8YHP
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![BU of 8yhp by Molmil](/molmil-images/mine/8yhp) | Structure of the PGK1 from Biortus. | 分子名称: | 1,2-ETHANEDIOL, Phosphoglycerate kinase 1 | 著者 | Wang, F, Cheng, W, Lv, Z, Ju, C, Wang, J. | 登録日 | 2024-02-28 | 公開日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | Structure of the PGK1 from Biortus. To Be Published
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8UZO
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![BU of 8uzo by Molmil](/molmil-images/mine/8uzo) | |
8Y6C
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![BU of 8y6c by Molmil](/molmil-images/mine/8y6c) | Norovirus GII.10 P domain and 2'-FL (powder) | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, GII.10 norovirus P domain in complex with 2'FL (powder), ... | 著者 | Hansman, G, Tame, J.R.H, Kher, G, Pancera, M. | 登録日 | 2024-02-02 | 公開日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Norovirus GII.10 P domain and 2'-FL (powder) To Be Published
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8YX9
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![BU of 8yx9 by Molmil](/molmil-images/mine/8yx9) | CD40 in complex with Dacetuzumab Fab | 分子名称: | Dacetuzumab, Heavy chain, light chain, ... | 著者 | Caaveiro, J.M.M, Fernandez-Perez, J, Tsumoto, K. | 登録日 | 2024-04-02 | 公開日 | 2024-05-08 | 最終更新日 | 2024-05-22 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Crystal structures of human CD40 in complex with monoclonal antibodies dacetuzumab and bleselumab. Biochem.Biophys.Res.Commun., 714, 2024
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8YTX
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![BU of 8ytx by Molmil](/molmil-images/mine/8ytx) | Tubulin-RB3-TTL in complex with compound SI9 | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-chloranyl-~{N}-(4-methoxyphenyl)-~{N}-methyl-thieno[2,3-d]pyrimidin-4-amine, CALCIUM ION, ... | 著者 | Wu, C.Y, Wang, Y.X. | 登録日 | 2024-03-26 | 公開日 | 2024-06-05 | 実験手法 | X-RAY DIFFRACTION (2.53 Å) | 主引用文献 | Tubulin-RB3-TTL in complex with compound SI9 To Be Published
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8V31
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![BU of 8v31 by Molmil](/molmil-images/mine/8v31) | |
8V4R
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![BU of 8v4r by Molmil](/molmil-images/mine/8v4r) | |
8W1F
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![BU of 8w1f by Molmil](/molmil-images/mine/8w1f) | Crystal Structure of DPS-like protein PA4880 from Pseudomonas aeruginosa (dodecamer, Mg bound) | 分子名称: | DPS-LIKE PROTEIN, FE (II) ION, MAGNESIUM ION, ... | 著者 | Lovell, S, Liu, L, Seibold, S, Battaile, K.P, Rivera, M. | 登録日 | 2024-02-15 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Pseudomonas aeruginosa gene PA4880 encodes a Dps-like protein with a Dps fold, bacterioferritin-type ferroxidase centers, and endonuclease activity. Front Mol Biosci, 11, 2024
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8VQW
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9EY5
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![BU of 9ey5 by Molmil](/molmil-images/mine/9ey5) | |
8XN7
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![BU of 8xn7 by Molmil](/molmil-images/mine/8xn7) | Crystal structure of HPK1 kinase domain T165E,S171E phosphomimetic mutant in complex with compound 9f | 分子名称: | 5-amino-2-((6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-yl)amino)-8-(2-(trifluoromethyl)benzyl)pyrido[2,3-d]pyrimidin-7(8H)-one, Mitogen-activated protein kinase kinase kinase kinase 1 | 著者 | Huang, W.X, Liu, R, Ding, K. | 登録日 | 2023-12-29 | 公開日 | 2024-04-10 | 実験手法 | X-RAY DIFFRACTION (2.65 Å) | 主引用文献 | Discovery of 5-aminopyrido[2,3-d]pyrimidin-7(8H)-one derivatives as new hematopoietic progenitor kinase 1 (HPK1) inhibitors. Eur.J.Med.Chem., 269, 2024
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8V98
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![BU of 8v98 by Molmil](/molmil-images/mine/8v98) | GII.24 Loreto 1972 norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Capsid protein VP1 | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 2024
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9AT1
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![BU of 9at1 by Molmil](/molmil-images/mine/9at1) | Crystal structure of SARS-CoV-2 3CL protease in complex with a methylcyclohexyl 2-pyrrolidone inhibitor (R-enantiomer) | 分子名称: | (1S,2S)-2-{[N-({[(2R)-1-(cyclohexylmethyl)-5-oxopyrrolidin-2-yl]methoxy}carbonyl)-L-leucyl]amino}-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, 3C-like proteinase nsp5, TETRAETHYLENE GLYCOL | 著者 | Lovell, S, Cooper, A, Battaile, K.P, Dampalla, C.S, Groutas, W.C. | 登録日 | 2024-02-26 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Structure-Guided Design of Potent Coronavirus Inhibitors with a 2-Pyrrolidone Scaffold: Biochemical, Crystallographic, and Virological Studies. J.Med.Chem., 2024
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8YHL
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![BU of 8yhl by Molmil](/molmil-images/mine/8yhl) | The Crystal Structure of Tgf-Beta Type I Receptor (Alk5) from Biortus | 分子名称: | 1,2-ETHANEDIOL, 2-fluoranyl-~{N}-[[5-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-1~{H}-imidazol-2-yl]methyl]aniline, ACETATE ION, ... | 著者 | Wang, F, Cheng, W, Lv, Z, Meng, Q, Xu, Y. | 登録日 | 2024-02-28 | 公開日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | The Crystal Structure of Tgf-Beta Type I Receptor (Alk5) from Biortus To Be Published
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8TU3
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![BU of 8tu3 by Molmil](/molmil-images/mine/8tu3) | Bruton's tyrosine kinase in complex with covalent inhibitor compound 10 | 分子名称: | 1-[(4R)-4-{[(6P,8S)-6-(1-methyl-1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrazin-4-yl]oxy}azepan-1-yl]propan-1-one, Tyrosine-protein kinase BTK | 著者 | Metrick, C.M. | 登録日 | 2023-08-15 | 公開日 | 2024-06-26 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Discovery and Preclinical Characterization of BIIB129, a Covalent, Selective, and Brain-Penetrant BTK Inhibitor for the Treatment of Multiple Sclerosis. J.Med.Chem., 67, 2024
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8YHH
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![BU of 8yhh by Molmil](/molmil-images/mine/8yhh) | The Crystal Structure of Mitotic Kinesin Eg5 from Biortus | 分子名称: | 1,2-ETHANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Wang, F, Cheng, W, Lv, Z, Qi, J, Wu, B. | 登録日 | 2024-02-28 | 公開日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (1.95 Å) | 主引用文献 | The Crystal Structure of Mitotic Kinesin Eg5 from Biortus To Be Published
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9EY7
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8VCN
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![BU of 8vcn by Molmil](/molmil-images/mine/8vcn) | GluER mutant - W66F F269Y Q293T F68Y T36E P263L | 分子名称: | ACETATE ION, FLAVIN MONONUCLEOTIDE, GLYCEROL, ... | 著者 | Jeffrey, P.D, Sorigue, D.R, Liu, Y, Hyster, T.K. | 登録日 | 2023-12-14 | 公開日 | 2024-03-13 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.47 Å) | 主引用文献 | Asymmetric Synthesis of alpha-Chloroamides via Photoenzymatic Hydroalkylation of Olefins. J.Am.Chem.Soc., 146, 2024
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9ATF
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![BU of 9atf by Molmil](/molmil-images/mine/9atf) | Crystal structure of MERS 3CL protease in complex with a 1-methyl-4,4-difluorocyclohexyl 2-pyrrolidone inhibitor | 分子名称: | (1R,2S)-2-({N-[({(2S)-1-[(4,4-difluorocyclohexyl)methyl]-5-oxopyrrolidin-2-yl}methoxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, (1S,2S)-2-({N-[({(2S)-1-[(4,4-difluorocyclohexyl)methyl]-5-oxopyrrolidin-2-yl}methoxy)carbonyl]-L-leucyl}amino)-1-hydroxy-3-[(3S)-2-oxopyrrolidin-3-yl]propane-1-sulfonic acid, 3C-like proteinase nsp5 | 著者 | Liu, L, Lovell, S, Battaile, K.P, Dampalla, C.S, Groutas, W.C. | 登録日 | 2024-02-26 | 公開日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structure-Guided Design of Potent Coronavirus Inhibitors with a 2-Pyrrolidone Scaffold: Biochemical, Crystallographic, and Virological Studies. J.Med.Chem., 2024
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8V95
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![BU of 8v95 by Molmil](/molmil-images/mine/8v95) | GII.8 Amsterdam norovirus protruding domain | 分子名称: | 1,2-ETHANEDIOL, Capsid protein (Fragment) | 著者 | Kher, G, Prewitt, A, Pancera, M, Hansman, G. | 登録日 | 2023-12-07 | 公開日 | 2024-06-19 | 最終更新日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | Development of a broad-spectrum therapeutic Fc-nanobody for human noroviruses. J.Virol., 2024
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8YHW
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![BU of 8yhw by Molmil](/molmil-images/mine/8yhw) | The Crystal Structure of NF-kB-inducing Kinase (NIK) from Biortus | 分子名称: | 1,2-ETHANEDIOL, 3,6,9,12,15,18,21-HEPTAOXATRICOSANE-1,23-DIOL, MAGNESIUM ION, ... | 著者 | Wang, F, Cheng, W, Lv, Z, Meng, Q, Xu, Y. | 登録日 | 2024-02-28 | 公開日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | The Crystal Structure of NF-kB-inducing Kinase (NIK) from Biortus To Be Published
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8W1D
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![BU of 8w1d by Molmil](/molmil-images/mine/8w1d) | CRYSTAL STRUCTURE OF DPS-LIKE PROTEIN PA4880 FROM PSEUDOMONAS AERUGINOSA (DIMERIC FORM) | 分子名称: | DPS-LIKE PROTEIN, FE (II) ION | 著者 | Lovell, S, Battaile, K.P, Rivera, M. | 登録日 | 2024-02-15 | 公開日 | 2024-05-29 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.3 Å) | 主引用文献 | Pseudomonas aeruginosa gene PA4880 encodes a Dps-like protein with a Dps fold, bacterioferritin-type ferroxidase centers, and endonuclease activity. Front Mol Biosci, 11, 2024
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9AV7
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8YFJ
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8XOY
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![BU of 8xoy by Molmil](/molmil-images/mine/8xoy) | The Crystal Structure of PTP1B from Biortus. | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GLYCEROL, ... | 著者 | Wang, F, Cheng, W, Lv, Z, Meng, Q, Li, J. | 登録日 | 2024-01-02 | 公開日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | The Crystal Structure of PTP1B from Biortus. To Be Published
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