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PDB: 5 件

2C77
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BU of 2c77 by Molmil
EF-Tu complexed with a GTP analog and the antibiotic GE2270 A
分子名称: DI(HYDROXYETHYL)ETHER, ELONGATION FACTOR TU-B, MAGNESIUM ION, ...
著者Parmeggiani, A, Krab, I.M, Okamura, S, Nielsen, R.C, Nyborg, J, Nissen, P.
登録日2005-11-18
公開日2006-03-16
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Structural basis of the action of pulvomycin and GE2270 A on elongation factor Tu.
Biochemistry, 45, 2006
3U6B
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Ef-tu (escherichia coli) in complex with nvp-ldi028
分子名称: Elongation factor Tu 1, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Palestrant, D.J.
登録日2011-10-12
公開日2012-02-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.12 Å)
主引用文献Antibacterial optimization of 4-aminothiazolyl analogues of the natural product GE2270 A: identification of the cycloalkylcarboxylic acids.
J.Med.Chem., 54, 2011
1D8T
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CRYSTAL STRUCTURE OF ELONGATION FACTOR, TU (EF-TU-MGGDP) COMPLEXED WITH GE2270A, A THIAZOLYL PEPTIDE ANTIBIOTIC
分子名称: ACETATE ION, ELONGATION FACTOR TU, GUANOSINE-5'-DIPHOSPHATE, ...
著者Heffron, S.E, Jurnak, F.
登録日1999-10-25
公開日2000-10-25
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structure of an EF-TU Complex with a Thiazolyl Peptide Antibiotic Determined at 2.35 A Resolution: Atomic Basis for Ge2270A Inhibition of EF-TU.
Biochemistry, 39, 2000
3U6K
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Ef-tu (escherichia coli) in complex with nvp-ldk733
分子名称: Elongation factor Tu 1, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Palestrant, D.J.
登録日2011-10-12
公開日2012-02-08
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献Antibacterial optimization of 4-aminothiazolyl analogues of the natural product GE2270 A: identification of the cycloalkylcarboxylic acids.
J.Med.Chem., 54, 2011
3U2Q
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BU of 3u2q by Molmil
EF-Tu (Escherichia coli) in complex with NVP-LFF571
分子名称: Elongation factor Tu 1, GUANOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ...
著者Palestrant, D.J.
登録日2011-10-04
公開日2012-05-02
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Discovery of LFF571: an investigational agent for Clostridium difficile infection.
J.Med.Chem., 55, 2012

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件を2024-10-09に公開中

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