7XAR
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 7xar by Molmil](/molmil-images/mine/7xar) | Crystal structure of 3C-like protease from SARS-CoV-2 in complex with covalent inhibitor | 分子名称: | 3C-like proteinase, 4-fluoranyl-~{N}-[(2~{S})-1-[2-(2-fluoranylethanoyl)-2-[[(3~{S})-2-oxidanylidenepyrrolidin-3-yl]methyl]hydrazinyl]-4-methyl-1-oxidanylidene-pentan-2-yl]-1~{H}-indole-2-carboxamide, CHLORIDE ION, ... | 著者 | Caaveiro, J.M.M, Ochi, J, Takahashi, D, Ueda, T, Ojida, A. | 登録日 | 2022-03-18 | 公開日 | 2022-11-09 | 最終更新日 | 2023-11-29 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | Discovery of Chlorofluoroacetamide-Based Covalent Inhibitors for Severe Acute Respiratory Syndrome Coronavirus 2 3CL Protease. J.Med.Chem., 65, 2022
|
|
8E32
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8e32 by Molmil](/molmil-images/mine/8e32) | E. coli 50S ribosome bound to compound streptogramin analogs SA1 and SB1 | 分子名称: | (3R,4R,5E,10E,12E,14S,16R,23S,26aR)-16-fluoro-14-hydroxy-12-methyl-3-(propan-2-yl)-4-(prop-2-yn-1-yl)-3,4,8,9,14,15,16,17,24,25,26,26a-dodecahydro-1H,7H,22H-21,18-(azeno)pyrrolo[2,1-c][1,8,4,19]dioxadiazacyclotetracosine-1,7,22-trione, 23S ribosomal RNA, 50S ribosomal protein L13, ... | 著者 | Pellegrino, J, Lee, D.J, Fraser, J.S, Seiple, I.B. | 登録日 | 2022-08-16 | 公開日 | 2023-06-28 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (2.35 Å) | 主引用文献 | Potential for clicked streptogramin analogs To Be Published
|
|
8E35
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8e35 by Molmil](/molmil-images/mine/8e35) | E. coli 50S ribosome bound to compound SAB002 | 分子名称: | 23S ribosomal RNA, 50S ribosomal protein L13, 50S ribosomal protein L15, ... | 著者 | Pellegrino, J, Lee, D.J, Fraser, J.S, Seiple, I.B. | 登録日 | 2022-08-16 | 公開日 | 2023-06-28 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (2.27 Å) | 主引用文献 | Potential for clicked streptogramin analogs To Be Published
|
|
8E33
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 8e33 by Molmil](/molmil-images/mine/8e33) | E. coli 50S ribosome bound to compound streptogramin analog SAB001 | 分子名称: | 23S ribosomal RNA, 50S ribosomal protein L13, 50S ribosomal protein L15, ... | 著者 | Pellegrino, J, Lee, D.J, Fraser, J.S, Seiple, I.B. | 登録日 | 2022-08-16 | 公開日 | 2023-06-28 | 実験手法 | ELECTRON MICROSCOPY (2.23 Å) | 主引用文献 | Potential for clicked streptogramin analogs To Be Published
|
|
5ZV2
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5zv2 by Molmil](/molmil-images/mine/5zv2) | FGFR-1 in complex with ligand lenvatinib | 分子名称: | 4-{3-chloro-4-[(cyclopropylcarbamoyl)amino]phenoxy}-7-methoxyquinoline-6-carboxamide, Fibroblast growth factor receptor 1 | 著者 | Matsuki, M, Hoshi, T, Yamamoto, Y, Ikemori-Kawada, M, Minoshima, Y, Funahashi, Y, Matsui, J. | 登録日 | 2018-05-09 | 公開日 | 2018-07-11 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.86 Å) | 主引用文献 | Lenvatinib inhibits angiogenesis and tumor fibroblast growth factor signaling pathways in human hepatocellular carcinoma models. Cancer Med, 7, 2018
|
|
5YCH
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ych by Molmil](/molmil-images/mine/5ych) | Ancestral myoglobin aMbWb of Basilosaurus relative (monophyly) | 分子名称: | Ancestral myoglobin aMbWb of Basilosaurus relative (monophyly), PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION | 著者 | Isogai, Y, Imamura, H, Nakae, S, Sumi, T, Takahashi, K, Nakagawa, T, Tsuneshige, A, Shirai, T. | 登録日 | 2017-09-07 | 公開日 | 2018-09-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.354 Å) | 主引用文献 | Tracing whale myoglobin evolution by resurrecting ancient proteins. Sci Rep, 8, 2018
|
|
5YCG
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ycg by Molmil](/molmil-images/mine/5ycg) | Ancestral myoglobin aMbWp of Pakicetus relative | 分子名称: | Ancestral myoglobin aMbWp of Pakicetus relative, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Isogai, Y, Imamura, H, Nakae, S, Sumi, T, Takahashi, K, Nakagawa, T, Tsuneshige, A, Shirai, T. | 登録日 | 2017-09-07 | 公開日 | 2018-09-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Tracing whale myoglobin evolution by resurrecting ancient proteins. Sci Rep, 8, 2018
|
|
5YCI
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yci by Molmil](/molmil-images/mine/5yci) | Ancestral myoglobin aMbWb' of Basilosaurus relative (polyphyly) | 分子名称: | Ancestral myoglobin aMbWb' of Basilosaurus relative (polyphyly), PROTOPORPHYRIN IX CONTAINING FE | 著者 | Isogai, Y, Imamura, H, Nakae, S, Sumi, T, Takahashi, K, Nakagawa, T, Tsuneshige, A, Shirai, T. | 登録日 | 2017-09-07 | 公開日 | 2018-09-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.97 Å) | 主引用文献 | Tracing whale myoglobin evolution by resurrecting ancient proteins. Sci Rep, 8, 2018
|
|
5YCE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yce by Molmil](/molmil-images/mine/5yce) | Sperm whale myoglobin swMb | 分子名称: | Myoglobin, PROTOPORPHYRIN IX CONTAINING FE, SULFATE ION | 著者 | Isogai, Y, Imamura, H, Nakae, S, Sumi, T, Takahashi, K, Nakagawa, T, Tsuneshige, A, Shirai, T. | 登録日 | 2017-09-07 | 公開日 | 2018-09-19 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (0.77 Å) | 主引用文献 | Tracing whale myoglobin evolution by resurrecting ancient proteins. Sci Rep, 8, 2018
|
|
5YCJ
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ycj by Molmil](/molmil-images/mine/5ycj) | Ancestral myoglobin aMbWb' of Basilosaurus relative (polyphyly) imidazole-ligand | 分子名称: | Ancestral myoglobin aMbWb' of Basilosaurus relative (polyphyly), IMIDAZOLE, PROTOPORPHYRIN IX CONTAINING FE | 著者 | Isogai, Y, Imamura, H, Nakae, S, Sumi, T, Takahashi, K, Nakagawa, T, Tsuneshige, A, Shirai, T. | 登録日 | 2017-09-07 | 公開日 | 2018-09-19 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | Tracing whale myoglobin evolution by resurrecting ancient proteins. Sci Rep, 8, 2018
|
|
5WRL
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5wrl by Molmil](/molmil-images/mine/5wrl) | Mu2 subunit of the clathrin adaptor complex AP2 in complex with IRS-1 Y628 peptide | 分子名称: | AP-2 complex subunit mu, Insulin receptor substrate 1 | 著者 | Yoneyama, Y, Niwa, H, Umehara, T, Yokoyama, S, Hakuno, F, Takahashi, S. | 登録日 | 2016-12-02 | 公開日 | 2017-12-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (3.095 Å) | 主引用文献 | IRS-1 acts as an endocytic regulator of IGF-I receptor to facilitate sustained IGF signaling Elife, 7, 2018
|
|
5WRK
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5wrk by Molmil](/molmil-images/mine/5wrk) | Mu2 subunit of the clathrin adaptor complex AP2 in complex with IRS-1 Y608 peptide | 分子名称: | AP-2 complex subunit mu, Insulin receptor substrate 1, NICKEL (II) ION | 著者 | Yoneyama, Y, Niwa, H, Umehara, T, Yokoyama, S, Hakuno, F, Takahashi, S. | 登録日 | 2016-12-02 | 公開日 | 2017-12-06 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | IRS-1 acts as an endocytic regulator of IGF-I receptor to facilitate sustained IGF signaling Elife, 7, 2018
|
|
5XCA
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xca by Molmil](/molmil-images/mine/5xca) | Crystal structure of GH45 endoglucanase EG27II D137A mutant in complex with cellobiose | 分子名称: | Endo-beta-1,4-glucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-22 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XC8
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xc8 by Molmil](/molmil-images/mine/5xc8) | Crystal structure of GH45 endoglucanase EG27II at pH5.5, in complex with cellobiose | 分子名称: | Endo-beta-1,4-glucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-22 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XBX
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xbx by Molmil](/molmil-images/mine/5xbx) | Crystal structure of GH45 endoglucanase EG27II in complex with cellobiose | 分子名称: | Endo-beta-1,4-glucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-21 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.04 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XC4
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xc4 by Molmil](/molmil-images/mine/5xc4) | Crystal structure of GH45 endoglucanase EG27II at pH4.0, in complex with cellobiose | 分子名称: | Endo-beta-1,4-glucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-22 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XC9
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xc9 by Molmil](/molmil-images/mine/5xc9) | Crystal structure of GH45 endoglucanase EG27II at pH8.0, in complex with cellobiose | 分子名称: | Endo-beta-1,4-glucanase, beta-D-glucopyranose-(1-4)-beta-D-glucopyranose | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-22 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.28 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XBU
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xbu by Molmil](/molmil-images/mine/5xbu) | Crystal structure of GH45 endoglucanase EG27II in apo-form | 分子名称: | Endo-beta-1,4-glucanase | 著者 | Nomura, T, Mizutani, K, Iwase, H, Takahashi, N, Mikami, B. | 登録日 | 2017-03-21 | 公開日 | 2018-03-28 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1 Å) | 主引用文献 | High-resolution crystal structures of the glycoside hydrolase family 45 endoglucanase EG27II from the snail Ampullaria crossean. Acta Crystallogr D Struct Biol, 75, 2019
|
|
5XXN
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5xxn by Molmil](/molmil-images/mine/5xxn) | Crystal Structure of mutant (D286N) beta-glucosidase from Bacteroides thetaiotaomicron in complex with sophorose | 分子名称: | DI(HYDROXYETHYL)ETHER, MAGNESIUM ION, Periplasmic beta-glucosidase, ... | 著者 | Nakajima, M, Ishiguro, R, Tanaka, N, Abe, K, Maeda, T, Miyanaga, A, Takahashi, Y, Sugimono, N, Nakai, H, Taguchi, H. | 登録日 | 2017-07-04 | 公開日 | 2017-12-13 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.05 Å) | 主引用文献 | Function and structure relationships of a beta-1,2-glucooligosaccharide-degrading beta-glucosidase. FEBS Lett., 591, 2017
|
|
5YNA
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yna by Molmil](/molmil-images/mine/5yna) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 1 mM alpha-cyclodextrin | 分子名称: | ACETATE ION, CALCIUM ION, Cyclohexakis-(1-4)-(alpha-D-glucopyranose), ... | 著者 | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | 登録日 | 2017-10-24 | 公開日 | 2018-10-24 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.96 Å) | 主引用文献 | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YNC
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ync by Molmil](/molmil-images/mine/5ync) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 1 mM beta-cyclodextrin | 分子名称: | ACETATE ION, CALCIUM ION, Cycloheptakis-(1-4)-(alpha-D-glucopyranose), ... | 著者 | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | 登録日 | 2017-10-24 | 公開日 | 2018-10-24 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.32 Å) | 主引用文献 | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YBW
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ybw by Molmil](/molmil-images/mine/5ybw) | Crystal structure of pyridoxal 5'-phosphate-dependent aspartate racemase | 分子名称: | Aspartate racemase | 著者 | Mizobuchi, T, Nonaka, R, Yoshimura, M, Abe, K, Takahashi, S, Kera, Y, Goto, M. | 登録日 | 2017-09-05 | 公開日 | 2017-12-20 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Crystal structure of a pyridoxal 5'-phosphate-dependent aspartate racemase derived from the bivalve mollusc Scapharca broughtonii Acta Crystallogr F Struct Biol Commun, 73, 2017
|
|
5YKY
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yky by Molmil](/molmil-images/mine/5yky) | Crystal Structure of Cross-Linked Tetragonal Hen Egg White Lysozyme Soaked with 10 mM Rose Bengal and 10mM H2PtCl6 | 分子名称: | CHLORIDE ION, Lysozyme C, PLATINUM (II) ION, ... | 著者 | Tabe, H, Takahashi, H, Shimoi, T, Abe, S, Ueno, T, Yamada, Y. | 登録日 | 2017-10-16 | 公開日 | 2018-09-26 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (1.88 Å) | 主引用文献 | Photocatalytic hydrogen evolution systems constructed in cross-linked porous protein crystals Appl Catal B, 237, 2018
|
|
5YNE
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5yne by Molmil](/molmil-images/mine/5yne) | Crystal structure of Pullulanase from Klebsiella pneumoniae complex at 10 mM alpha-cyclodextrin | 分子名称: | CALCIUM ION, Cyclohexakis-(1-4)-(alpha-D-glucopyranose), DI(HYDROXYETHYL)ETHER, ... | 著者 | Saka, N, Iwamoto, H, Takahashi, N, Mizutani, K, Mikami, B. | 登録日 | 2017-10-24 | 公開日 | 2018-10-24 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.199 Å) | 主引用文献 | Elucidation of the mechanism of interaction between Klebsiella pneumoniae pullulanase and cyclodextrin Acta Crystallogr D Struct Biol, 74, 2018
|
|
5YPX
![Download](/newweb/media/icons/dl.png) ![Visualize](/newweb/media/icons/hoh_3d.png)
![BU of 5ypx by Molmil](/molmil-images/mine/5ypx) | Crystal structure of calaxin with magnesium | 分子名称: | Calaxin, MAGNESIUM ION | 著者 | Shojima, T, Hou, F, Takahashi, Y, Okai, M, Mizuno, K, Inaba, K, Miyakawa, T, Tanokura, M. | 登録日 | 2017-11-04 | 公開日 | 2018-03-14 | 最終更新日 | 2024-03-27 | 実験手法 | X-RAY DIFFRACTION (2.64 Å) | 主引用文献 | Crystal structure of a Ca2+-dependent regulator of flagellar motility reveals the open-closed structural transition Sci Rep, 8, 2018
|
|