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5LAT
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BU of 5lat by Molmil
HIF prolyl hydroxylase 2 (PHD2/EGLN1) P317R variant in complex with Mn(II) and N-[(1-chloro-4-hydroxyisoquinolin-3-yl)carbonyl]glycine (IOX3/UN9)
分子名称: BICARBONATE ION, Egl nine homolog 1, GLYCEROL, ...
著者Chowdhury, R, Schofield, C.J.
登録日2016-06-15
公開日2016-08-31
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural basis for oxygen degradation domain selectivity of the HIF prolyl hydroxylases.
Nat Commun, 7, 2016
3ISE
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BU of 3ise by Molmil
Structure of mineralized Bfrb (double soak) from Pseudomonas aeruginosa to 2.8A Resolution
分子名称: Bacterioferritin, FE (III) ION, POTASSIUM ION, ...
著者Lovell, S, Weeratunga, S.K, Battaile, K.P, Rivera, M.
登録日2009-08-25
公開日2010-02-02
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Structural Studies of Bacterioferritin B from Pseudomonas aeruginosa Suggest a Gating Mechanism for Iron Uptake via the Ferroxidase Center
Biochemistry, 49, 2010
7TAK
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BU of 7tak by Molmil
Structure of a NAT transporter
分子名称: GUANINE, Putative membrane protein PurT
著者Weng, J, Zhou, X, Ren, Z, Chen, K, Zhou, M.
登録日2021-12-21
公開日2023-01-25
最終更新日2024-08-07
実験手法X-RAY DIFFRACTION (2.79828 Å)
主引用文献Insight into the mechanism of H + -coupled nucleobase transport.
Proc.Natl.Acad.Sci.USA, 120, 2023
8PO5
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BU of 8po5 by Molmil
Lactobacillus plantarum LpdD
分子名称: MANGANESE (II) ION, Protein LpdD
著者Gahloth, D, Leys, D.
登録日2023-07-03
公開日2024-01-17
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献Gallate decarboxylase subunit D, LpdD
To Be Published
7QHM
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BU of 7qhm by Molmil
Cytochrome bcc-aa3 supercomplex (respiratory supercomplex III2/IV2) from Corynebacterium glutamicum (stigmatellin and azide bound)
分子名称: (2R)-2-(hexadecanoyloxy)-3-{[(S)-hydroxy{[(1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9S)-9-methyloctadecanoate, 1,2-Distearoyl-sn-glycerophosphoethanolamine, AZIDE ION, ...
著者Kao, W.-C, Hunte, C.
登録日2021-12-13
公開日2022-05-18
実験手法ELECTRON MICROSCOPY (2.8 Å)
主引用文献Structural basis for safe and efficient energy conversion in a respiratory supercomplex.
Nat Commun, 13, 2022
8PZH
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BU of 8pzh by Molmil
LpdD (H61A) mutant
分子名称: MANGANESE (II) ION, PHOSPHATE ION, Protein LpdD
著者Gahloth, D, Leys, D.
登録日2023-07-27
公開日2024-01-17
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献Structure of LpdD (H61A) mutant from Lactobacillus plantarum.
To Be Published
7QHO
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BU of 7qho by Molmil
Cytochrome bcc-aa3 supercomplex (respiratory supercomplex III2/IV2) from Corynebacterium glutamicum (as isolated)
分子名称: (2R)-2-(hexadecanoyloxy)-3-{[(S)-hydroxy{[(1R,2R,3R,4R,5R,6S)-2,3,4,5,6-pentahydroxycyclohexyl]oxy}phosphoryl]oxy}propyl (9S)-9-methyloctadecanoate, 1,2-DIACYL-GLYCEROL-3-SN-PHOSPHATE, 1,2-Distearoyl-sn-glycerophosphoethanolamine, ...
著者Kao, W.-C, Hunte, C.
登録日2021-12-13
公開日2022-05-18
実験手法ELECTRON MICROSCOPY (3.1 Å)
主引用文献Structural basis for safe and efficient energy conversion in a respiratory supercomplex
Nature Communications, 13, 2022
7TEK
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BU of 7tek by Molmil
SARS-CoV-2 3CLPro in complex with N-(4-(1H-pyrazol-4-yl)phenyl)-N-(3-chlorobenzyl)-2-(pyridin-3-yl)acetamide
分子名称: 3C-like proteinase, N-[(3-chlorophenyl)methyl]-N-[4-(1H-pyrazol-4-yl)phenyl]-2-(pyridin-3-yl)acetamide
著者Goins, C.M, Stauffer, S.R.
登録日2022-01-05
公開日2023-01-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献SARS-CoV-2 3CL-protease inhibitors derived from ML300: investigation of P1 and replacements of the 1,2,3-benzotriazole
Med.Chem.Res., 2023
2IL8
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BU of 2il8 by Molmil
THREE-DIMENSIONAL STRUCTURE OF INTERLEUKIN 8 IN SOLUTION
分子名称: INTERLEUKIN-8
著者Clore, G.M.
登録日1990-03-08
公開日1991-01-15
最終更新日2022-03-09
実験手法SOLUTION NMR
主引用文献Three-dimensional structure of interleukin 8 in solution.
Biochemistry, 29, 1990
3IOF
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BU of 3iof by Molmil
Crystal structure of CphA N220G mutant with inhibitor 10a
分子名称: Beta-lactamase, GLYCEROL, SULFATE ION, ...
著者Delbruck, H, Bebrone, C, Hoffmann, K.M.V.
登録日2009-08-14
公開日2010-06-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.44 Å)
主引用文献Mercaptophosphonate Compounds as Broad-Spectrum Inhibitors of the Metallo-beta-lactamases
J.Med.Chem., 53, 2010
3IUD
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BU of 3iud by Molmil
Cu2+-bound form of Pseudomonas stutzeri L-rhamnose isomerase
分子名称: COPPER (II) ION, L-rhamnose isomerase
著者Yoshida, H, Yamaji, M, Ishii, T, Izumori, K, Kamitori, S.
登録日2009-08-31
公開日2010-02-02
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献Catalytic reaction mechanism of Pseudomonas stutzeri l-rhamnose isomerase deduced from X-ray structures
Febs J., 277, 2010
8Q62
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BU of 8q62 by Molmil
Early closed conformation of the g-tubulin ring complex
分子名称: Gamma-tubulin complex component 2, Gamma-tubulin complex component 3, Gamma-tubulin complex component 4, ...
著者Llorca, O, Serna, M, Fernandez-Leiro, R.
登録日2023-08-10
公開日2024-02-07
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.72 Å)
主引用文献Transition of human gamma-tubulin ring complex into a closed conformation during microtubule nucleation.
Science, 383, 2024
7FEM
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BU of 7fem by Molmil
SARS-CoV-2 B.1.1.7 S-ACE2 complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Angiotensin-converting enzyme 2, ...
著者Wen, Z.L, Zhu, Y, Sun, F.
登録日2021-07-21
公開日2021-12-15
実験手法ELECTRON MICROSCOPY (4.1 Å)
主引用文献Structure-based evidence for the enhanced transmissibility of the dominant SARS-CoV-2 B.1.1.7 variant (Alpha).
Cell Discov, 7, 2021
7T23
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BU of 7t23 by Molmil
E. coli DnaB bound to two DnaG C-terminal domains, ssDNA, ADP and AlF4
分子名称: ADENOSINE-5'-DIPHOSPHATE, DNA (5'-D(*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*TP*T)-3'), DNA primase, ...
著者Oakley, A.J, Xu, Z.Q.
登録日2021-12-02
公開日2023-01-18
最終更新日2023-05-31
実験手法ELECTRON MICROSCOPY (4.2 Å)
主引用文献Sequence of conformation changes of DnaB helicase during DNA unwinding and priming in Escherichia coli
To Be Published
8PH4
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BU of 8ph4 by Molmil
Co-Crystal structure of the SARS-CoV2 main protease Nsp5 with an Uracil-carrying X77-like inhibitor
分子名称: 3C-like proteinase nsp5, DIMETHYL SULFOXIDE, MALONATE ION, ...
著者Barthel, T, Altincekic, N, Jores, N, Wollenhaupt, J, Weiss, M.S, Schwalbe, H.
登録日2023-06-18
公開日2024-01-31
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Targeting the Main Protease (M pro , nsp5) by Growth of Fragment Scaffolds Exploiting Structure-Based Methodologies.
Acs Chem.Biol., 19, 2024
7TEL
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BU of 7tel by Molmil
SARS-CoV-2 3CLPro in complex with N-(4-(1H-imidazol-4-yl)phenyl)-N-(3-chloro-5-fluorobenzyl)-2-(isoquinolin-4-yl)acetamide
分子名称: 3C-like proteinase, N-[(3-chloro-5-fluorophenyl)methyl]-N-[4-(1H-imidazol-4-yl)phenyl]-2-(isoquinolin-4-yl)acetamide
著者Goins, C.M, Stauffer, S.R.
登録日2022-01-05
公開日2023-01-11
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SARS-CoV-2 3CL-protease inhibitors derived from ML300: investigation of P1 and replacements of the 1,2,3-benzotriazole
Med.Chem.Res., 2023
5L6M
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BU of 5l6m by Molmil
Structure of Caulobacter crescentus VapBC1 (VapB1deltaC:VapC1 form)
分子名称: GLYCEROL, MALONATE ION, Ribonuclease VapC, ...
著者Bendtsen, K.L, Xu, K, Luckmann, M, Brodersen, D.E.
登録日2016-05-30
公開日2016-12-28
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Toxin inhibition in C. crescentus VapBC1 is mediated by a flexible pseudo-palindromic protein motif and modulated by DNA binding.
Nucleic Acids Res., 45, 2017
2XTM
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BU of 2xtm by Molmil
Crystal structure of GDP-bound human GIMAP2, amino acid residues 1- 234
分子名称: GLYCEROL, GTPASE IMAP FAMILY MEMBER 2, GUANOSINE-5'-DIPHOSPHATE, ...
著者Schwefel, D, Froehlich, C, Daumke, O.
登録日2010-10-11
公開日2010-10-20
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structural Basis of Oligomerization in Septin-Like Gtpase of Immunity-Associated Protein 2 (Gimap2)
Proc.Natl.Acad.Sci.USA, 107, 2010
7FHR
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BU of 7fhr by Molmil
Crystal Structure of a Rieske Oxygenase from Cupriavidus metallidurans
分子名称: 1,2-ETHANEDIOL, FE (II) ION, FE2/S2 (INORGANIC) CLUSTER, ...
著者Mahto, J.K, Dhankhar, P, Kumar, P.
登録日2021-07-30
公開日2021-12-15
最終更新日2024-05-29
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献Molecular insights into substrate recognition and catalysis by phthalate dioxygenase from Comamonas testosteroni.
J.Biol.Chem., 297, 2021
7TC7
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BU of 7tc7 by Molmil
Cryo-EM structure of methane monooxygenase hydroxylase (by quantifoil)
分子名称: FE (III) ION, Methane monooxygenase component A alpha chain, Methane monooxygenase component A beta chain, ...
著者Cho, U.S, Kim, B.C.
登録日2021-12-23
公開日2023-01-25
最終更新日2024-06-05
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Batch Production of High-Quality Graphene Grids for Cryo-EM: Cryo-EM Structure of Methylococcus capsulatus Soluble Methane Monooxygenase Hydroxylase.
Acs Nano, 17, 2023
5L6V
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BU of 5l6v by Molmil
Crystal structure of E. coli ADP-glucose pyrophosphorylase (AGPase) in complex with a negative allosteric regulator adenosine monophosphate (AMP) - AGPase*AMP
分子名称: ADENOSINE MONOPHOSPHATE, Glucose-1-phosphate adenylyltransferase, PHOSPHATE ION, ...
著者Cifuente, J.O, Albesa-Jove, D, Comino, N, Madariaga-Marcos, J, Agirre, J, Lopez-Fernandez, S, Garcia-Alija, M, Guerin, M.E.
登録日2016-05-31
公開日2016-09-07
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.667 Å)
主引用文献Structural Basis of Glycogen Biosynthesis Regulation in Bacteria.
Structure, 24, 2016
3IVY
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BU of 3ivy by Molmil
Crystal structure of Mycobacterium tuberculosis cytochrome P450 CYP125, p212121 crystal form
分子名称: Cytochrome P450 CYP125, PROTOPORPHYRIN IX CONTAINING FE
著者McLean, K.J, Levy, C, Munro, A.W, Leys, D.
登録日2009-09-02
公開日2009-11-03
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.352 Å)
主引用文献The Structure of Mycobacterium tuberculosis CYP125: molecular basis for cholesterol binding in a P450 needed for host infection.
J.Biol.Chem., 284, 2009
2XRP
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BU of 2xrp by Molmil
Human Doublecortin N-DC Repeat (1MJD) and Mammalian Tubulin (1JFF and 3HKE) Docked into the 8-Angstrom Cryo-EM Map of Doublecortin- Stabilised Microtubules
分子名称: GUANOSINE-5'-DIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, NEURONAL MIGRATION PROTEIN DOUBLECORTIN, ...
著者Fourniol, F.J, Sindelar, C.V, Amigues, B, Clare, D.K, Thomas, G, Perderiset, M, Francis, F, Houdusse, A, Moores, C.A.
登録日2010-09-18
公開日2010-11-24
最終更新日2024-05-08
実験手法ELECTRON MICROSCOPY (8.2 Å)
主引用文献Template-Free 13-Protofilament Microtubule-Map Assembly Visualized at 8 A Resolution.
J.Cell Biol., 191, 2010
7AKT
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BU of 7akt by Molmil
CrPetF variant - A39G_A41V
分子名称: BENZAMIDINE, CHLORIDE ION, FE2/S2 (INORGANIC) CLUSTER, ...
著者Kurisu, G, Ohnishi, Y, Engelbrecht, V, Happe, T.
登録日2020-10-02
公開日2021-10-13
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.11 Å)
主引用文献Ferredoxin 2.0: an electron transfer protein designed into a photosystem I-driven hydrogenase
To Be Published
2XSN
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BU of 2xsn by Molmil
Crystal Structure of Human Tyrosine Hydroxylase Catalytic Domain
分子名称: TYROSINE 3-MONOOXYGENASE, ZINC ION
著者Muniz, J.R.C, Cooper, C.D.O, Yue, W.W, Krysztofinska, E, von Delft, F, Knapp, S, Gileadi, O, Arrowsmith, C.H, Edwards, A.M, Weigelt, J, Bountra, C, Kavanagh, K.L, Oppermann, U.
登録日2010-10-29
公開日2010-11-17
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.68 Å)
主引用文献Crystal Structure of Human Tyrosine Hydroxylase Catalytic Domain
To be Published

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件を2024-08-21に公開中

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