8V3O
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![BU of 8v3o by Molmil](/molmil-images/mine/8v3o) | CCP5 in complex with Glu-P-peptide 1 transition state analog | 分子名称: | Cytosolic carboxypeptidase-like protein 5, D-MALATE, POTASSIUM ION, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation Nature, 2024
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8V3M
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![BU of 8v3m by Molmil](/molmil-images/mine/8v3m) | CCP5 apo structure | 分子名称: | Cytosolic carboxypeptidase-like protein 5, D-MALATE, IMIDAZOLE, ... | 著者 | Chen, J, Zehr, E.A, Gruschus, J.M, Szyk, A, Liu, Y, Tanner, M.E, Tjandra, N, Roll-Mecak, A. | 登録日 | 2023-11-28 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Tubulin code eraser CCP5 binds branch glutamates by substrate deformation Nature, 2024
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9FZK
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![BU of 9fzk by Molmil](/molmil-images/mine/9fzk) | |
9FZC
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![BU of 9fzc by Molmil](/molmil-images/mine/9fzc) | |
8W4D
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![BU of 8w4d by Molmil](/molmil-images/mine/8w4d) | |
8W4C
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![BU of 8w4c by Molmil](/molmil-images/mine/8w4c) | The sigma-1 receptor from Xenopus laevis in complex with progesterone by soaking | 分子名称: | PROGESTERONE, Sigma non-opioid intracellular receptor 1 | 著者 | Xiao, Y, Fu, C, Sun, Z, Zhou, X. | 登録日 | 2023-08-23 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.676 Å) | 主引用文献 | Insight into binding of endogenous neurosteroid ligands to the sigma-1 receptor. Nat Commun, 15, 2024
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8W4B
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![BU of 8w4b by Molmil](/molmil-images/mine/8w4b) | The sigma-1 receptor from Xenopus laevis in complex with progesterone by co-crystallization | 分子名称: | PROGESTERONE, Sigma non-opioid intracellular receptor 1 | 著者 | Xiao, Y, Fu, C, Sun, Z, Zhou, X. | 登録日 | 2023-08-23 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.152 Å) | 主引用文献 | Insight into binding of endogenous neurosteroid ligands to the sigma-1 receptor. Nat Commun, 15, 2024
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8WWB
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![BU of 8wwb by Molmil](/molmil-images/mine/8wwb) | |
8WUE
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![BU of 8wue by Molmil](/molmil-images/mine/8wue) | |
8X20
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![BU of 8x20 by Molmil](/molmil-images/mine/8x20) | HIV-1 reverse transcriptase mutant Q151M/Y115F/F116Y/L74V:DNA:E-CFCP-TP ternary complex | 分子名称: | DNA/RNA (38-MER), E-CFCP-triphosphate, GLYCEROL, ... | 著者 | Yasutake, Y, Hattori, S.I, Mitsuya, H. | 登録日 | 2023-11-09 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.7 Å) | 主引用文献 | Deviated binding of anti-HBV nucleoside analog E-CFCP-TP to the reverse transcriptase active site attenuates the effect of drug-resistant mutations. Sci Rep, 14, 2024
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8X21
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![BU of 8x21 by Molmil](/molmil-images/mine/8x21) | HIV-1 reverse transcriptase mutant Q151M/Y115F/F116Y/L74V:DNA:ETV-TP ternary complex | 分子名称: | DNA/RNA (38-MER), GLYCEROL, HIV-1 RT p51 subunit, ... | 著者 | Yasutake, Y, Hattori, S.I, Mitsuya, H. | 登録日 | 2023-11-09 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.33 Å) | 主引用文献 | Deviated binding of anti-HBV nucleoside analog E-CFCP-TP to the reverse transcriptase active site attenuates the effect of drug-resistant mutations. Sci Rep, 14, 2024
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8X1Z
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![BU of 8x1z by Molmil](/molmil-images/mine/8x1z) | HIV-1 reverse transcriptase mutant Q151M/Y115F/F116Y:DNA:E-CFCP-TP ternary complex | 分子名称: | DNA/RNA (38-MER), E-CFCP-triphosphate, GLYCEROL, ... | 著者 | Yasutake, Y, Hattori, S.I, Mitsuya, H. | 登録日 | 2023-11-09 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.62 Å) | 主引用文献 | Deviated binding of anti-HBV nucleoside analog E-CFCP-TP to the reverse transcriptase active site attenuates the effect of drug-resistant mutations. Sci Rep, 14, 2024
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8YBB
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![BU of 8ybb by Molmil](/molmil-images/mine/8ybb) | |
6Y6S
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![BU of 6y6s by Molmil](/molmil-images/mine/6y6s) | Mouse Galactocerebrosidase complexed with galacto-noeurostegine GNS at pH 6.8 | 分子名称: | (1~{R},2~{S},3~{S},4~{R},5~{R})-4-(hydroxymethyl)-8-azabicyclo[3.2.1]octane-1,2,3-triol, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Deane, J.E, McLoughlin, J. | 登録日 | 2020-02-27 | 公開日 | 2021-01-13 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | The Bicyclic Form of galacto -Noeurostegine Is a Potent Inhibitor of beta-Galactocerebrosidase. Acs Med.Chem.Lett., 12, 2021
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8VVK
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![BU of 8vvk by Molmil](/molmil-images/mine/8vvk) | CCHFV GP38 bound to ADI-46143 Fab | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ADI-46143 Fab Heavy Chain, ADI-46143 Fab Light Chain, ... | 著者 | Hjorth, C.K, McLellan, J.S. | 登録日 | 2024-01-31 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.61 Å) | 主引用文献 | Crimean-Congo Hemorrhagic Fever Survivors Elicit Protective Non-Neutralizing Antibodies that Target 11 Overlapping Regions on Viral Glycoprotein GP38 To Be Published
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9FE7
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![BU of 9fe7 by Molmil](/molmil-images/mine/9fe7) | Crystal Structure of oxidized NuoEF variant P228R(NuoF) from Aquifex aeolicus | 分子名称: | 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.28 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FE5
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![BU of 9fe5 by Molmil](/molmil-images/mine/9fe5) | Crystal Structure of NuoEF variant R66G(NuoF) from Aquifex aeolicus bound to NADH under anoxic conditions after 10 min soaking | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, CHLORIDE ION, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.1 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FE8
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![BU of 9fe8 by Molmil](/molmil-images/mine/9fe8) | Crystal Structure of reduced NuoEF variant P228R(NuoF) from Aquifex aeolicus | 分子名称: | 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, 3[N-MORPHOLINO]PROPANE SULFONIC ACID, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.34 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FDJ
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![BU of 9fdj by Molmil](/molmil-images/mine/9fdj) | Crystal structure of the NuoEF variant R66G (NuoF) from Aquifex aeolicus bound to NADH under anoxic conditions (short soak) | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.7 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FDV
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![BU of 9fdv by Molmil](/molmil-images/mine/9fdv) | Crystal Structure of reduced NuoEF variant R66G(NuoF) from Aquifex aeolicus | 分子名称: | 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3[N-MORPHOLINO]PROPANE SULFONIC ACID, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.986 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FE0
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![BU of 9fe0 by Molmil](/molmil-images/mine/9fe0) | Crystal Structure of reduced NuoEF variant R66G(NuoF) from Aquifex aeolicus bound to NAD+ | 分子名称: | 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-17 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FIH
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![BU of 9fih by Molmil](/molmil-images/mine/9fih) | Crystal Structure of NuoEF variant P228R(NuoF) from Aquifex aeolicus bound to NADH under anoxic conditions after 10 min soaking | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-29 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.08 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FIF
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![BU of 9fif by Molmil](/molmil-images/mine/9fif) | Crystal Structure of NuoEF variant P228R(NuoF) from Aquifex aeolicus bound to NADH under anoxic conditions | 分子名称: | 1,4-DIHYDRONICOTINAMIDE ADENINE DINUCLEOTIDE, 3[N-MORPHOLINO]PROPANE SULFONIC ACID, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-29 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (1.77 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FIJ
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![BU of 9fij by Molmil](/molmil-images/mine/9fij) | Crystal Structure of reduced NuoEF variant E222K(NuoF) from Aquifex aeolicus | 分子名称: | 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-29 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.35 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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9FIL
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![BU of 9fil by Molmil](/molmil-images/mine/9fil) | Crystal Structure of reduced NuoEF variant E222K(NuoF) from Aquifex aeolicus bound to NAD+ | 分子名称: | 1-DEOXY-1-(7,8-DIMETHYL-2,4-DIOXO-3,4-DIHYDRO-2H-BENZO[G]PTERIDIN-1-ID-10(5H)-YL)-5-O-PHOSPHONATO-D-RIBITOL, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ... | 著者 | Wohlwend, D, Friedrich, T, Goeppert-Asadollahpour, S. | 登録日 | 2024-05-29 | 公開日 | 2024-07-17 | 実験手法 | X-RAY DIFFRACTION (2.54 Å) | 主引用文献 | Structural robustness of the NADH binding site in NADH:ubiquinone oxidoreductase (complex I). Biochim Biophys Acta Bioenerg, 1865, 2024
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