8A08
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![BU of 8a08 by Molmil](/molmil-images/mine/8a08) | |
8A06
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![BU of 8a06 by Molmil](/molmil-images/mine/8a06) | |
8A05
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![BU of 8a05 by Molmil](/molmil-images/mine/8a05) | |
8A04
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![BU of 8a04 by Molmil](/molmil-images/mine/8a04) | |
8A03
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![BU of 8a03 by Molmil](/molmil-images/mine/8a03) | |
8A02
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![BU of 8a02 by Molmil](/molmil-images/mine/8a02) | |
8A01
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![BU of 8a01 by Molmil](/molmil-images/mine/8a01) | |
7ZZZ
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![BU of 7zzz by Molmil](/molmil-images/mine/7zzz) | Bacteriophage phiCjT23 capsid | 分子名称: | Major capsid protein P5, Spike protein P13 N-terminal, capsid internal domain, ... | 著者 | Rissanen, I, Kejzar, N, Huiskonen, J.T. | 登録日 | 2022-05-26 | 公開日 | 2022-12-14 | 実験手法 | ELECTRON MICROSCOPY (4.1 Å) | 主引用文献 | Cryo-EM structure of ssDNA bacteriophage Phi CjT23 provides insight into early virus evolution. Nat Commun, 13, 2022
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7ZZR
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![BU of 7zzr by Molmil](/molmil-images/mine/7zzr) | HDAC2 in complex with inhibitory ligand | 分子名称: | 1,2-ETHANEDIOL, 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, CALCIUM ION, ... | 著者 | Cleasby, A, Tisi, D. | 登録日 | 2022-05-26 | 公開日 | 2022-09-21 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2.168 Å) | 主引用文献 | Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor. Acs Med.Chem.Lett., 13, 2022
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7ZZP
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![BU of 7zzp by Molmil](/molmil-images/mine/7zzp) | Structure of HDAC2 complexed with an inhibitory ligand | 分子名称: | (2S)-2-HYDROXYPROPANOIC ACID, 1,2-ETHANEDIOL, 2-[N-CYCLOHEXYLAMINO]ETHANE SULFONIC ACID, ... | 著者 | Cleasby, A, Tisi, D. | 登録日 | 2022-05-25 | 公開日 | 2022-09-21 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor. Acs Med.Chem.Lett., 13, 2022
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7ZZO
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![BU of 7zzo by Molmil](/molmil-images/mine/7zzo) | HDAC2 in complex with an inhibitor | 分子名称: | 2-(cyclohexylazaniumyl)ethanesulfonate, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ... | 著者 | Cleasby, A, Tisi, D. | 登録日 | 2022-05-25 | 公開日 | 2022-09-21 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Fragment-Based Discovery of a Novel, Brain Penetrant, Orally Active HDAC2 Inhibitor. Acs Med.Chem.Lett., 13, 2022
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7ZZK
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![BU of 7zzk by Molmil](/molmil-images/mine/7zzk) | Structure of the N-acetyl-D-glucosamine oxidase from Ralstonia Solanacearum | 分子名称: | ALANINE, DI(HYDROXYETHYL)ETHER, FLAVIN-ADENINE DINUCLEOTIDE, ... | 著者 | Boverio, A, Rozeboom, H.J, Fraaije, M.W. | 登録日 | 2022-05-25 | 公開日 | 2022-08-03 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (1.5 Å) | 主引用文献 | Structural Elucidation and Engineering of a Bacterial Carbohydrate Oxidase. Biochemistry, 62, 2023
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7ZZD
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![BU of 7zzd by Molmil](/molmil-images/mine/7zzd) | Crystal structure of NAD kinase 1 from Listeria monocytogenes in complex with a linear di-adenosine derivative | 分子名称: | 2-[[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl-[3-[6-azanyl-9-[(2~{R},3~{R},4~{S},5~{R})-5-[(3-azanylpropanoylamino)methyl]-3,4-bis(oxidanyl)oxolan-2-yl]purin-8-yl]prop-2-ynyl]amino]ethanoic acid, CITRIC ACID, NAD kinase 1 | 著者 | Gelin, M, Labesse, G. | 登録日 | 2022-05-25 | 公開日 | 2023-01-11 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.79 Å) | 主引用文献 | Synthesis and structure-activity relationship studies of original cyclic diadenosine derivatives as nanomolar inhibitors of NAD kinase from pathogenic bacteria. Eur.J.Med.Chem., 246, 2023
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7ZZC
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![BU of 7zzc by Molmil](/molmil-images/mine/7zzc) | Crystal structure of NAD kinase 1 from Listeria monocytogenes in complex with a linear di-adenosine derivative | 分子名称: | 2-[[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl-[3-[6-azanyl-9-[(2~{R},3~{R},4~{S},5~{R})-5-[(2-azanylethylsulfonylamino)methyl]-3,4-bis(oxidanyl)oxolan-2-yl]purin-8-yl]prop-2-ynyl]amino]ethanoic acid, CITRIC ACID, GLYCEROL, ... | 著者 | Gelin, M, Labesse, G. | 登録日 | 2022-05-25 | 公開日 | 2023-01-11 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Synthesis and structure-activity relationship studies of original cyclic diadenosine derivatives as nanomolar inhibitors of NAD kinase from pathogenic bacteria. Eur.J.Med.Chem., 246, 2023
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7ZZ9
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![BU of 7zz9 by Molmil](/molmil-images/mine/7zz9) | Crystal structure of NAD kinase 1 from Listeria monocytogenes in complex with a linear di-adenosine derivative | 分子名称: | 3-[[(2~{R},3~{S},4~{R},5~{R})-5-[8-[3-[[(2~{R},3~{S},4~{R},5~{R})-5-(6-aminopurin-9-yl)-3,4-bis(oxidanyl)oxolan-2-yl]methyl-(2-azanylethyl)amino]prop-1-ynyl]-6-azanyl-purin-9-yl]-3,4-bis(oxidanyl)oxolan-2-yl]methylamino]-3-oxidanylidene-propanoic acid, CITRIC ACID, NAD kinase 1 | 著者 | Gelin, M, Labesse, G. | 登録日 | 2022-05-25 | 公開日 | 2023-01-11 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.89 Å) | 主引用文献 | Synthesis and structure-activity relationship studies of original cyclic diadenosine derivatives as nanomolar inhibitors of NAD kinase from pathogenic bacteria. Eur.J.Med.Chem., 246, 2023
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7ZZ8
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![BU of 7zz8 by Molmil](/molmil-images/mine/7zz8) | Cryo-EM structure of Lactococcus lactis pyruvate carboxylase with acetyl-CoA and cyclic di-AMP | 分子名称: | (2R,3R,3aS,5R,7aR,9R,10R,10aS,12R,14aR)-2,9-bis(6-amino-9H-purin-9-yl)octahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8 ]tetraoxadiphosphacyclododecine-3,5,10,12-tetrol 5,12-dioxide, ACETYL COENZYME *A, ADENOSINE-5'-DIPHOSPHATE, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (3.29 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ6
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![BU of 7zz6 by Molmil](/molmil-images/mine/7zz6) | Cryo-EM structure of "CT-CT dimer" of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | MAGNESIUM ION, MANGANESE (II) ION, PYRUVIC ACID, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-12-28 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.15 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ5
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![BU of 7zz5 by Molmil](/molmil-images/mine/7zz5) | Cryo-EM structure of "BC open" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | ACETYL COENZYME *A, BICARBONATE ION, Pyruvate carboxylase | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2022-10-26 | 実験手法 | ELECTRON MICROSCOPY (2.43 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ4
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![BU of 7zz4 by Molmil](/molmil-images/mine/7zz4) | Cryo-EM structure of "BC closed" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | ACETYL COENZYME *A, ADENOSINE-5'-TRIPHOSPHATE, MAGNESIUM ION, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2022-11-02 | 実験手法 | ELECTRON MICROSCOPY (2.63 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ3
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![BU of 7zz3 by Molmil](/molmil-images/mine/7zz3) | Cryo-EM structure of "BC react" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | ACETYL COENZYME *A, ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.41 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ2
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![BU of 7zz2 by Molmil](/molmil-images/mine/7zz2) | Cryo-EM structure of "CT pyr" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | MAGNESIUM ION, MANGANESE (II) ION, PYRUVIC ACID, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.48 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ1
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![BU of 7zz1 by Molmil](/molmil-images/mine/7zz1) | Cryo-EM structure of "CT react" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | BIOTIN, MAGNESIUM ION, MANGANESE (II) ION, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2022-11-02 | 実験手法 | ELECTRON MICROSCOPY (2.27 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZZ0
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![BU of 7zz0 by Molmil](/molmil-images/mine/7zz0) | Cryo-EM structure of "CT empty" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | MAGNESIUM ION, MANGANESE (II) ION, Pyruvate carboxylase | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2022-11-02 | 実験手法 | ELECTRON MICROSCOPY (2.26 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZYZ
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![BU of 7zyz by Molmil](/molmil-images/mine/7zyz) | Cryo-EM structure of "CT oxa" conformation of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | MANGANESE (II) ION, OXALOACETATE ION, Pyruvate carboxylase | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2022-11-02 | 実験手法 | ELECTRON MICROSCOPY (2.47 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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7ZYY
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![BU of 7zyy by Molmil](/molmil-images/mine/7zyy) | Cryo-EM structure of Lactococcus lactis pyruvate carboxylase with acetyl-CoA | 分子名称: | ACETYL COENZYME *A, ADENOSINE-5'-DIPHOSPHATE, BICARBONATE ION, ... | 著者 | Lopez-Alonso, J.P, Lazaro, M, Gil, D, Choi, P.H, Tong, L, Valle, M. | 登録日 | 2022-05-25 | 公開日 | 2022-10-12 | 最終更新日 | 2023-11-15 | 実験手法 | ELECTRON MICROSCOPY (2.12 Å) | 主引用文献 | CryoEM structural exploration of catalytically active enzyme pyruvate carboxylase. Nat Commun, 13, 2022
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