-5,6-BIS(HYDROXY)-[1,3-BIS([4-HYDROXYMETHYL-PHENYL]METHYL)-4,7-BIS(PHEN YLMETHYL)]-2H-1,3-DIAZEPINONE
著者Ala, P, Chang, C.-H.
登録日1997-04-11
公開日1998-04-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Molecular basis of HIV-1 protease drug resistance: structural analysis of mutant proteases complexed with cyclic urea inhibitors.
Biochemistry, 36, 1997
2FBD
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The crystallographic structure of the digestive lysozyme 1 from Musca domestica at 1.90 Ang.
分子名称: DI(HYDROXYETHYL)ETHER, Lysozyme 1, SULFATE ION
著者Cancado, F.C, Marana, S.R, Barbosa, J.A.R.G.
登録日2005-12-09
公開日2006-12-12
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystallization, data collection and phasing of two digestive lysozymes from Musca domestica.
Acta Crystallogr.,Sect.F, 62, 2006
2FC8
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Solution structure of the RRM_1 domain of NCL protein
分子名称: NCL protein
著者Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI)
登録日2005-12-12
公開日2006-06-12
最終更新日2024-05-29
実験手法SOLUTION NMR
主引用文献Solution structure of the RRM_1 domain of NCL protein
To be published
2FDY
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Microsomal P450 2A6 with the inhibitor Adrithiol bound
分子名称: 4,4'-DIPYRIDYL DISULFIDE, Cytochrome P450 2A6, PROTOPORPHYRIN IX CONTAINING FE, ...
著者Yano, J.K, Stout, C.D, Johnson, E.F.
登録日2005-12-14
公開日2006-11-28
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Synthetic Inhibitors of Cytochrome P-450 2A6: Inhibitory Activity, Difference Spectra, Mechanism of Inhibition, and Protein Cocrystallization.
J.Med.Chem., 49, 2006
2FE6
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P450CAM from Pseudomonas putida reconstituted with manganic protoporphyrin IX
分子名称: Cytochrome P450-cam, POTASSIUM ION, PROTOPORPHYRIN IX CONTAINING MN
著者von Koenig, K, Makris, T.M, Sligar, S.G, Schlichting, I.
登録日2005-12-15
公開日2006-03-14
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献The status of high-valent metal oxo complexes in the P450 cytochromes.
J.Inorg.Biochem., 100, 2006
1MIQ
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Crystal structure of proplasmepsin from the human malarial pathogen Plasmodium vivax
分子名称: plasmepsin
著者Bernstein, N.K, Cherney, M.M, Yowell, C.A, Dame, J.B, James, M.N.
登録日2002-08-23
公開日2002-09-18
最終更新日2018-01-31
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural insights into the activation of P. vivax plasmepsin.
J.Mol.Biol., 329, 2003
2FFB
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The crystal structure of the HlyB-NBD E631Q mutant in complex with ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, Alpha-hemolysin translocation ATP-binding protein hlyB
著者Zaitseva, J, Oswald, C, Jumpertz, T, Jenewein, S, Holland, I.B, Schmitt, L.
登録日2005-12-19
公開日2006-08-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A structural analysis of asymmetry required for catalytic activity of an ABC-ATPase domain dimer.
Embo J., 25, 2006
1M2R
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Crystal structure of 5,8-di-amino-1,4-di-hydroxy-anthraquinone/CK2 kinase complex
分子名称: 5,8-DI-AMINO-1,4-DIHYDROXY-ANTHRAQUINONE, CASEIN kinase II, alpha chain
著者De Moliner, E, Moro, S, Sarno, S, Zagotto, G, Zanotti, G, Pinna, L.A, Battistutta, R.
登録日2002-06-25
公開日2003-06-17
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Inhibition of protein kinase CK2 by anthraquinone-related compounds. A structural insight
J.Biol.Chem., 278, 2003
1M5O
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Transition State Stabilization by a Catalytic RNA
分子名称: CALCIUM ION, RNA SUBSTRATE, RNA HAIRPIN RIBOZYME, ...
著者Rupert, P.B, Massey, A.P, Sigurdsson, S.T, Ferre-D'Amare, A.R.
登録日2002-07-09
公開日2002-10-12
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Transition state stabilization by a catalytic RNA
Science, 298, 2002
1M61
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Crystal structure of the apo SH2 domains of ZAP-70
分子名称: PHOSPHATE ION, TYROSINE-PROTEIN KINASE ZAP-70
著者Folmer, R.H.A, Geschwindner, S, Xue, Y.
登録日2002-07-11
公開日2003-07-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Crystal structure and NMR studies of the apo SH2 domains of ZAP-70: two bikes rather than a tandem
Biochemistry, 41, 2002
2FKA
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Crystal structure of Mg(2+) and BeF(3)(-)-bound CheY in complex with CheZ(200-214) solved from a F432 crystal grown in CAPS (pH 10.5)
分子名称: 3-CYCLOHEXYL-1-PROPYLSULFONIC ACID, BERYLLIUM TRIFLUORIDE ION, C-terminal 15-mer from Chemotaxis protein cheZ, ...
著者Guhaniyogi, J, Robinson, V.L, Stock, A.M.
登録日2006-01-04
公開日2006-05-23
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal Structures of Beryllium Fluoride-free and Beryllium Fluoride-bound CheY in Complex with the Conserved C-terminal Peptide of CheZ Reveal Dual Binding Modes Specific to CheY Conformation.
J.Mol.Biol., 359, 2006
1M7B
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Crystal structure of Rnd3/RhoE: functional implications
分子名称: GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Rnd3/RhoE small GTP-binding protein
著者Fiegen, D, Blumenstein, L, Stege, P, Vetter, I.R, Ahmadian, M.R.
登録日2002-07-19
公開日2002-08-07
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of Rnd3/RhoE: functional implications
FEBS LETT., 525, 2002
1M5A
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Crystal Structure of 2-Co(2+)-Insulin at 1.2A Resolution
分子名称: COBALT (II) ION, INSULIN A CHAIN, INSULIN B CHAIN
著者Nicholson, J.M, Perkins, L.C, Korber, F.C.
登録日2002-07-09
公開日2002-08-14
最終更新日2017-10-11
実験手法X-RAY DIFFRACTION (1.2 Å)
主引用文献The high-resolution structure of hexameric T6 cobalt insulin: A possible pathway for the T to R transition.
Recent Research Developments in Molecular Biology, 3, 2006
1MB3
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CRYSTAL STRUCTURE OF THE RESPONSE REGULATOR DIVK AT PH 8.5 IN COMPLEX WITH MG2+
分子名称: MAGNESIUM ION, cell division response regulator DivK
著者Guillet, V, Ohta, N, Cabantous, S, Newton, A, Samama, J.-P, Structural Proteomics in Europe (SPINE)
登録日2002-08-02
公開日2002-12-04
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.41 Å)
主引用文献Crystallographic and Biochemical Studies of DivK Reveal Novel Features of an Essential Response Regulator in Caulobacter crescentus.
J.Biol.Chem., 277, 2002
1MBD
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X-ray structure of sperm whale deoxymoglobin refined at 1.4A resolution
分子名称: MYOGLOBIN, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION
著者Phillips, S.E.V.
登録日1981-08-27
公開日1982-02-03
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献X-ray structure of sperm whale deoxymoglobin refined at 1.4A resolution
to be published

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