4KQR
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![BU of 4kqr by Molmil](/molmil-images/mine/4kqr) | CRYSTAL STRUCTURE OF PENICILLIN-BINDING PROTEIN 3 FROM PSEUDOMONAS AERUGINOSA IN COMPLEX WITH (5S)-Penicilloic Acid | 分子名称: | (2S,4S)-2-[(R)-carboxy{[(2R)-2-{[(4-ethyl-2,3-dioxopiperazin-1-yl)carbonyl]amino}-2-phenylacetyl]amino}methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, CHLORIDE ION, GLYCEROL, ... | 著者 | Nettleship, J.E, Stuart, D.I, Owens, R.J, Ren, J. | 登録日 | 2013-05-15 | 公開日 | 2013-11-06 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.01 Å) | 主引用文献 | Binding of (5S)-Penicilloic Acid to Penicillin Binding Protein 3. Acs Chem.Biol., 8, 2013
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2JCH
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![BU of 2jch by Molmil](/molmil-images/mine/2jch) | Structural and mechanistic basis of penicillin binding protein inhibition by lactivicins | 分子名称: | (2E)-2-({(2S)-2-CARBOXY-2-[(PHENOXYACETYL)AMINO]ETHOXY}IMINO)PENTANEDIOIC ACID, 1,2-ETHANEDIOL, CHLORIDE ION, ... | 著者 | Macheboeuf, P, Fisher, D.S, Brown, T.J, Zervosen, A, Luxen, A, Joris, B, Dessen, A, Schofield, C.J. | 登録日 | 2006-12-23 | 公開日 | 2007-08-14 | 最終更新日 | 2023-12-13 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural and Mechanistic Basis of Penicillin-Binding Protein Inhibition by Lactivicins Nat.Chem.Biol., 3, 2007
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5M19
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![BU of 5m19 by Molmil](/molmil-images/mine/5m19) | Crystal structure of PBP2a from MRSA in the presence of Oxacillin ligand | 分子名称: | CADMIUM ION, Penicillin-binding protein 2, beta-muramic acid | 著者 | Molina, R, Batuecas, M.T, Hermoso, J.A. | 登録日 | 2016-10-07 | 公開日 | 2017-02-08 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Conformational Dynamics in Penicillin-Binding Protein 2a of Methicillin-Resistant Staphylococcus aureus, Allosteric Communication Network and Enablement of Catalysis. J. Am. Chem. Soc., 139, 2017
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5LP5
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![BU of 5lp5 by Molmil](/molmil-images/mine/5lp5) | Complex between Penicillin-Binding Protein (PBP2) and MreC from Helicobacter pylori | 分子名称: | Penicillin-binding protein 2 (Pbp2), Rod shape-determining protein (MreC) | 著者 | Contreras-Martel, C, Martins, A, Ecobichon, C, Maragno, D.M, Mattei, P.J, El Ghachi, M, Hicham, S, Hardouin, P, Boneca, I.G, Dessen, A. | 登録日 | 2016-08-11 | 公開日 | 2017-08-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.74 Å) | 主引用文献 | Molecular architecture of the PBP2-MreC core bacterial cell wall synthesis complex. Nat Commun, 8, 2017
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5M1A
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![BU of 5m1a by Molmil](/molmil-images/mine/5m1a) | Crystal structure of PBP2a from MRSA in the presence of Ceftazidime ligand | 分子名称: | CADMIUM ION, Penicillin-binding protein 2, beta-muramic acid | 著者 | Molina, R, Batuecas, M.T, Hermoso, J.A. | 登録日 | 2016-10-07 | 公開日 | 2017-02-08 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Conformational Dynamics in Penicillin-Binding Protein 2a of Methicillin-Resistant Staphylococcus aureus, Allosteric Communication Network and Enablement of Catalysis. J. Am. Chem. Soc., 139, 2017
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5LP4
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![BU of 5lp4 by Molmil](/molmil-images/mine/5lp4) | Penicillin-Binding Protein (PBP2) from Helicobacter pylori | 分子名称: | Penicillin-binding protein 2 (Pbp2), SULFATE ION | 著者 | Contreras-Martel, C, Martins, A, Ecobichon, C, Maragno, D.M, Mattei, P.J, El Ghachi, M, Boneca, I.G, Dessen, A. | 登録日 | 2016-08-11 | 公開日 | 2017-08-23 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (3.03 Å) | 主引用文献 | Molecular architecture of the PBP2-MreC core bacterial cell wall synthesis complex. Nat Commun, 8, 2017
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5M18
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![BU of 5m18 by Molmil](/molmil-images/mine/5m18) | Crystal structure of PBP2a from MRSA in the presence of Cefepime ligand | 分子名称: | CADMIUM ION, Penicillin-binding protein 2, beta-muramic acid | 著者 | Molina, R, Batuecas, M.T, Hermoso, J.A. | 登録日 | 2016-10-07 | 公開日 | 2017-02-08 | 最終更新日 | 2024-01-17 | 実験手法 | X-RAY DIFFRACTION (1.98 Å) | 主引用文献 | Conformational Dynamics in Penicillin-Binding Protein 2a of Methicillin-Resistant Staphylococcus aureus, Allosteric Communication Network and Enablement of Catalysis. J. Am. Chem. Soc., 139, 2017
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5OAU
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![BU of 5oau by Molmil](/molmil-images/mine/5oau) | |
3VSL
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![BU of 3vsl by Molmil](/molmil-images/mine/3vsl) | Crystal structure of penicillin-binding protein 3 (PBP3) from methicilin-resistant Staphylococcus aureus in the cefotaxime bound form. | 分子名称: | CEFOTAXIME, C3' cleaved, open, ... | 著者 | Yoshida, H, Tame, J.R, Park, S.Y. | 登録日 | 2012-04-25 | 公開日 | 2012-10-31 | 最終更新日 | 2017-03-15 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Crystal Structures of Penicillin-Binding Protein 3 (PBP3) from Methicillin-Resistant Staphylococcus aureus in the Apo and Cefotaxime-Bound Forms. J.Mol.Biol., 423, 2012
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3ZG0
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![BU of 3zg0 by Molmil](/molmil-images/mine/3zg0) | Crystal structure of ceftaroline acyl-PBP2a from MRSA with non- covalently bound ceftaroline and muramic acid at allosteric site obtained by cocrystallization | 分子名称: | CADMIUM ION, CHLORIDE ION, Ceftaroline, ... | 著者 | Otero, L.H, Rojas-Altuve, A, Hermoso, J.A. | 登録日 | 2012-12-13 | 公開日 | 2013-10-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | How Allosteric Control of Staphylococcus Aureus Penicillin Binding Protein 2A Enables Methicillin Resistance and Physiological Function Proc.Natl.Acad.Sci.USA, 110, 2013
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3ZFZ
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![BU of 3zfz by Molmil](/molmil-images/mine/3zfz) | Crystal structure of ceftaroline acyl-PBP2a from MRSA with non- covalently bound ceftaroline and muramic acid at allosteric site obtained by soaking | 分子名称: | CADMIUM ION, CHLORIDE ION, Ceftaroline, ... | 著者 | Otero, L.H, Rojas-Altuve, A, Hermoso, J.A. | 登録日 | 2012-12-13 | 公開日 | 2013-10-09 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.25 Å) | 主引用文献 | How Allosteric Control of Staphylococcus Aureus Penicillin Binding Protein 2A Enables Methicillin Resistance and Physiological Function Proc.Natl.Acad.Sci.USA, 110, 2013
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3ZGA
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![BU of 3zga by Molmil](/molmil-images/mine/3zga) | Crystal Structure of Penicillin-Binding Protein 4 from Listeria monocytogenes in the Carbenicillin bound form | 分子名称: | (2R,4S)-2-[(1R)-1-{[(2S)-2-carboxy-2-phenylacetyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, GLYCEROL, PENICILLIN-BINDING PROTEIN 4 | 著者 | Jeong, J.H, Kim, Y.G. | 登録日 | 2012-12-17 | 公開日 | 2013-05-29 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.005 Å) | 主引用文献 | Crystal Structures of Bifunctional Penicillin-Binding Protein 4 from Listeria Monocytogenes. Antimicrob.Agents Chemother., 57, 2013
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3ZG5
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![BU of 3zg5 by Molmil](/molmil-images/mine/3zg5) | Crystal structure of PBP2a from MRSA in complex with peptidoglycan analogue at allosteric | 分子名称: | CADMIUM ION, CHLORIDE ION, PEPTIDOGLYCAN ANALOGUE, ... | 著者 | Otero, L.H, Rojas-Altuve, A, Hermoso, J.A. | 登録日 | 2012-12-14 | 公開日 | 2013-10-09 | 最終更新日 | 2024-02-07 | 実験手法 | X-RAY DIFFRACTION (2.55 Å) | 主引用文献 | How Allosteric Control of Staphylococcus Aureus Penicillin Binding Protein 2A Enables Methicillin Resistance and Physiological Function Proc.Natl.Acad.Sci.USA, 110, 2013
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3ZG9
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![BU of 3zg9 by Molmil](/molmil-images/mine/3zg9) | |
3ZG7
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![BU of 3zg7 by Molmil](/molmil-images/mine/3zg7) | |
4BL3
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![BU of 4bl3 by Molmil](/molmil-images/mine/4bl3) | Crystal structure of PBP2a clinical mutant N146K from MRSA | 分子名称: | CADMIUM ION, CHLORIDE ION, PENICILLIN BINDING PROTEIN 2 PRIME, ... | 著者 | Otero, L.H, Rojas-Altuve, A, Carrasco-Lopez, C, Hermoso, J.A. | 登録日 | 2013-04-30 | 公開日 | 2014-05-21 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (3 Å) | 主引用文献 | Disruption of Allosteric Response as an Unprecedented Mechanism of Resistance to Antibiotics. J.Am.Chem.Soc., 136, 2014
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3ZG8
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![BU of 3zg8 by Molmil](/molmil-images/mine/3zg8) | Crystal Structure of Penicillin Binding Protein 4 from Listeria monocytogenes in the Ampicillin bound form | 分子名称: | (2R,4S)-2-[(1R)-1-{[(2R)-2-amino-2-phenylacetyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, GLYCEROL, PENICILLIN-BINDING PROTEIN, ... | 著者 | Jeong, J.H, Kim, Y.G. | 登録日 | 2012-12-17 | 公開日 | 2013-05-29 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.094 Å) | 主引用文献 | Crystal Structures of Bifunctional Penicillin-Binding Protein 4 from Listeria Monocytogenes. Antimicrob.Agents Chemother., 57, 2013
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4BL2
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![BU of 4bl2 by Molmil](/molmil-images/mine/4bl2) | |
4QJG
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![BU of 4qjg by Molmil](/molmil-images/mine/4qjg) | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with penicillin V | 分子名称: | (2R,4S)-5,5-dimethyl-2-{(1R)-2-oxo-1-[(phenoxyacetyl)amino]ethyl}-1,3-thiazolidine-4-carboxylic acid, Peptidoglycan glycosyltransferase | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Clancy, S, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2014-06-03 | 公開日 | 2014-07-09 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.85 Å) | 主引用文献 | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with penicillin V To be Published
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6SYN
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![BU of 6syn by Molmil](/molmil-images/mine/6syn) | Crystal structure of Y. pestis penicillin-binding protein 3 | 分子名称: | (2R,4S)-2-[(1R)-1-{[(2S)-2-carboxy-2-phenylacetyl]amino}-2-oxoethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, ACETATE ION, Peptidoglycan D,D-transpeptidase FtsI | 著者 | Pankov, G, Hunter, W.N, Dawson, A. | 登録日 | 2019-09-30 | 公開日 | 2020-10-14 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.63 Å) | 主引用文献 | The structure of penicillin-binding protein 3 from Yersinia pestis To Be Published
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4R0Q
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![BU of 4r0q by Molmil](/molmil-images/mine/4r0q) | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cephalothin | 分子名称: | 2-[3-(2-HYDROXY-1,1-DIHYDROXYMETHYL-ETHYLAMINO)-PROPYLAMINO]-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, CEPHALOTHIN GROUP, Peptidoglycan glycosyltransferase, ... | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Clancy, S, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2014-08-01 | 公開日 | 2014-08-27 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2 Å) | 主引用文献 | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cephalothin To be Published
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4R1G
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![BU of 4r1g by Molmil](/molmil-images/mine/4r1g) | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cloxacillin | 分子名称: | CLOXACILLIN (OPEN FORM), Peptidoglycan glycosyltransferase | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Clancy, S, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2014-08-05 | 公開日 | 2014-08-27 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.92 Å) | 主引用文献 | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cloxacillin To be Published
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4R3J
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![BU of 4r3j by Molmil](/molmil-images/mine/4r3j) | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cefapirin | 分子名称: | (2R)-2-[(1R)-1-(acetylamino)-2-oxoethyl]-5-methyl-3,6-dihydro-2H-1,3-thiazine-4-carboxylic acid, GLYCEROL, PHOSPHATE ION, ... | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Clancy, S, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2014-08-15 | 公開日 | 2014-09-17 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (2.44 Å) | 主引用文献 | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with cefapirin To be Published
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6TII
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![BU of 6tii by Molmil](/molmil-images/mine/6tii) | |
4RA7
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![BU of 4ra7 by Molmil](/molmil-images/mine/4ra7) | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with nafcillin | 分子名称: | (2R,4S)-2-[(1R)-2-hydroxy-1-{[(2-hydroxynaphthalen-1-yl)carbonyl]amino}ethyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, Peptidoglycan glycosyltransferase | 著者 | Filippova, E.V, Minasov, G, Kiryukhina, O, Clancy, S, Joachimiak, A, Anderson, W.F, Midwest Center for Structural Genomics (MCSG) | 登録日 | 2014-09-09 | 公開日 | 2014-09-24 | 最終更新日 | 2023-12-06 | 実験手法 | X-RAY DIFFRACTION (1.94 Å) | 主引用文献 | Structure of a putative peptidoglycan glycosyltransferase from Atopobium parvulum in complex with nafcillin To be Published
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