2AFU
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![BU of 2afu by Molmil](/molmil-images/mine/2afu) | Crystal structure of human glutaminyl cyclase in complex with glutamine t-butyl ester | 分子名称: | Glutaminyl-peptide cyclotransferase, TERT-BUTYL D-ALPHA-GLUTAMINATE, ZINC ION | 著者 | Huang, K.F, Liu, Y.L, Cheng, W.J, Ko, T.P, Wang, A.H.J. | 登録日 | 2005-07-26 | 公開日 | 2005-08-23 | 最終更新日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Crystal structures of human glutaminyl cyclase, an enzyme responsible for protein N-terminal pyroglutamate formation Proc.Natl.Acad.Sci.Usa, 102, 2005
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2JNU
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![BU of 2jnu by Molmil](/molmil-images/mine/2jnu) | Solution structure of the RGS domain of human RGS14 | 分子名称: | Regulator of G-protein signaling 14 | 著者 | Dowler, E.F, Diehl, A, Bray, J, Elkins, J, Soundararajan, M, Doyle, D.A, Gileadi, C, Phillips, C, Schoch, G.A, Yang, X, Brockmann, C, Leidert, M, Rehbein, K, Schmieder, P, Kuhne, R, Higman, V.A, Sundstrom, M, Arrowsmith, C, Weigelt, J, Edwards, A, Oschkinat, H, Ball, L.J, Structural Genomics Consortium (SGC) | 登録日 | 2007-02-02 | 公開日 | 2007-02-27 | 最終更新日 | 2024-05-08 | 実験手法 | SOLUTION NMR | 主引用文献 | Structural diversity in the RGS domain and its interaction with heterotrimeric G protein alpha-subunits. Proc.Natl.Acad.Sci.Usa, 105, 2008
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4B1Z
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![BU of 4b1z by Molmil](/molmil-images/mine/4b1z) | Structure of the Phactr1 RPEL domain bound to G-actin | 分子名称: | ACTIN, ALPHA SKELETAL MUSCLE, ADENOSINE-5'-TRIPHOSPHATE, ... | 著者 | Mouilleron, S, Wiezlak, M, O'Reilly, N, Treisman, R, McDonald, N.Q. | 登録日 | 2012-07-12 | 公開日 | 2012-11-07 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (3.3 Å) | 主引用文献 | Structures of the Phactr1 RPEL domain and RPEL motif complexes with G-actin reveal the molecular basis for actin binding cooperativity. Structure, 20, 2012
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4B1T
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![BU of 4b1t by Molmil](/molmil-images/mine/4b1t) | Structure of the factor Xa-like trypsin variant triple-Ala (TA) in complex with eglin C | 分子名称: | 1,2-ETHANEDIOL, CALCIUM ION, CATIONIC TRYPSIN, ... | 著者 | Menzel, A, Neumann, P, Stubbs, M.T. | 登録日 | 2012-07-12 | 公開日 | 2012-08-01 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (1.78 Å) | 主引用文献 | Thermodynamic signatures in macromolecular interactions involving conformational flexibility. Biol.Chem., 395, 2014
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1ZO3
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![BU of 1zo3 by Molmil](/molmil-images/mine/1zo3) | The P-site and P/E-site tRNA structures fitted to P/I site codon. | 分子名称: | tRNA | 著者 | Allen, G.S, Zavialov, A, Gursky, R, Ehrenberg, M, Frank, J. | 登録日 | 2005-05-12 | 公開日 | 2005-06-14 | 最終更新日 | 2024-02-14 | 実験手法 | ELECTRON MICROSCOPY (13.8 Å) | 主引用文献 | The Cryo-EM Structure of a Translation Initiation Complex from Escherichia coli. Cell(Cambridge,Mass.), 121, 2005
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2A1M
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1ZZZ
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![BU of 1zzz by Molmil](/molmil-images/mine/1zzz) | Trypsin inhibitors with rigid tripeptidyl aldehydes | 分子名称: | 2-{(3S)-3-[(benzylsulfonyl)amino]-2-oxopiperidin-1-yl}-N-{(2S)-1-[(3R)-1-carbamimidoylpiperidin-3-yl]-3-oxopropan-2-yl}acetamide, CALCIUM ION, TRYPSIN | 著者 | Krishnan, R, Zhang, E, Hakansson, K, Arni, R.K, Tulinsky, A, Lim-Wilby, M.S.L, Levy, O.E, Semple, J.E, Brunck, T.K. | 登録日 | 1998-06-02 | 公開日 | 1999-06-15 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Highly selective mechanism-based thrombin inhibitors: structures of thrombin and trypsin inhibited with rigid peptidyl aldehydes. Biochemistry, 37, 1998
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2JWZ
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![BU of 2jwz by Molmil](/molmil-images/mine/2jwz) | Mutations in the hydrophobic core of ubiquitin differentially affect its recognition by receptor proteins | 分子名称: | Ubiquitin | 著者 | Haririnia, A, Verma, R, Purohit, N, Twarog, M, Deshaies, R, Bolon, D, Fushman, D. | 登録日 | 2007-10-31 | 公開日 | 2008-01-08 | 最終更新日 | 2024-05-29 | 実験手法 | SOLUTION NMR | 主引用文献 | Mutations in the hydrophobic core of ubiquitin differentially affect its recognition by receptor proteins. J.Mol.Biol., 375, 2008
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2LSQ
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![BU of 2lsq by Molmil](/molmil-images/mine/2lsq) | Analog of the fragment 197-221 of beta-1 adrenoreceptor | 分子名称: | ANALOG OF THE FRAGMENT 197-221 OF BETA-1 ADRENORECEPTOR | 著者 | Bushuev, V.N, Zykov, K.A, Bespalova, Z.D, Bibilashvili, R.S, Efremov, E.E, Golitsyn, S.P, Kaznacheeva, L.I, Kuzhetsova, T.V, Levashov, P.S, Masenko, V.P, Mironova, N.A, Molokoedov, F.S, Rutkevich, P.N, Rvacheva, A.V, Sharf, T.V, Sidorova, M.V, Vlasik, T.N, Yanushevskaya, E.V. | 登録日 | 2012-05-04 | 公開日 | 2013-05-08 | 最終更新日 | 2023-06-14 | 実験手法 | SOLUTION NMR | 主引用文献 | Analog of the fragment 197-221 of 1-adrenoreceptor To be Published
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2R55
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![BU of 2r55 by Molmil](/molmil-images/mine/2r55) | Human StAR-related lipid transfer protein 5 | 分子名称: | StAR-related lipid transfer protein 5 | 著者 | Lehtio, L, Busam, R.D, Arrowsmith, C.H, Berglund, H, Collins, R, Dahlgren, L.G, Edwards, A.M, Flodin, S, Flores, A, Graslund, S, Hammarstrom, M, Hallberg, B.M, Herman, M.D, Johansson, I, Kallas, A, Karlberg, T, Kotenyova, T, Moche, M, Nordlund, P, Nyman, T, Sagemark, J, Sundstrom, M, Thorsell, A.G, Tresaugues, L, Van Den Berg, S, Weigelt, J, Welin, M, Persson, C, Structural Genomics Consortium (SGC) | 登録日 | 2007-09-03 | 公開日 | 2007-09-18 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Comparative structural analysis of lipid binding START domains. Plos One, 6, 2011
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7GSL
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7GSM
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7GT0
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7GTA
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![BU of 7gta by Molmil](/molmil-images/mine/7gta) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOMB000065a | 分子名称: | (5S)-N-(4-fluorophenyl)-5-methyl-4,5-dihydro-1,3-thiazol-2-amine, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2.06 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GTH
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![BU of 7gth by Molmil](/molmil-images/mine/7gth) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000637a | 分子名称: | (6aR,8R,12R,12aS)-2-methyl-6a,10,11,12a-tetrahydro-6H,7H,9H-[1]benzopyrano[4,3-c]pyrazolo[1,2-a]pyrazol-9-one, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.66 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GTL
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![BU of 7gtl by Molmil](/molmil-images/mine/7gtl) | PanDDA analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000554a | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1, benzyl (3aS,8aS)-1-oxooctahydropyrrolo[3,4-d]azepine-6(1H)-carboxylate | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSD
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![BU of 7gsd by Molmil](/molmil-images/mine/7gsd) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOPL000605a | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 4-(5-amino-1,3,4-thiadiazol-2-yl)phenol, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSO
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7GSW
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7GSF
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7GT4
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![BU of 7gt4 by Molmil](/molmil-images/mine/7gt4) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000528a | 分子名称: | (4R)-4-hydroxy-2-(2-hydroxyethyl)-3,4-dihydro-1lambda~6~,2-benzothiazine-1,1(2H)-dione, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GSZ
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![BU of 7gsz by Molmil](/molmil-images/mine/7gsz) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMSOA000686b | 分子名称: | 1-[4-methyl-2-(pyridin-4-yl)-1,3-thiazol-5-yl]methanamine, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GTG
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![BU of 7gtg by Molmil](/molmil-images/mine/7gtg) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOOA000684a | 分子名称: | (5R,7S,8R,8aS)-2-(cyclopropylmethyl)-8-phenyloctahydropyrrolo[1,2-a]pyrazine-7-carboxamide, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.69 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GST
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![BU of 7gst by Molmil](/molmil-images/mine/7gst) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOMB000056a | 分子名称: | 1-(methanesulfonyl)-1,2,3,4-tetrahydroquinoline, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1 | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (1.64 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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7GTQ
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![BU of 7gtq by Molmil](/molmil-images/mine/7gtq) | PanDDA Analysis group deposition -- Crystal structure of PTP1B in complex with FMOPL000311a | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Tyrosine-protein phosphatase non-receptor type 1, ~{N}-(2-ethyl-1,2,3,4-tetrazol-5-yl)butanamide | 著者 | Mehlman, T, Ginn, H.M, Keedy, D.A. | 登録日 | 2024-01-03 | 公開日 | 2024-01-24 | 最終更新日 | 2024-04-24 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | An expanded view of ligandability in the allosteric enzyme PTP1B from computational reanalysis of large-scale crystallographic data. Biorxiv, 2024
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