1M3C
| Solution structure of a circular form of the N-terminal SH3 domain (E132C, E133G, R191G mutant) from oncogene protein c-Crk | 分子名称: | Proto-oncogene C-crk | 著者 | Schumann, F.H, Varadan, R, Tayakuniyil, P.P, Hall, J.B, Camarero, J.A, Fushman, D. | 登録日 | 2002-06-27 | 公開日 | 2003-08-05 | 最終更新日 | 2021-10-27 | 実験手法 | SOLUTION NMR | 主引用文献 | Changing protein backbone topology: Structural and dynamic consequences of the backbone cyclization in SH3 domain To be Published
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1LYY
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1LZ8
| LYSOZYME PHASED ON ANOMALOUS SIGNAL OF SULFURS AND CHLORINES | 分子名称: | CHLORIDE ION, PROTEIN (LYSOZYME), SODIUM ION | 著者 | Dauter, Z, Dauter, M, De La Fortelle, E, Bricogne, G, Sheldrick, G.M. | 登録日 | 1999-03-14 | 公開日 | 1999-05-26 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Can anomalous signal of sulfur become a tool for solving protein crystal structures? J.Mol.Biol., 289, 1999
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1M7Q
| Crystal structure of p38 MAP kinase in complex with a dihydroquinazolinone inhibitor | 分子名称: | 1-(2,6-DICHLOROPHENYL)-5-(2,4-DIFLUOROPHENYL)-7-PIPERAZIN-1-YL-3,4-DIHYDROQUINAZOLIN-2(1H)-ONE, Mitogen-activated protein kinase 14, SULFATE ION | 著者 | Stelmach, J.E, Liu, L, Patel, S.B, Pivnichny, J.V, Scapin, G, Singh, S, Hop, C.E.C.A, Wang, Z, Cameron, P.M, Nichols, E.A, O'Keefe, S.J, O'Neill, E.A, Schmatz, D.M, Schwartz, C.D, Thompson, C.M, Zaller, D.M, Doherty, J.B. | 登録日 | 2002-07-22 | 公開日 | 2002-12-11 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Design and synthesis of potent, orally bioavailable dihydroquinazolinone inhibitors of p38 MAP kinase. Bioorg.Med.Chem.Lett., 13, 2003
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2FJW
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1M5V
| Transition State Stabilization by a Catalytic RNA | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, CALCIUM ION, RNA HAIRPIN RIBOZYME, ... | 著者 | Rupert, P.B, Massey, A.P, Sigurdsson, S.T, Ferre-D'Amare, A.R. | 登録日 | 2002-07-09 | 公開日 | 2002-10-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Transition state stabilization by a catalytic RNA Science, 298, 2002
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2FLE
| Structural analysis of asymmetric inhibitor bound to the HIV-1 Protease V82A mutant | 分子名称: | (2S,2'S)-N,N'-[(2S,3S,4S,5S)-1-CYCLOHEXYL-3,4-DIHYDROXY-6-PHENYLHEXANE-2,5-DIYL]BIS[3-METHYL-2-({[METHYL(PYRIDIN-2-YLMETHYL)AMINO]CARBONYL}AMINO)BUTANAMIDE], GLYCEROL, pol protein | 著者 | Clemente, J.C, Robbins, A, Dunn, B.M, Sussman, F. | 登録日 | 2006-01-05 | 公開日 | 2007-01-16 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Design, synthesis, evaluation, and crystallographic-based structural studies of HIV-1 protease inhibitors with reduced response to the V82A mutation. J.Med.Chem., 51, 2008
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2FLJ
| Fatty acid binding protein from locust flight muscle in complex with oleate | 分子名称: | Fatty acid-binding protein, OLEIC ACID | 著者 | Luecke, C, Qiao, Y, van Moerkerk, H.T.B, Veerkamp, J.H, Hamilton, J.A. | 登録日 | 2006-01-06 | 公開日 | 2006-05-23 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Fatty-acid-binding protein from the flight muscle of Locusta migratoria: evolutionary variations in fatty acid binding. Biochemistry, 45, 2006
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1M6C
| V68N MYOGLOBIN WITH CO | 分子名称: | CARBON MONOXIDE, PROTEIN (MYOGLOBIN), PROTOPORPHYRIN IX CONTAINING FE | 著者 | Murshudov, G.N, Krzywda, S, Brzozowski, A.M, Jaskolski, M, Scott, E.E, Klizas, S.A, Gibson, Q.H, Olson, J.S, Wilkinson, A.J. | 登録日 | 1998-08-12 | 公開日 | 1998-08-19 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Stabilizing bound O2 in myoglobin by valine68 (E11) to asparagine substitution. Biochemistry, 37, 1998
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1LVY
| PORCINE ELASTASE | 分子名称: | CALCIUM ION, ELASTASE, SULFATE ION | 著者 | Schiltz, M, Prange, T. | 登録日 | 1996-07-20 | 公開日 | 1997-01-27 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.87 Å) | 主引用文献 | High-pressure krypton gas and statistical heavy-atom refinement: a successful combination of tools for macromolecular structure determination. Acta Crystallogr.,Sect.D, 53, 1997
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1MEU
| HIV-1 MUTANT (V82F, I84V) PROTEASE COMPLEXED WITH DMP323 | 分子名称: | HIV-1 PROTEASE, [4-R-(-4-ALPHA,5-ALPHA,6-BETA,7-BETA)]-HEXAHYDRO-5,6-BIS(HYDROXY)-[1,3-BIS([4-HYDROXYMETHYL-PHENYL]METHYL)-4,7-BIS(PHEN YLMETHYL)]-2H-1,3-DIAZEPINONE | 著者 | Ala, P, Chang, C.-H. | 登録日 | 1997-04-11 | 公開日 | 1998-04-15 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Molecular basis of HIV-1 protease drug resistance: structural analysis of mutant proteases complexed with cyclic urea inhibitors. Biochemistry, 36, 1997
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2FBD
| The crystallographic structure of the digestive lysozyme 1 from Musca domestica at 1.90 Ang. | 分子名称: | DI(HYDROXYETHYL)ETHER, Lysozyme 1, SULFATE ION | 著者 | Cancado, F.C, Marana, S.R, Barbosa, J.A.R.G. | 登録日 | 2005-12-09 | 公開日 | 2006-12-12 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystallization, data collection and phasing of two digestive lysozymes from Musca domestica. Acta Crystallogr.,Sect.F, 62, 2006
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2FC8
| Solution structure of the RRM_1 domain of NCL protein | 分子名称: | NCL protein | 著者 | Dang, W, Muto, Y, Inoue, M, Kigawa, T, Shirouzu, M, Terada, T, Yokoyama, S, RIKEN Structural Genomics/Proteomics Initiative (RSGI) | 登録日 | 2005-12-12 | 公開日 | 2006-06-12 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Solution structure of the RRM_1 domain of NCL protein To be published
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2FDY
| Microsomal P450 2A6 with the inhibitor Adrithiol bound | 分子名称: | 4,4'-DIPYRIDYL DISULFIDE, Cytochrome P450 2A6, PROTOPORPHYRIN IX CONTAINING FE, ... | 著者 | Yano, J.K, Stout, C.D, Johnson, E.F. | 登録日 | 2005-12-14 | 公開日 | 2006-11-28 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Synthetic Inhibitors of Cytochrome P-450 2A6: Inhibitory Activity, Difference Spectra, Mechanism of Inhibition, and Protein Cocrystallization. J.Med.Chem., 49, 2006
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2FE6
| P450CAM from Pseudomonas putida reconstituted with manganic protoporphyrin IX | 分子名称: | Cytochrome P450-cam, POTASSIUM ION, PROTOPORPHYRIN IX CONTAINING MN | 著者 | von Koenig, K, Makris, T.M, Sligar, S.G, Schlichting, I. | 登録日 | 2005-12-15 | 公開日 | 2006-03-14 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | The status of high-valent metal oxo complexes in the P450 cytochromes. J.Inorg.Biochem., 100, 2006
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1MIQ
| Crystal structure of proplasmepsin from the human malarial pathogen Plasmodium vivax | 分子名称: | plasmepsin | 著者 | Bernstein, N.K, Cherney, M.M, Yowell, C.A, Dame, J.B, James, M.N. | 登録日 | 2002-08-23 | 公開日 | 2002-09-18 | 最終更新日 | 2018-01-31 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural insights into the activation of P. vivax plasmepsin. J.Mol.Biol., 329, 2003
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2FFB
| The crystal structure of the HlyB-NBD E631Q mutant in complex with ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, Alpha-hemolysin translocation ATP-binding protein hlyB | 著者 | Zaitseva, J, Oswald, C, Jumpertz, T, Jenewein, S, Holland, I.B, Schmitt, L. | 登録日 | 2005-12-19 | 公開日 | 2006-08-08 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | A structural analysis of asymmetry required for catalytic activity of an ABC-ATPase domain dimer. Embo J., 25, 2006
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1M2R
| Crystal structure of 5,8-di-amino-1,4-di-hydroxy-anthraquinone/CK2 kinase complex | 分子名称: | 5,8-DI-AMINO-1,4-DIHYDROXY-ANTHRAQUINONE, CASEIN kinase II, alpha chain | 著者 | De Moliner, E, Moro, S, Sarno, S, Zagotto, G, Zanotti, G, Pinna, L.A, Battistutta, R. | 登録日 | 2002-06-25 | 公開日 | 2003-06-17 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Inhibition of protein kinase CK2 by anthraquinone-related compounds. A
structural insight J.Biol.Chem., 278, 2003
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1M5O
| Transition State Stabilization by a Catalytic RNA | 分子名称: | CALCIUM ION, RNA SUBSTRATE, RNA HAIRPIN RIBOZYME, ... | 著者 | Rupert, P.B, Massey, A.P, Sigurdsson, S.T, Ferre-D'Amare, A.R. | 登録日 | 2002-07-09 | 公開日 | 2002-10-12 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Transition state stabilization by a catalytic RNA Science, 298, 2002
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1M61
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2FKA
| Crystal structure of Mg(2+) and BeF(3)(-)-bound CheY in complex with CheZ(200-214) solved from a F432 crystal grown in CAPS (pH 10.5) | 分子名称: | 3-CYCLOHEXYL-1-PROPYLSULFONIC ACID, BERYLLIUM TRIFLUORIDE ION, C-terminal 15-mer from Chemotaxis protein cheZ, ... | 著者 | Guhaniyogi, J, Robinson, V.L, Stock, A.M. | 登録日 | 2006-01-04 | 公開日 | 2006-05-23 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal Structures of Beryllium Fluoride-free and Beryllium Fluoride-bound CheY in Complex with the Conserved C-terminal Peptide of CheZ Reveal Dual Binding Modes Specific to CheY Conformation. J.Mol.Biol., 359, 2006
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1M7B
| Crystal structure of Rnd3/RhoE: functional implications | 分子名称: | GUANOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, Rnd3/RhoE small GTP-binding protein | 著者 | Fiegen, D, Blumenstein, L, Stege, P, Vetter, I.R, Ahmadian, M.R. | 登録日 | 2002-07-19 | 公開日 | 2002-08-07 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of Rnd3/RhoE: functional implications FEBS LETT., 525, 2002
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1M5A
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1MB3
| CRYSTAL STRUCTURE OF THE RESPONSE REGULATOR DIVK AT PH 8.5 IN COMPLEX WITH MG2+ | 分子名称: | MAGNESIUM ION, cell division response regulator DivK | 著者 | Guillet, V, Ohta, N, Cabantous, S, Newton, A, Samama, J.-P, Structural Proteomics in Europe (SPINE) | 登録日 | 2002-08-02 | 公開日 | 2002-12-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (1.41 Å) | 主引用文献 | Crystallographic and Biochemical Studies of DivK Reveal Novel Features of
an Essential Response Regulator in Caulobacter crescentus. J.Biol.Chem., 277, 2002
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1MBD
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