4Q1F
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![BU of 4q1f by Molmil](/molmil-images/mine/4q1f) | Human dCK C4S-S74E mutant in complex with UDP and the inhibitor 12R {N-{2-[5-(4-{(1R)-1-[(4,6-diaminopyrimidin-2-yl)sulfanyl]ethyl}-5-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]ethyl}methanesulfonamide} | 分子名称: | Deoxycytidine kinase, N-{2-[5-(4-{(1R)-1-[(4,6-diaminopyrimidin-2-yl)sulfanyl]ethyl}-5-methyl-1,3-thiazol-2-yl)-2-methoxyphenoxy]ethyl}methanesulfonamide, URIDINE-5'-DIPHOSPHATE | 著者 | Nomme, J, Lavie, A. | 登録日 | 2014-04-03 | 公開日 | 2014-11-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structure-guided development of deoxycytidine kinase inhibitors with nanomolar affinity and improved metabolic stability. J.Med.Chem., 57, 2014
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4Q1C
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![BU of 4q1c by Molmil](/molmil-images/mine/4q1c) | Human dCK C4S-S74E mutant in complex with UDP and the inhibitor 8 {2,2'-[{4-[(2R)-4-{[(4,6-diaminopyrimidin-2-yl)sulfanyl]methyl}-5-propyl-2,3-dihydro-1,3-thiazol-2-yl]benzene-1,2-diyl}bis(oxy)]diethanol} | 分子名称: | 2,2'-((4-(4-(((4,6-diaminopyrimidin-2-yl)thio)methyl)-5-propylthiazol-2-yl)-1,2-phenylene)bis(oxy))bis(ethan-1-ol), Deoxycytidine kinase, URIDINE-5'-DIPHOSPHATE | 著者 | Nomme, J, Lavie, A. | 登録日 | 2014-04-03 | 公開日 | 2014-11-05 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-guided development of deoxycytidine kinase inhibitors with nanomolar affinity and improved metabolic stability. J.Med.Chem., 57, 2014
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3NBA
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![BU of 3nba by Molmil](/molmil-images/mine/3nba) | Phosphopantetheine Adenylyltranferase from Mycobacterium tuberculosis in complex with adenosine-5'-[(alpha,beta)-methyleno]triphosphate (AMPCPP) | 分子名称: | DIPHOSPHOMETHYLPHOSPHONIC ACID ADENOSYL ESTER, MAGNESIUM ION, Phosphopantetheine adenylyltransferase | 著者 | Wubben, T.J, Mesecar, A.D. | 登録日 | 2010-06-03 | 公開日 | 2010-09-15 | 最終更新日 | 2024-02-21 | 実験手法 | X-RAY DIFFRACTION (2.68 Å) | 主引用文献 | Kinetic, thermodynamic, and structural insight into the mechanism of phosphopantetheine adenylyltransferase from Mycobacterium tuberculosis. J.Mol.Biol., 404, 2010
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4Q7E
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8UBY
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![BU of 8uby by Molmil](/molmil-images/mine/8uby) | Choline-bound FLVCR1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, CHOLINE ION, Heme transporter FLVCR1 | 著者 | Hite, R.K, Son, Y. | 登録日 | 2023-09-25 | 公開日 | 2024-03-27 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (2.67 Å) | 主引用文献 | Structural basis of lipid head group entry to the Kennedy pathway by FLVCR1. Nature, 629, 2024
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8UBZ
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![BU of 8ubz by Molmil](/molmil-images/mine/8ubz) | Choline-bound FLVCR1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, CHOLINE ION, Heme transporter FLVCR1 | 著者 | Hite, R.K, Son, Y. | 登録日 | 2023-09-25 | 公開日 | 2024-03-27 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (3.02 Å) | 主引用文献 | Structural basis of lipid head group entry to the Kennedy pathway by FLVCR1. Nature, 629, 2024
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8UBX
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![BU of 8ubx by Molmil](/molmil-images/mine/8ubx) | Ethanolamine-bound FLVCR1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, ETHANOLAMINE, Heme transporter FLVCR1 | 著者 | Hite, R.K, Son, Y. | 登録日 | 2023-09-25 | 公開日 | 2024-03-27 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Structural basis of lipid head group entry to the Kennedy pathway by FLVCR1. Nature, 629, 2024
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8UBW
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![BU of 8ubw by Molmil](/molmil-images/mine/8ubw) | Choline-bound FLVCR1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, CHOLINE ION, Heme transporter FLVCR1 | 著者 | Hite, R.K, Son, Y. | 登録日 | 2023-09-25 | 公開日 | 2024-03-27 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (2.59 Å) | 主引用文献 | Structural basis of lipid head group entry to the Kennedy pathway by FLVCR1. Nature, 629, 2024
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8UC0
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![BU of 8uc0 by Molmil](/molmil-images/mine/8uc0) | Endogenous ligand bound FLVCR1 | 分子名称: | CHOLESTEROL HEMISUCCINATE, Heme transporter FLVCR1 | 著者 | Hite, R.K, Son, Y. | 登録日 | 2023-09-25 | 公開日 | 2024-03-27 | 最終更新日 | 2024-05-29 | 実験手法 | ELECTRON MICROSCOPY (2.42 Å) | 主引用文献 | Structural basis of lipid head group entry to the Kennedy pathway by FLVCR1. Nature, 629, 2024
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3QVS
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![BU of 3qvs by Molmil](/molmil-images/mine/3qvs) | L-myo-inositol 1-phosphate synthase from Archaeoglobus fulgidus wild type | 分子名称: | GLYCEROL, Myo-inositol-1-phosphate synthase (Ino1), NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Neelon, K, Roberts, M.F, Stec, B. | 登録日 | 2011-02-25 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Crystal structure of a trapped catalytic intermediate suggests that forced atomic proximity drives the catalysis of mIPS. Biophys.J., 101, 2011
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6TGA
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![BU of 6tga by Molmil](/molmil-images/mine/6tga) | Cryo-EM Structure of as isolated form of NAD+-dependent Formate Dehydrogenase from Rhodobacter capsulatus | 分子名称: | 2-AMINO-5,6-DIMERCAPTO-7-METHYL-3,7,8A,9-TETRAHYDRO-8-OXA-1,3,9,10-TETRAAZA-ANTHRACEN-4-ONE GUANOSINE DINUCLEOTIDE, FE2/S2 (INORGANIC) CLUSTER, FLAVIN MONONUCLEOTIDE, ... | 著者 | Wendler, P, Radon, C, Mittelstaedt, G. | 登録日 | 2019-11-15 | 公開日 | 2020-04-22 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (3.26 Å) | 主引用文献 | Cryo-EM structures reveal intricate Fe-S cluster arrangement and charging in Rhodobacter capsulatus formate dehydrogenase. Nat Commun, 11, 2020
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3QW2
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![BU of 3qw2 by Molmil](/molmil-images/mine/3qw2) | L-myo-inositol 1-phosphate synthase from Archaeoglobus mutant N255A | 分子名称: | GLYCEROL, Myo-inositol-1-phosphate synthase (Ino1), NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Neelon, K, Roberts, M.F, Stec, B. | 登録日 | 2011-02-26 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.59 Å) | 主引用文献 | Crystal structure of a trapped catalytic intermediate suggests that forced atomic proximity drives the catalysis of mIPS. Biophys.J., 101, 2011
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8TQM
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3QVW
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![BU of 3qvw by Molmil](/molmil-images/mine/3qvw) | L-myo-inositol 1-phosphate synthase from Archaeoglobus fulgidus mutant K278A | 分子名称: | GLYCEROL, Myo-inositol-1-phosphate synthase (Ino1), NICOTINAMIDE-ADENINE-DINUCLEOTIDE, ... | 著者 | Neelon, K, Roberts, M.F, Stec, B. | 登録日 | 2011-02-26 | 公開日 | 2012-01-11 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Crystal structure of a trapped catalytic intermediate suggests that forced atomic proximity drives the catalysis of mIPS. Biophys.J., 101, 2011
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4Q1D
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![BU of 4q1d by Molmil](/molmil-images/mine/4q1d) | Human dCK C4S-S74E mutant in complex with UDP and the inhibitor 9 {2-{[(1R)-1-{2-[3-(2-fluoroethoxy)-4-methoxyphenyl]-5-propyl-1,3-thiazol-4-yl}ethyl]sulfanyl}pyrimidine-4,6-diamine} | 分子名称: | (R)-2-((1-(2-(3-(2-fluoroethoxy)-4-methoxyphenyl)-5-propylthiazol-4-yl)ethyl)thio)pyrimidine-4,6-diamine, Deoxycytidine kinase, URIDINE-5'-DIPHOSPHATE | 著者 | Nomme, J, Lavie, A. | 登録日 | 2014-04-03 | 公開日 | 2015-02-18 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure-guided development of deoxycytidine kinase inhibitors with nanomolar affinity and improved metabolic stability. J.Med.Chem., 57, 2014
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3OH3
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![BU of 3oh3 by Molmil](/molmil-images/mine/3oh3) | Protein structure of USP from L. major bound to URIDINE-5'-DIPHOSPHATE -Arabinose | 分子名称: | GLYCEROL, UDP-sugar pyrophosphorylase, [(2R,3S,4R,5R)-5-(2,4-dioxo-3,4-dihydropyrimidin-1(2H)-yl)-3,4-dihydroxytetrahydrofuran-2-yl]methyl (2S,3R,4S,5S)-3,4,5-trihydroxytetrahydro-2H-pyran-2-yl dihydrogen diphosphate | 著者 | Dickmanns, A, Damerow, S, Neumann, P, Schulz, E.-C, Lamerz, A, Routier, F, Ficner, R. | 登録日 | 2010-08-17 | 公開日 | 2010-11-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.03 Å) | 主引用文献 | Structural basis for the broad substrate range of the UDP-sugar pyrophosphorylase from Leishmania major. J.Mol.Biol., 405, 2011
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3OH2
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![BU of 3oh2 by Molmil](/molmil-images/mine/3oh2) | Protein structure of USP from L. major bound to URIDINE-5'-DIPHOSPHATE-GALACTOSE | 分子名称: | GALACTOSE-URIDINE-5'-DIPHOSPHATE, GLYCEROL, UDP-sugar pyrophosphorylase | 著者 | Dickmanns, A, Damerow, S, Neumann, P, Schulz, E.-C, Lamerz, A, Routier, F, Ficner, R. | 登録日 | 2010-08-17 | 公開日 | 2010-11-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.14 Å) | 主引用文献 | Structural basis for the broad substrate range of the UDP-sugar pyrophosphorylase from Leishmania major. J.Mol.Biol., 405, 2011
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8TQS
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3OH1
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![BU of 3oh1 by Molmil](/molmil-images/mine/3oh1) | Protein structure of USP from L. major bound to URIDINE-5'-DIPHOSPHATE-Galacturonic acid | 分子名称: | (2S,3R,4S,5R,6R)-6-[[[(2R,3S,4R,5R)-5-(2,4-dioxopyrimidin-1-yl)-3,4-dihydroxy-oxolan-2-yl]methoxy-hydroxy-phosphoryl]oxy-hydroxy-phosphoryl]oxy-3,4,5-trihydroxy-oxane-2-carboxylic acid, GLYCEROL, UDP-sugar pyrophosphorylase | 著者 | Dickmanns, A, Damerow, S, Neumann, P, Schulz, E.-C, Lamerz, A, Routier, F, Ficner, R. | 登録日 | 2010-08-17 | 公開日 | 2010-11-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.18 Å) | 主引用文献 | Structural basis for the broad substrate range of the UDP-sugar pyrophosphorylase from Leishmania major. J.Mol.Biol., 405, 2011
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3OH4
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![BU of 3oh4 by Molmil](/molmil-images/mine/3oh4) | Protein structure of USP from L. major bound to URIDINE-5'-DIPHOSPHATE Glucose | 分子名称: | GLYCEROL, UDP-sugar pyrophosphorylase, URIDINE-5'-DIPHOSPHATE-GLUCOSE | 著者 | Dickmanns, A, Damerow, S, Neumann, P, Schulz, E.-C, Lamerz, A, Routier, F.H, Ficner, R. | 登録日 | 2010-08-17 | 公開日 | 2010-11-17 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (2.21 Å) | 主引用文献 | Structural basis for the broad substrate range of the UDP-sugar pyrophosphorylase from Leishmania major. J.Mol.Biol., 405, 2011
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8TW0
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![BU of 8tw0 by Molmil](/molmil-images/mine/8tw0) | Crystal Structure of a synthetic ABC heterotrimeric Collagen-like Peptide at 1.53 A | 分子名称: | Collagen Mimetic Peptide A, Collagen Mimetic Peptide B, Collagen Mimetic Peptide C, ... | 著者 | Miller, M.D, Cole, C.C, Xu, W, Walker, D.R, Hulgan, S.A.H, Pogostin, B.H, Swain, J.W.R, Duella, R, Misiura, M, Wang, X, Kolomeisky, A.B, Phillips Jr, G.N, Hartgerink, J.D. | 登録日 | 2023-08-18 | 公開日 | 2024-05-29 | 実験手法 | X-RAY DIFFRACTION (1.53 Å) | 主引用文献 | Heterotrimeric Collagen Helix with High Specificity of Assembly Results in a Rapid Rate of Folding Nat.Chem., 2024
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6TFJ
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![BU of 6tfj by Molmil](/molmil-images/mine/6tfj) | Vip3Aa protoxin structure | 分子名称: | Vegetative insecticidal protein | 著者 | Nunez-Ramirez, R, Huesa, J, Bel, Y, Ferre, J, Casino, P, Arias-Palomo, E. | 登録日 | 2019-11-14 | 公開日 | 2020-08-12 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (2.9 Å) | 主引用文献 | Molecular architecture and activation of the insecticidal protein Vip3Aa from Bacillus thuringiensis. Nat Commun, 11, 2020
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4PY7
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![BU of 4py7 by Molmil](/molmil-images/mine/4py7) | Crystal Structure of Fab 3.1 | 分子名称: | antibody 3.1 heavy chain, antibody 3.1 light chain | 著者 | Dreyfus, C. | 登録日 | 2014-03-26 | 公開日 | 2014-05-21 | 最終更新日 | 2014-06-04 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Alternative Recognition of the Conserved Stem Epitope in Influenza A Virus Hemagglutinin by a VH3-30-Encoded Heterosubtypic Antibody. J.Virol., 88, 2014
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3R1R
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3RSR
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![BU of 3rsr by Molmil](/molmil-images/mine/3rsr) | Crystal Structure of 5-NITP Inhibition of Yeast Ribonucleotide Reductase | 分子名称: | 1-{2-DEOXY-5-O-[(R)-HYDROXY{[(R)-HYDROXY(PHOSPHONOOXY)PHOSPHORYL]OXY}PHOSPHORYL]-BETA-D-ERYTHRO-PENTOFURANOSYL}-5-NITRO-1H-INDOLE, MAGNESIUM ION, Ribonucleoside-diphosphate reductase large chain 1 | 著者 | Wan, Q, Mohammed, F, Jha, S, Motea, E, Berdis, A, Dealwis, C.G. | 登録日 | 2011-05-02 | 公開日 | 2012-11-14 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Evaluating the therapeutic potential of a non-natural nucleotide that inhibits human ribonucleotide reductase. Mol.Cancer Ther., 11, 2012
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