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7D23
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BU of 7d23 by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with one K ion bound to the active site
分子名称: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Glutaminyl-peptide cyclotransferase, POTASSIUM ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-15
公開日2021-04-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D17
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BU of 7d17 by Molmil
Crystal structure of Macrostomum lignano glutaminyl cyclase
分子名称: Glutaminyl-peptide cyclotransferase, ZINC ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-14
公開日2021-04-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.998 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D1N
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BU of 7d1n by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with three Cu ions bound to the active site
分子名称: BICARBONATE ION, COPPER (II) ION, Glutaminyl-peptide cyclotransferase
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-15
公開日2021-04-14
最終更新日2024-10-23
実験手法X-RAY DIFFRACTION (2.26 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D1Y
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BU of 7d1y by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with two Co ions bound to the active site
分子名称: COBALT (II) ION, Glutaminyl-peptide cyclotransferase
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-15
公開日2021-04-14
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D1P
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BU of 7d1p by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with three Cd ions bound to the active site
分子名称: BICARBONATE ION, CADMIUM ION, Glutaminyl-peptide cyclotransferase
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-15
公開日2021-04-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2.36 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D21
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BU of 7d21 by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with two Zn ions bound to the active site
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, Glutaminyl-peptide cyclotransferase, ZINC ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-15
公開日2021-04-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D2J
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BU of 7d2j by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with a Cd ion bound to the active site
分子名称: BICARBONATE ION, CADMIUM ION, Glutaminyl-peptide cyclotransferase
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-16
公開日2021-04-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D1E
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BU of 7d1e by Molmil
Crystal structure of Bacteroides thetaiotaomicron glutaminyl cyclase bound to N-acetylhistamine
分子名称: Leucine aminopeptidase, N-[2-(1H-IMIDAZOL-4-YL)ETHYL]ACETAMIDE, ZINC ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-14
公開日2021-04-14
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D1H
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BU of 7d1h by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with D238A mutation
分子名称: Glutaminyl-peptide cyclotransferase, ZINC ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-14
公開日2021-04-14
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
7D2D
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BU of 7d2d by Molmil
Crystal structure of Ixodes scapularis glutaminyl cyclase with a Mn ion bound to the active site
分子名称: Glutaminyl-peptide cyclotransferase, MANGANESE (II) ION
著者Huang, K.-F, Huang, J.-S, Wu, M.-L, Hsieh, W.-L, Wang, A.H.-J.
登録日2020-09-16
公開日2021-04-14
最終更新日2024-11-06
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A Unique Carboxylic-Acid Hydrogen-Bond Network (CAHBN) Confers Glutaminyl Cyclase Activity on M28 Family Enzymes.
J.Mol.Biol., 433, 2021
8UEL
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BU of 8uel by Molmil
Crystal structure of enolase from Litopenaeus vannamei
分子名称: Enolase, MAGNESIUM ION, PHOSPHOENOLPYRUVATE, ...
著者Chang, X, Zhao, G.
登録日2023-10-01
公開日2023-12-13
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献Characterization and Structural Analyses of Enolase from Shrimp ( Litopenaeus vannamei ).
J.Agric.Food Chem., 71, 2023
3FHO
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BU of 3fho by Molmil
Structure of S. pombe Dbp5
分子名称: ATP-dependent RNA helicase dbp5
著者Cheng, Z, Song, H.
登録日2008-12-09
公開日2009-10-13
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Solution and crystal structures of mRNA exporter Dbp5p and its interaction with nucleotides
J.Mol.Biol., 388, 2009
4I60
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BU of 4i60 by Molmil
Crystal structure of avidin - biotinylruthenocene complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Avidin, [(1,2,3,4,5-eta)-cyclopentadienyl][(1,2,3,4,5-eta)-{5-[(3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl]pentanoyl}cyclopentadienyl]ruthenium
著者Strzelczyk, P, Bujacz, A, Bujacz, G.
登録日2012-11-29
公開日2013-08-14
最終更新日2024-11-20
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Structural investigation of the interactions of biotinylruthenocene with avidin.
Chem.Biol.Interact, 204, 2013
7VUM
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BU of 7vum by Molmil
Crystal structure of SSB complexed with que
分子名称: 3,5,7,3',4'-PENTAHYDROXYFLAVONE, Single-stranded DNA-binding protein
著者Lin, E.S, Huang, Y.H, Huang, C.Y.
登録日2021-11-03
公開日2022-03-09
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.319 Å)
主引用文献A Complexed Crystal Structure of a Single-Stranded DNA-Binding Protein with Quercetin and the Structural Basis of Flavonol Inhibition Specificity.
Int J Mol Sci, 23, 2022
9GL5
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BU of 9gl5 by Molmil
X-ray structure of the Thermus thermophilus Q190E mutant of the PilF-GSPIIB domain in the c-di-GMP bound state
分子名称: 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), ACETIC ACID, ATP-binding motif-containing protein pilF, ...
著者Neissner, K, Woehnert, J.
登録日2024-08-27
公開日2025-06-25
最終更新日2025-07-09
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Protonated Glutamate and Aspartate Side Chains Can Recognize Phosphodiester Groups via Strong and Short Hydrogen Bonds in Biomacromolecular Complexes.
Angew.Chem.Int.Ed.Engl., 64, 2025
9GLG
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BU of 9glg by Molmil
X-ray structure of the Thermus thermophilus Q218E mutant of the PilF-GSPIIB domain in the c-di-GMP bound state
分子名称: 9,9'-[(2R,3R,3aS,5S,7aR,9R,10R,10aS,12S,14aR)-3,5,10,12-tetrahydroxy-5,12-dioxidooctahydro-2H,7H-difuro[3,2-d:3',2'-j][1,3,7,9,2,8]tetraoxadiphosphacyclododecine-2,9-diyl]bis(2-amino-1,9-dihydro-6H-purin-6-one), ACETATE ION, ATP-binding motif-containing protein pilF, ...
著者Neissner, K, Woehnert, J.
登録日2024-08-27
公開日2025-06-25
最終更新日2025-07-09
実験手法X-RAY DIFFRACTION (1.55 Å)
主引用文献Protonated Glutamate and Aspartate Side Chains Can Recognize Phosphodiester Groups via Strong and Short Hydrogen Bonds in Biomacromolecular Complexes.
Angew.Chem.Int.Ed.Engl., 64, 2025
6UTM
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BU of 6utm by Molmil
Native E. coli Glyceraldehyde 3-phosphate dehydrogenase
分子名称: GLYCEROL, Glyceraldehyde-3-phosphate dehydrogenase, SN-GLYCEROL-3-PHOSPHATE, ...
著者Rodriguez-Hernandez, A, Romo-Arevalo, E, Rodriguez-Romero, A.
登録日2019-10-29
公開日2019-12-11
最終更新日2024-03-06
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献A Novel Substrate-Binding Site in the X-Ray Structure of an Oxidized E. coli Glyceraldehyde 3-Phosphate Dehydrogenase Elucidated by Single-Wavelength Anomalous Dispersion
Crystals, 9, 2019
7M2T
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BU of 7m2t by Molmil
Crystallographic Structure of the Monoclinic Form of Satellite Tobacco Mosaic Virus
分子名称: Coat protein, MAGNESIUM ION, PHOSPHATE ION, ...
著者McPherson, A.
登録日2021-03-17
公開日2021-12-15
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.71 Å)
主引用文献Structures of additional crystal forms of Satellite tobacco mosaic virus grown from a variety of salts.
Acta Crystallogr.,Sect.F, 77, 2021
9IYK
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BU of 9iyk by Molmil
Crystal structure of hSOD1 in C121 space group
分子名称: ACETATE ION, COPPER (II) ION, SULFATE ION, ...
著者Yapici, I, DeMirci, H.
登録日2024-07-30
公開日2024-08-14
最終更新日2025-05-28
実験手法X-RAY DIFFRACTION (2.34 Å)
主引用文献Structural Insights into the Dynamics of Water in SOD1 Catalysis and Drug Interactions.
Int J Mol Sci, 26, 2025
7A4L
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BU of 7a4l by Molmil
PRE-only solution structure of the Iron-Sulfur protein PioC from Rhodopseudomonas palustris TIE-1
分子名称: IRON/SULFUR CLUSTER, PioC
著者Trindade, I, Invernici, M, Cantini, F, Louro, R, Piccioli, M.
登録日2020-08-19
公開日2020-11-11
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献PRE-driven protein NMR structures: an alternative approach in highly paramagnetic systems.
Febs J., 288, 2021
7U9K
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BU of 7u9k by Molmil
Staphylococcus aureus D-alanine-D-alanine ligase in complex with ATP, D-ala-D-ala, Mg2+ and K+
分子名称: ADENOSINE-5'-DIPHOSPHATE, ADENOSINE-5'-TRIPHOSPHATE, D-alanine--D-alanine ligase, ...
著者Pederick, J.L, Bruning, J.B.
登録日2022-03-10
公開日2023-03-15
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structure-guided design and synthesis of ATP-competitive N-acyl-substituted sulfamide d-alanine-d-alanine ligase inhibitors.
Bioorg.Med.Chem., 96, 2023
6XTK
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BU of 6xtk by Molmil
Y114C Transthyretin structure in complex with Tolcalpone
分子名称: Tolcapone, Transthyretin
著者Varejao, N, Reverter, D, Pinheiro, F, Pallares, I, Ventura, S.
登録日2020-01-16
公開日2020-05-13
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Tolcapone, a potent aggregation inhibitor for the treatment of familial leptomeningeal amyloidosis.
Febs J., 288, 2021
7LK3
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BU of 7lk3 by Molmil
Crystal structure of untwinned human GABARAPL2
分子名称: 1,2-ETHANEDIOL, Gamma-aminobutyric acid receptor-associated protein-like 2
著者Scicluna, K, Dewson, G, Czabotar, P.E, Birkinshaw, R.W.
登録日2021-02-01
公開日2021-05-12
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献A new crystal form of GABARAPL2.
Acta Crystallogr.,Sect.F, 77, 2021
7A58
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BU of 7a58 by Molmil
NOE-only solution structure of the Iron-Sulfur protein PioC from Rhodopseudomonas palustris TIE-1
分子名称: IRON/SULFUR CLUSTER, PioC
著者Cantini, F, Trindade, I.
登録日2020-08-20
公開日2020-11-11
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献PRE-driven protein NMR structures: an alternative approach in highly paramagnetic systems.
Febs J., 288, 2021
7NC4
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BU of 7nc4 by Molmil
Crystal structure of human carbonic anhydrase VII (hCA VII) in complex with a 4-(4-aroylpiperazine-1-carbonyl)benzenesulfonamide derivative.
分子名称: 4-[4-(2-chlorophenyl)carbonylpiperazin-1-yl]carbonylbenzenesulfonamide, Carbonic anhydrase 7, GLYCEROL, ...
著者Di Fiore, A, De Simone, G.
登録日2021-01-28
公開日2021-07-14
最終更新日2024-11-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Design, synthesis and biochemical evaluation of novel carbonic anhydrase inhibitors triggered by structural knowledge on hCA VII.
Bioorg.Med.Chem., 44, 2021

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件を2025-07-09に公開中

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