1PUA
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![BU of 1pua by Molmil](/molmil-images/mine/1pua) | Crystal Structure of Tetrahymena GCN5 with Bound Coenzyme A and a Phosphorylated, 19-residue Histone H3 peptide | 分子名称: | COENZYME A, HAT A1, Histone H3 | 著者 | Clements, A, Poux, A.N, Lo, W.S, Pillus, L, Berger, S.L, Marmorstein, R. | 登録日 | 2003-06-24 | 公開日 | 2003-09-23 | 最終更新日 | 2023-08-16 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Structural basis for histone and phospho-histone binding by the GCN5 histone acetyltransferase Mol.Cell, 12, 2003
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2FIW
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![BU of 2fiw by Molmil](/molmil-images/mine/2fiw) | Crystal Structure of the GCN5-Related N-acetyltransferase: Aminotransferase, Class-II from Rhodopseudomonas palustris | 分子名称: | ACETYL COENZYME *A, GCN5-related N-acetyltransferase:Aminotransferase, class-II, ... | 著者 | Kim, Y, Skarina, T, Onopriyenko, O, Savchenko, A, Edwards, A, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2005-12-30 | 公開日 | 2006-02-14 | 最終更新日 | 2018-01-24 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Crystal Structure of the GCN5-Related N-acetyltransferase: Aminotransferase, Class-II from Rhodopseudomonas palustris To be Published, 2006
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3TT2
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![BU of 3tt2 by Molmil](/molmil-images/mine/3tt2) | Crystal Structure of GCN5-related N-Acetyltransferase from Sphaerobacter thermophilus | 分子名称: | 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GCN5-related N-acetyltransferase, GLYCEROL, ... | 著者 | Kim, Y, Li, H, Clancy, S, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2011-09-13 | 公開日 | 2011-10-05 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Crystal Structure of GCN5-related N-Acetyltransferase from Sphaerobacter thermophilus To be Published
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2OZG
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![BU of 2ozg by Molmil](/molmil-images/mine/2ozg) | |
2Q0Y
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4MY0
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![BU of 4my0 by Molmil](/molmil-images/mine/4my0) | Crystal Structure of GCN5-related N-acetyltransferase from Kribbella flavida | 分子名称: | 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETYL COENZYME *A, GCN5-related N-acetyltransferase, ... | 著者 | Kim, Y, Mack, J, Endres, M, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2013-09-26 | 公開日 | 2013-11-06 | 実験手法 | X-RAY DIFFRACTION (2.101 Å) | 主引用文献 | Crystal Structure of GCN5-related N-acetyltransferase from Kribbella flavida To be Published
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1R57
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![BU of 1r57 by Molmil](/molmil-images/mine/1r57) | NMR Solution Structure of a GCN5-like putative N-acetyltransferase from Staphylococcus aureus. Northeast Structural Genomics Consortium Target ZR31 | 分子名称: | conserved hypothetical protein | 著者 | Cort, J.R, Acton, T.B, Ma, L, Xiao, R.B, Montelione, G.T, Kennedy, M.A, Northeast Structural Genomics Consortium (NESG) | 登録日 | 2003-10-09 | 公開日 | 2004-03-09 | 最終更新日 | 2024-05-01 | 実験手法 | SOLUTION NMR | 主引用文献 | Structure of an acetyl-CoA binding protein from Staphylococcus aureus representing a novel subfamily of GCN5-related N-acetyltransferase-like proteins. J.STRUCT.FUNCT.GENOM., 9, 2008
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4MY3
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![BU of 4my3 by Molmil](/molmil-images/mine/4my3) | Crystal Structure of GCN5-related N-acetyltransferase from Kribbella flavida | 分子名称: | 1,2-ETHANEDIOL, CHLORIDE ION, GCN5-related N-acetyltransferase | 著者 | Kim, Y, Mack, J, Endres, M, Joachimiak, A, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2013-09-27 | 公開日 | 2013-10-09 | 実験手法 | X-RAY DIFFRACTION (2.57 Å) | 主引用文献 | Crystal Structure of GCN5-related N-acetyltransferase from Kribbella flavida To be Published
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4QNS
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![BU of 4qns by Molmil](/molmil-images/mine/4qns) | Crystal structure of bromodomain from Plasmodium faciparum GCN5, PF3D7_0823300 | 分子名称: | 1,2-ETHANEDIOL, ACETATE ION, Histone acetyltransferase GCN5, ... | 著者 | Fonseca, M, Tallant, C, Knapp, S, Loppnau, P, von Delft, F, Wernimont, A.K, Arrowsmith, C.H, Edwards, A.M, Bountra, C, Hui, R, Structural Genomics Consortium (SGC) | 登録日 | 2014-06-18 | 公開日 | 2014-07-16 | 最終更新日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (1.497 Å) | 主引用文献 | Crystal structure of bromodomain from Plasmodium faciparum GCN5, PF3D7_0823300 TO BE PUBLISHED
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7KPS
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![BU of 7kps by Molmil](/molmil-images/mine/7kps) | Structure of a GNAT superfamily PA3944 acetyltransferase in complex with AcCoA | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, ACETYL COENZYME *A, ... | 著者 | Czub, M.P, Porebski, P.J, Cymborowski, M, Reidl, C.T, Becker, D.P, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2020-11-12 | 公開日 | 2020-11-25 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Gcn5-Related N- Acetyltransferases (GNATs) With a Catalytic Serine Residue Can Play Ping-Pong Too. Front Mol Biosci, 8, 2021
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7KPP
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![BU of 7kpp by Molmil](/molmil-images/mine/7kpp) | Structure of the E102A mutant of a GNAT superfamily PA3944 acetyltransferase | 分子名称: | 1,2-ETHANEDIOL, Acetyltransferase PA3944, COENZYME A, ... | 著者 | Czub, M.P, Porebski, P.J, Majorek, K.A, Cymborowski, M, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2020-11-12 | 公開日 | 2020-11-25 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.45 Å) | 主引用文献 | Gcn5-Related N- Acetyltransferases (GNATs) With a Catalytic Serine Residue Can Play Ping-Pong Too. Front Mol Biosci, 8, 2021
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5VDB
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![BU of 5vdb by Molmil](/molmil-images/mine/5vdb) | Crystal structure of a GNAT superfamily acetyltransferase PA4794 in complex with bisubstrate analog 3 | 分子名称: | (3R,5S,9R,26S)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]-3,5,9-trihydroxy-8,8-dimethyl-10,14,20-trioxo-26-({[(phenylacetyl)amino]acetyl}amino)-2,4,6-trioxa-18-thia-11,15,21-triaza-3,5-diphosphaheptacosan-27-oic acid 3,5-dioxide (non-preferred name), SULFATE ION, acetyltransferase PA4794 | 著者 | Majorek, K.A, Joachimiak, A, Minor, W, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2017-04-01 | 公開日 | 2017-07-26 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Generating enzyme and radical-mediated bisubstrates as tools for investigating Gcn5-related N-acetyltransferases. FEBS Lett., 591, 2017
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5VD6
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![BU of 5vd6 by Molmil](/molmil-images/mine/5vd6) | Crystal structure of a GNAT superfamily acetyltransferase PA4794 in complex with bisubstrate analog 6 | 分子名称: | (3R,5S,9R,23S)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)tetrahydrofuran-2-yl]-3,5,9-trihydroxy-8,8-dimethyl-10,14-dioxo-23-({[(phenylacetyl)amino]acetyl}amino)-2,4,6-trioxa-18-thia-11,15-diaza-3,5-diphosphatetracosan-24-oic acid 3,5-dioxide (non-preferred name), SULFATE ION, acetyltransferase PA4794 | 著者 | Majorek, K.A, Joachimiak, A, Minor, W, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2017-04-01 | 公開日 | 2017-07-26 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (1.2 Å) | 主引用文献 | Generating enzyme and radical-mediated bisubstrates as tools for investigating Gcn5-related N-acetyltransferases. FEBS Lett., 591, 2017
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8E6O
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![BU of 8e6o by Molmil](/molmil-images/mine/8e6o) | Crystal structure of human GCN5 histone acetyltransferase domain | 分子名称: | Histone acetyltransferase KAT2A, S-{(3S,5R,9R)-1-[(2R,3S,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-hydroxy-3-(phosphonooxy)oxolan-2-yl]-3,5,9-trihydroxy-8,8-dimethyl-3,5,10,14-tetraoxo-2,4,6-trioxa-11,15-diaza-3lambda~5~,5lambda~5~-diphosphaheptadecan-17-yl} (2R)-2-hydroxypropanethioate | 著者 | Lu, X.T, Tao, Y.J. | 登録日 | 2022-08-23 | 公開日 | 2024-02-28 | 実験手法 | X-RAY DIFFRACTION (2.37 Å) | 主引用文献 | Crystal structure of human GCN5 histone acetyltransferase domain To Be Published
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3PGP
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![BU of 3pgp by Molmil](/molmil-images/mine/3pgp) | Crystal structure of PA4794 - GNAT superfamily protein in complex with AcCoA | 分子名称: | 1,2-ETHANEDIOL, ACETYL COENZYME *A, CHLORIDE ION, ... | 著者 | Majorek, K.A, Chruszcz, M, Joachimiak, A, Minor, W, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2010-11-02 | 公開日 | 2010-12-01 | 最終更新日 | 2023-09-06 | 実験手法 | X-RAY DIFFRACTION (1.42 Å) | 主引用文献 | Structural, functional, and inhibition studies of a Gcn5-related N-acetyltransferase (GNAT) superfamily protein PA4794: a new C-terminal lysine protein acetyltransferase from pseudomonas aeruginosa. J.Biol.Chem., 288, 2013
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1Z4R
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![BU of 1z4r by Molmil](/molmil-images/mine/1z4r) | Human GCN5 Acetyltransferase | 分子名称: | ACETYL COENZYME *A, General control of amino acid synthesis protein 5-like 2 | 著者 | Dong, A, Bernstein, G, Schuetz, A, Antoshenko, T, Wu, H, Loppnau, P, Sundstrom, M, Arrowsmith, C, Edwards, A, Bochkarev, A, Plotnikov, A, Structural Genomics Consortium (SGC) | 登録日 | 2005-03-16 | 公開日 | 2005-03-29 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (1.74 Å) | 主引用文献 | Crystal structure of a binary complex between human GCN5 histone acetyltransferase domain and acetyl coenzyme A Proteins, 68, 2007
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6EDV
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![BU of 6edv by Molmil](/molmil-images/mine/6edv) | Structure of a GNAT superfamily acetyltransferase PA3944 in complex with CoA | 分子名称: | 1,2-ETHANEDIOL, Acetyltransferase PA3944, CALCIUM ION, ... | 著者 | Majorek, K.A, Satchell, K.J.F, Joachimiak, A, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2018-08-12 | 公開日 | 2018-12-26 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.35 Å) | 主引用文献 | A Gcn5-Related N-Acetyltransferase (GNAT) Capable of Acetylating Polymyxin B and Colistin Antibiotics in Vitro. Biochemistry, 57, 2018
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6EDD
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![BU of 6edd by Molmil](/molmil-images/mine/6edd) | Crystal structure of a GNAT Superfamily PA3944 acetyltransferase in complex with CoA (P1 space group) | 分子名称: | 1,2-ETHANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Acetyltransferase PA3944, ... | 著者 | Czub, M.P, Porebski, P.J, Majorek, K.A, Satchell, K.J, Joachimiak, A, Minor, W, Center for Structural Genomics of Infectious Diseases (CSGID) | 登録日 | 2018-08-09 | 公開日 | 2018-08-22 | 最終更新日 | 2023-10-11 | 実験手法 | X-RAY DIFFRACTION (1.55 Å) | 主引用文献 | A Gcn5-Related N-Acetyltransferase (GNAT) Capable of Acetylating Polymyxin B and Colistin Antibiotics in Vitro. Biochemistry, 57, 2018
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5MKX
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5MKY
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![BU of 5mky by Molmil](/molmil-images/mine/5mky) | BROMODOMAIN OF HUMAN BRD9 WITH 4-chloro-2-methyl-5-((2-methyl-1,2,3,4-tetrahydroisoquinolin-5-yl)amino)pyridazin-3(2H)-one | 分子名称: | 4-chloranyl-2-methyl-5-[(2-methyl-3,4-dihydro-1~{H}-isoquinolin-5-yl)amino]pyridazin-3-one, Bromodomain-containing protein 9 | 著者 | Chung, C.-W. | 登録日 | 2016-12-05 | 公開日 | 2017-12-20 | 最終更新日 | 2024-06-19 | 実験手法 | X-RAY DIFFRACTION (1.67 Å) | 主引用文献 | Discovery of a Potent, Cell Penetrant, and Selective p300/CBP-Associated Factor (PCAF)/General Control Nonderepressible 5 (GCN5) Bromodomain Chemical Probe. J. Med. Chem., 60, 2017
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5MKZ
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5ML0
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![BU of 5ml0 by Molmil](/molmil-images/mine/5ml0) | |
5MLI
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5TPX
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![BU of 5tpx by Molmil](/molmil-images/mine/5tpx) | Bromodomain from Plasmodium Faciparum Gcn5, complexed with compound | 分子名称: | (1S,2S)-N~1~,N~1~-dimethyl-N~2~-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)-1-phenylpropane-1,2-diamine, CHLORIDE ION, Histone acetyltransferase GCN5, ... | 著者 | Lin, Y.H, Hou, C.F.D, MOUSTAKIM, M, DIXON, D.J, Loppnau, P, Tempel, W, Bountra, C, Edwards, A.M, Arrowsmith, C.H, Hui, R, BRENNAN, P.E, Walker, J.R, Structural Genomics Consortium (SGC) | 登録日 | 2016-10-21 | 公開日 | 2017-01-04 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Discovery of a PCAF Bromodomain Chemical Probe. Angew. Chem. Int. Ed. Engl., 56, 2017
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1YK3
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![BU of 1yk3 by Molmil](/molmil-images/mine/1yk3) | Crystal structure of Rv1347c from Mycobacterium tuberculosis | 分子名称: | Hypothetical protein Rv1347c/MT1389, octyl beta-D-glucopyranoside | 著者 | Card, G.L, Peterson, N.A, Smith, C.A, Rupp, B, Schick, B.M, Baker, E.N, TB Structural Genomics Consortium (TBSGC) | 登録日 | 2005-01-16 | 公開日 | 2005-02-01 | 最終更新日 | 2024-03-13 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | The crystal structure of Rv1347c, a putative antibiotic resistance protein from Mycobacterium tuberculosis, reveals a GCN5-related fold and suggests an alternative function in siderophore biosynthesis J.Biol.Chem., 280, 2005
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