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4EU1
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Structure of a mitochondrial aspartate aminotransferase from Trypanosoma brucei
分子名称: 1,2-ETHANEDIOL, CHLORIDE ION, Mitochondrial aspartate aminotransferase
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2012-04-25
公開日2012-05-16
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Structures of aspartate aminotransferases from Trypanosoma brucei, Leishmania major and Giardia lamblia.
Acta Crystallogr F Struct Biol Commun, 71, 2015
2HUI
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BU of 2hui by Molmil
Crystal structure of Aedes aegypti alanine glyoxylate aminotransferase in complex with glyoxylic acid
分子名称: Alanine glyoxylate aminotransferase, GLYOXYLIC ACID
著者Han, Q, Robinson, H, Gao, Y.G, Vogelaar, N, Wilson, S.R, Rizzi, M, Li, J.
登録日2006-07-26
公開日2006-09-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystal Structures of Aedes aegypti Alanine Glyoxylate Aminotransferase.
J.Biol.Chem., 281, 2006
2HUF
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Crystal structure of Aedes aegypti alanine glyoxylate aminotransferase
分子名称: 1-BUTANOL, Alanine glyoxylate aminotransferase
著者Han, Q, Robinson, H, Gao, Y.G, Vogelaar, N, Wilson, S.R, Rizzi, M, Li, J.
登録日2006-07-26
公開日2006-09-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Crystal Structures of Aedes aegypti Alanine Glyoxylate Aminotransferase.
J.Biol.Chem., 281, 2006
3R9A
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Human alanine-glyoxylate aminotransferase in complex with the TPR domain of human PEX5P
分子名称: 2-[BIS-(2-HYDROXY-ETHYL)-AMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Peroxisomal targeting signal 1 receptor, Serine--pyruvate aminotransferase
著者Fodor, K, Wilmanns, M.
登録日2011-03-25
公開日2011-05-11
最終更新日2012-05-02
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Molecular requirements for peroxisomal targeting of alanine-glyoxylate aminotransferase as an essential determinant in primary hyperoxaluria type 1
Plos Biol., 10, 2012
2AY5
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-INDOLEPROPIONIC ACID
分子名称: AROMATIC AMINO ACID AMINOTRANSFERASE, INDOLYLPROPIONIC ACID, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
4H51
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Crystal structure of a putative Aspartate Aminotransferase from Leishmania major Friedlin
分子名称: 1,2-ETHANEDIOL, Aspartate aminotransferase
著者Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2012-09-18
公開日2012-10-10
最終更新日2015-05-20
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structures of aspartate aminotransferases from Trypanosoma brucei, Leishmania major and Giardia lamblia.
Acta Crystallogr F Struct Biol Commun, 71, 2015
5MED
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BU of 5med by Molmil
Cyanothece lipoxygenase 2 (CspLOX2)
分子名称: 1,3-PROPANDIOL, 1,4-BUTANEDIOL, 1-BUTANOL, ...
著者Newie, J, Neumann, P, Werner, M, Mata, R.A, Ficner, R, Feussner, I.
登録日2016-11-14
公開日2017-05-31
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Lipoxygenase 2 from Cyanothece sp. controls dioxygen insertion by steric shielding and substrate fixation.
Sci Rep, 7, 2017
2AY7
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 4-PHENYLBUTYRIC ACID
分子名称: 4-PHENYL-BUTANOIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2AY2
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH CYCLOHEXANE PROPIONIC ACID
分子名称: AROMATIC AMINO ACID AMINOTRANSFERASE, CYCLOHEXANE PROPIONIC ACID, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2AY3
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-(3,4-DIMETHOXYPHENYL)PROPIONIC ACID
分子名称: 3-(3,4-DIMETHOXYPHENYL)PROPIONIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2AY9
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BU of 2ay9 by Molmil
AROMATIC AMINO ACID AMINOTRANSFERASE WITH 5-PHENYLVALERIC ACID
分子名称: 5-PHENYLVALERIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2HUU
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BU of 2huu by Molmil
Crystal structure of Aedes aegypti alanine glyoxylate aminotransferase in complex with alanine
分子名称: 1-BUTANOL, ALANINE, Alanine glyoxylate aminotransferase
著者Han, Q, Robinson, H, Gao, Y.G, Vogelaar, N, Wilson, S.R, Rizzi, M, Li, J.
登録日2006-07-27
公開日2006-09-26
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Crystal Structures of Aedes aegypti Alanine Glyoxylate Aminotransferase.
J.Biol.Chem., 281, 2006
1YIY
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Aedes aegypti kynurenine aminotransferase
分子名称: 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, BROMIDE ION, kynurenine aminotransferase; glutamine transaminase K
著者Han, Q, Gao, Y.G, Robinson, H, Ding, H, Wilson, S, Li, J.
登録日2005-01-13
公開日2005-05-10
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of Aedes aegypti kynurenine aminotransferase.
FEBS J., 272, 2005
1YIZ
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Aedes aegypti kynurenine aminotrasferase
分子名称: BROMIDE ION, kynurenine aminotransferase; glutamine transaminase
著者Han, Q, Gao, Y.G, Robinson, H, Ding, H, Wilson, S, Li, J.
登録日2005-01-13
公開日2005-05-10
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Crystal structures of Aedes aegypti kynurenine aminotransferase.
FEBS J., 272, 2005
2AY8
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 4-(2-THIENYL)BUTYRIC ACID
分子名称: 4-(2-THIENYL)BUTYRIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
4I8A
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BU of 4i8a by Molmil
Alanine-glyoxylate aminotransferase variant S187F
分子名称: GLYCEROL, Serine-pyruvate aminotransferase
著者Fodor, K, Oppici, E, Williams, C, Cellini, B, Wilmanns, M.
登録日2012-12-03
公開日2013-05-01
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Crystal structure of the S187F variant of human liver alanine: Aminotransferase associated with primary hyperoxaluria type I and its functional implications.
Proteins, 81, 2013
2AY6
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-INDOLEBUTYRIC ACID
分子名称: 3-INDOLEBUTYRIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2R2N
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The crystal structure of human kynurenine aminotransferase II in complex with kynurenine
分子名称: (2S)-2-amino-4-(2-aminophenyl)-4-oxobutanoic acid, 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, GLYCEROL, ...
著者Han, Q, Robinson, H, Li, J.
登録日2007-08-27
公開日2007-12-04
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Crystal structure of human kynurenine aminotransferase II.
J.Biol.Chem., 283, 2008
2AY1
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 4-AMINOHYDROCINNAMIC ACID
分子名称: 4-AMINOHYDROCINNAMIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2AY4
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AROMATIC AMINO ACID AMINOTRANSFERASE WITH 3-(P-TOLYL)PROPIONIC ACID
分子名称: 3-(P-TOLYL)PROPIONIC ACID, AROMATIC AMINO ACID AMINOTRANSFERASE, PYRIDOXAL-5'-PHOSPHATE
著者Okamoto, A, Hirotsu, K, Kagamiyama, H.
登録日1998-08-06
公開日1999-02-02
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献The active site of Paracoccus denitrificans aromatic amino acid aminotransferase has contrary properties: flexibility and rigidity.
Biochemistry, 38, 1999
2QLR
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Crystal structure of human kynurenine aminotransferase II
分子名称: GLYCEROL, Kynurenine/alpha-aminoadipate aminotransferase mitochondrial
著者Han, Q, Robinson, R, Li, J.
登録日2007-07-13
公開日2007-12-04
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structure of Human Kynurenine Aminotransferase II
J.Biol.Chem., 283, 2008
2QB3
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Structural Studies Reveal the Inactivation of E. coli L-Aspartate Aminotransferase by (s)-4,5-dihydro-2-thiophenecarboxylic acid (SADTA) via Two Mechanisms (at pH 7.5)
分子名称: 4'-DEOXY-4'-AMINOPYRIDOXAL-5'-PHOSPHATE, 4-[({3-HYDROXY-2-METHYL-5-[(PHOSPHONOOXY)METHYL]PYRIDIN-4-YL}METHYL)AMINO]THIOPHENE-2-CARBOXYLIC ACID, Aspartate aminotransferase, ...
著者Liu, D, Pozharski, E, Lepore, B, Fu, M, Silverman, R.B, Petsko, G.A, Ringe, D.
登録日2007-06-15
公開日2007-12-04
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.45 Å)
主引用文献Inactivation of Escherichia coli L-aspartate aminotransferase by (S)-4-amino-4,5-dihydro-2-thiophenecarboxylic acid reveals "a tale of two mechanisms".
Biochemistry, 46, 2007
2R5C
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Aedes Kynurenine Aminotransferase in Complex with Cysteine
分子名称: Kynurenine aminotransferase, N-({3-HYDROXY-2-METHYL-5-[(PHOSPHONOOXY)METHYL]PYRIDIN-4-YL}METHYL)-L-CYSTEINE
著者Han, Q, Gao, Y.G, Robinson, H, Li, J.
登録日2007-09-03
公開日2008-03-18
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structural insight into the mechanism of substrate specificity of aedes kynurenine aminotransferase.
Biochemistry, 47, 2008
2BKW
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Yeast alanine:glyoxylate aminotransferase YFL030w
分子名称: ALANINE-GLYOXYLATE AMINOTRANSFERASE 1, GLYOXYLIC ACID, PYRIDOXAL-5'-PHOSPHATE
著者Meyer, P, Liger, D, Leulliot, N, Quevillon-Cheruel, S, Zhou, C.Z, Borel, F, Ferrer, J.L, Poupon, A, Janin, J, van Tilbeurgh, H.
登録日2005-02-21
公開日2005-11-02
最終更新日2015-11-18
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Crystal Structure and Confirmation of the Alanine:Glyoxylate Aminotransferase Activity of the Yfl030W Yeast Protein
Biochimie, 87, 2005
3UE8
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Kynurenine Aminotransferase II Inhibitors
分子名称: (5-hydroxy-4-{[(1-hydroxy-2-oxo-1,2-dihydroquinolin-3-yl)amino]methyl}-6-methylpyridin-3-yl)methyl dihydrogen phosphate, CHLORIDE ION, Kynurenine/alpha-aminoadipate aminotransferase, ...
著者Dounay, A.B, Anderson, M, Bechle, B.M, Campbell, B.M, Claffey, M.M, Evdokimov, A, Edelweiss, E, Fonseca, K.R, Gan, X, Ghosh, S, Hayward, M.M, Horner, W, Kim, J.Y, McAllister, L.A, Pandit, J, Paradis, V, Parikh, V.D, Reese, M.R, Rong, S.B, Salafia, M.A, Schuyten, K, Strick, C.A, Tuttle, J.B, Valentine, J, Wang, H, Zawadzke, L.E, Verhoest, P.R.
登録日2011-10-28
公開日2012-02-01
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (3.22 Å)
主引用文献Discovery of Brain-Penetrant, Irreversible Kynurenine Aminotransferase II Inhibitors for Schizophrenia.
ACS Med Chem Lett, 3, 2012

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