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2CHG
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Replication Factor C domains 1 and 2
分子名称: MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, REPLICATION FACTOR C SMALL SUBUNIT
著者Seybert, A, Singleton, M.R, Cook, N, Hall, D.R, Wigley, D.B.
登録日2006-03-14
公開日2006-06-06
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Communication between Subunits within an Archaeal Clamp-Loader Complex.
Embo J., 25, 2006
2CHH
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RALSTONIA SOLANACEARUM HIGH-AFFINITY MANNOSE-BINDING LECTIN
分子名称: CALCIUM ION, PROTEIN RSC3288, UNKNOWN ATOM OR ION, ...
著者Mitchell, E.P, Wimmerova, M, Imberty, A.
登録日2006-03-15
公開日2006-03-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1 Å)
主引用文献A new Ralstonia solanacearum high-affinity mannose-binding lectin RS-IIL structurally resembling the Pseudomonas aeruginosa fucose-specific lectin PA-IIL.
Mol. Microbiol., 52, 2004
2CHI
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Recombinant human H ferritin, K86Q and E27D mutant
分子名称: CALCIUM ION, FERRITIN HEAVY CHAIN, GLYCEROL, ...
著者Toussaint, L, Crichton, R.R, Declercq, J.P.
登録日2006-03-15
公開日2006-12-13
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献High-Resolution X-Ray Structures of Human Apoferritin H-Chain Mutants Correlated with Their Activity and Metal-Binding Sites.
J.Mol.Biol., 365, 2007
2CHJ
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NMR structure of TGLGLT quadruplex
分子名称: 5'-D(*TP*G LCGP*G LCGP*TP)-3'
著者Nielsen, J.T, Petersen, M.
登録日2006-03-15
公開日2006-04-19
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献NMR Solution Structures of Lna (Locked Nucleic Acid) Modified Quadruplexes
Nucleic Acids Res., 34, 2006
2CHK
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NMR structure of TLLLLT quadruplex
分子名称: 5'-D(*T LCG LCG LCG LCGP*TP)-3'
著者Nielsen, J.T, Petersen, M.
登録日2006-03-15
公開日2006-04-19
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献NMR Solution Structures of Lna (Locked Nucleic Acid) Modified Quadruplexes
Nucleic Acids Res., 34, 2006
2CHL
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Structure of casein kinase 1 gamma 3
分子名称: 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE, CASEIN KINASE I ISOFORM GAMMA-3, SULFATE ION
著者Bunkoczi, G, Salah, E, Rellos, P, Das, S, Fedorov, O, Savitsky, P, Gileadi, O, Sundstrom, M, Edwards, A, Arrowsmith, C, Ugochukwu, E, Weigelt, J, von Delft, F, Knapp, S.
登録日2006-03-15
公開日2006-03-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure of Casein Kinase 1 Gamma 3
To be Published
2CHM
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Crystal structure of N2 substituted pyrazolo pyrimidinones - a flipped binding mode in PDE5
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 5-[2-(BUT-3-EN-1-YLOXY)-5-(1-HYDROXYVINYL)PYRIDIN-3-YL]-3-ETHYL-2-(1-ETHYLAZETIDIN-3-YL)-1,2,6,7A-TETRAHYDRO-7H-PYRAZOLO[4,3-D]PYRIMIDIN-7-ONE, CGMP-SPECIFIC 3', ...
著者Allerton, C.M.N, Barber, C.G, Beaumont, K.C, Brown, D.G, Cole, S.M, Ellis, D, Lane, C.A.L, Maw, G.N, Mount, N.M, Rawson, D.J, Robinson, C.M, Street, S.D.A, Summerhill, N.W.
登録日2006-03-15
公開日2006-06-08
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献A Novel Series of Potent and Selective Pde5 Inhibitors with Potential for High and Dose-Independent Oral Bioavailability
J.Med.Chem., 49, 2006
2CHN
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Bacteroides thetaiotaomicron hexosaminidase with O-GlcNAcase activity- NAG-thiazoline complex
分子名称: 3AR,5R,6S,7R,7AR-5-HYDROXYMETHYL-2-METHYL-5,6,7,7A-TETRAHYDRO-3AH-PYRANO[3,2-D]THIAZOLE-6,7-DIOL, CALCIUM ION, GLUCOSAMINIDASE, ...
著者Dennis, R.J, Taylor, E.J, Macauley, M.S, Stubbs, K.A, Turkenburg, J.P, Hart, S.J, Black, G.N, Vocadlo, D.J, Davies, G.J.
登録日2006-03-15
公開日2006-05-08
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure and Mechanism of a Bacterial B-Glucosaminidase Having O-Glcnacase Activity
Nat.Struct.Mol.Biol., 13, 2006
2CHO
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Bacteroides thetaiotaomicron hexosaminidase with O-GlcNAcase activity
分子名称: ACETATE ION, CALCIUM ION, GLUCOSAMINIDASE, ...
著者Dennis, R.J, Taylor, E.J, Macauley, M.S, Stubbs, K.A, Turkenburg, J.P, Hart, S.J, Black, G.N, Vocadlo, D.J, Davies, G.J.
登録日2006-03-16
公開日2006-06-19
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Structure and Mechanism of a Bacterial B-Glucosaminidase Having O-Glcnacase Activity
Nat.Struct.Mol.Biol., 13, 2006
2CHP
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Crystal structure of the dodecameric ferritin MrgA from B. subtilis 168
分子名称: METALLOREGULATION DNA-BINDING STRESS PROTEIN, PHOSPHATE ION
著者Essen, L.-O, Morbitzer, A.
登録日2006-03-16
公開日2007-04-03
最終更新日2024-05-01
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Morphology of Dry Solid-Supported Protein Monolayers Dependent on the Substrate and Protein Surface Properties.
Langmuir, 22, 2006
2CHQ
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Replication Factor C ADPNP complex
分子名称: PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, REPLICATION FACTOR C SMALL SUBUNIT
著者Seybert, A, Singleton, M.R, Cook, N, Hall, D.R, Wigley, D.B.
登録日2006-03-16
公開日2006-06-06
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献Communication between Subunits within an Archaeal Clamp-Loader Complex.
Embo J., 25, 2006
2CHR
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A RE-EVALUATION OF THE CRYSTAL STRUCTURE OF CHLOROMUCONATE CYCLOISOMERASE
分子名称: CHLORIDE ION, CHLOROMUCONATE CYCLOISOMERASE, MANGANESE (II) ION
著者Kleywegt, G.J, Jones, T.A.
登録日1995-02-24
公開日1995-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献A re-evaluation of the crystal structure of chloromuconate cycloisomerase.
Acta Crystallogr.,Sect.D, 52, 1996
2CHS
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CRYSTAL STRUCTURES OF THE MONOFUNCTIONAL CHORISMATE MUTASE FROM BACILLUS SUBTILIS AND ITS COMPLEX WITH A TRANSITION STATE ANALOG
分子名称: CHORISMATE MUTASE
著者Chook, Y.M, Ke, H, Lipscomb, W.N.
登録日1994-04-08
公開日1994-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structures of the monofunctional chorismate mutase from Bacillus subtilis and its complex with a transition state analog.
Proc.Natl.Acad.Sci.USA, 90, 1993
2CHT
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CRYSTAL STRUCTURES OF THE MONOFUNCTIONAL CHORISMATE MUTASE FROM BACILLUS SUBTILIS AND ITS COMPLEX WITH A TRANSITION STATE ANALOG
分子名称: 8-HYDROXY-2-OXA-BICYCLO[3.3.1]NON-6-ENE-3,5-DICARBOXYLIC ACID, CHORISMATE MUTASE
著者Chook, Y.M, Ke, H, Lipscomb, W.N.
登録日1994-04-08
公開日1994-07-31
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Crystal structures of the monofunctional chorismate mutase from Bacillus subtilis and its complex with a transition state analog.
Proc.Natl.Acad.Sci.USA, 90, 1993
2CHU
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CeuE in complex with mecam
分子名称: ENTEROCHELIN UPTAKE PERIPLASMIC BINDING PROTEIN, FE (III) ION, N,N',N''-[BENZENE-1,3,5-TRIYLTRIS(METHYLENE)]TRIS(2,3-DIHYDROXYBENZAMIDE), ...
著者Muller, A, Wilkinson, A.J, Wilson, K.S, Duhme-Klair, A.K.
登録日2006-03-16
公開日2006-08-14
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献An [{Fe(Mecam)}(2)](6-) Bridge in the Crystal Structure of a Ferric Enterobactin Binding Protein.
Angew.Chem.Int.Ed.Engl., 45, 2006
2CHV
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Replication Factor C ADPNP complex
分子名称: REPLICATION FACTOR C SMALL SUBUNIT
著者Seybert, A, Singleton, M.R, Cook, N, Hall, D.R, Wigley, D.B.
登録日2006-03-16
公開日2006-06-06
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Communication between Subunits within an Archaeal Clamp-Loader Complex.
Embo J., 25, 2006
2CHW
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A pharmacological map of the PI3-K family defines a role for p110 alpha in signaling: The structure of complex of phosphoinositide 3- kinase gamma with inhibitor PIK-39
分子名称: 2-((9H-PURIN-6-YLTHIO)METHYL)-5-CHLORO-3-(2-METHOXYPHENYL)QUINAZOLIN-4(3H)-ONE, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM
著者Knight, Z.A, Gonzalez, B, Feldman, M.E, Zunder, E.R, Goldenberg, D.D, Williams, O, Loewith, R, Stokoe, D, Balla, A, Toth, B, Balla, T, Weiss, W.A, Williams, R.L, Shokat, K.M.
登録日2006-03-16
公開日2006-05-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献A Pharmacological Map of the Pi3-K Family Defines a Role for P110Alpha in Signaling
Cell(Cambridge,Mass.), 125, 2006
2CHX
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A pharmacological map of the PI3-K family defines a role for p110alpha in signaling: The structure of complex of phosphoinositide 3-kinase gamma with inhibitor PIK-90
分子名称: N-(2,3-DIHYDRO-7,8-DIMETHOXYIMIDAZO[1,2-C] QUINAZOLIN-5-YL)NICOTINAMIDE, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM
著者Knight, Z.A, Gonzalez, B, Feldman, M.E, Zunder, E.R, Goldenberg, D.D, Williams, O, Loewith, R, Stokoe, D, Balla, A, Toth, B, Balla, T, Weiss, W.A, Williams, R.L, Shokat, K.M.
登録日2006-03-16
公開日2006-05-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献A Pharmacological Map of the Pi3-K Family Defines a Role for P110Alpha in Signaling
Cell(Cambridge,Mass.), 125, 2006
2CHY
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THREE-DIMENSIONAL STRUCTURE OF CHEY, THE RESPONSE REGULATOR OF BACTERIAL CHEMOTAXIS
分子名称: CHEY
著者Mottonen, J.M, Stock, A.M, Stock, J.B, Schutt, C.E.
登録日1990-05-17
公開日1990-07-15
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Three-dimensional structure of CheY, the response regulator of bacterial chemotaxis.
Nature, 337, 1989
2CHZ
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A pharmacological map of the PI3-K family defines a role for p110alpha in signaling: The structure of complex of phosphoinositide 3-kinase gamma with inhibitor PIK-93
分子名称: N-(5-(4-CHLORO-3-(2-HYDROXY-ETHYLSULFAMOYL)- PHENYLTHIAZOLE-2-YL)-ACETAMIDE, PHOSPHATIDYLINOSITOL-4,5-BISPHOSPHATE 3-KINASE CATALYTIC SUBUNIT GAMMA ISOFORM
著者Knight, Z.A, Gonzalez, B, Feldman, M.E, Zunder, E.R, Goldenberg, D.D, Williams, O, Loewith, R, Stokoe, D, Balla, A, Toth, B, Balla, T, Weiss, W.A, Williams, R.L, Shokat, K.M.
登録日2006-03-16
公開日2006-05-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献A Pharmacological Map of the Pi3-K Family Defines a Role for P110Alpha in Signaling
Cell(Cambridge,Mass.), 125, 2006
2CI0
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High throughput screening and x-ray crystallography assisted evaluation of small molecule scaffolds for CYP51 inhibitors
分子名称: (2R)-2-PHENYL-N-PYRIDIN-4-YLBUTANAMIDE, CYTOCHROME P450 51, PROTOPORPHYRIN IX CONTAINING FE
著者Podust, L.M, Kim, Y, Yermalitskaya, L.V, Von Kries, J.P, Waterman, M.R.
登録日2006-03-16
公開日2007-07-03
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.53 Å)
主引用文献Small Molecule Scaffolds for Cyp51 Inhibitors Identified by High Throughput Screening and Defined by X-Ray Crystallography
Antimicrob.Agents Chemother., 51, 2007
2CI1
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Crystal Structure of dimethylarginine dimethylaminohydrolase I in complex with S-nitroso-Lhomocysteine
分子名称: CITRIC ACID, NG, NG-DIMETHYLARGININE DIMETHYLAMINOHYDROLASE 1
著者Frey, D, Braun, O, Briand, C, Vasak, M, Grutter, M.G.
登録日2006-03-17
公開日2006-05-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.08 Å)
主引用文献Structure of the Mammalian Nos Regulator Dimethylarginine Dimethylaminohydrolase: A Basis for the Design of Specific Inhibitors.
Structure, 14, 2006
2CI2
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CRYSTAL AND MOLECULAR STRUCTURE OF THE SERINE PROTEINASE INHIBITOR CI-2 FROM BARLEY SEEDS
分子名称: CHYMOTRYPSIN INHIBITOR 2
著者Mcphalen, C.A, James, M.N.G.
登録日1988-09-05
公開日1988-09-07
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal and molecular structure of the serine proteinase inhibitor CI-2 from barley seeds.
Biochemistry, 26, 1987
2CI3
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Crystal Structure of Dimethylarginine dimethylaminohydrolase crystal form I
分子名称: NG, NG-DIMETHYLARGININE DIMETHYLAMINOHYDROLASE 1
著者Frey, D, Braun, O, Briand, C, Vasak, M, Grutter, M.G.
登録日2006-03-17
公開日2006-05-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of the Mammalian Nos Regulator Dimethylarginine Dimethylaminohydrolase: A Basis for the Design of Specific Inhibitors.
Structure, 14, 2006
2CI4
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Crystal Structure of Dimethylarginine dimethylaminohydrolase I crystal form II
分子名称: NG, NG-DIMETHYLARGININE DIMETHYLAMINOHYDROLASE 1
著者Frey, D, Braun, O, Briand, C, Vasak, M, Grutter, M.G.
登録日2006-03-17
公開日2006-05-17
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure of the Mammalian Nos Regulator Dimethylarginine Dimethylaminohydrolase: A Basis for the Design of Specific Inhibitors.
Structure, 14, 2006

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