6ZCC
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![BU of 6zcc by Molmil](/molmil-images/mine/6zcc) | X-ray structure of the Haloalkane dehalogenase HOB (HaloTag7-based Oligonucleotide Binder) labeled with a chloroalkane-tetramethylrhodamine fluorophore substrate | 分子名称: | ACETATE ION, CALCIUM ION, Haloalkane dehalogenase, ... | 著者 | Tarnawski, M, Johnsson, K, Hiblot, J. | 登録日 | 2020-06-10 | 公開日 | 2021-04-21 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (1.52 Å) | 主引用文献 | Kinetic and Structural Characterization of the Self-Labeling Protein Tags HaloTag7, SNAP-tag, and CLIP-tag. Biochemistry, 60, 2021
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7A43
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![BU of 7a43 by Molmil](/molmil-images/mine/7a43) | |
7A42
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![BU of 7a42 by Molmil](/molmil-images/mine/7a42) | |
5HZ2
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![BU of 5hz2 by Molmil](/molmil-images/mine/5hz2) | Crystal structure of PhaC1 from Ralstonia eutropha | 分子名称: | GLYCEROL, Poly-beta-hydroxybutyrate polymerase, SULFATE ION | 著者 | Kim, J, Kim, K.-J. | 登録日 | 2016-02-02 | 公開日 | 2016-12-07 | 最終更新日 | 2017-04-05 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Crystal structure of Ralstonia eutropha polyhydroxyalkanoate synthase C-terminal domain and reaction mechanisms. Biotechnol J, 12, 2017
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7AC0
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6ZVY
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![BU of 6zvy by Molmil](/molmil-images/mine/6zvy) | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-Q165H-P174R LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE | 分子名称: | CHLORIDE ION, GLYCEROL, Haloalkane dehalogenase, ... | 著者 | Tarnawski, M, Frei, M, Hiblot, J, Johnsson, K. | 登録日 | 2020-07-27 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | Engineered HaloTag variants for fluorescence lifetime multiplexing. Nat.Methods, 19, 2022
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7A7G
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![BU of 7a7g by Molmil](/molmil-images/mine/7a7g) | Soluble epoxide hydrolase in complex with TK90 | 分子名称: | (2~{R})-2-[[4-[[4-methoxy-2-(trifluoromethyl)phenyl]methylcarbamoyl]phenyl]methyl]butanoic acid, Bifunctional epoxide hydrolase 2 | 著者 | Ni, X, Kramer, J.S, Kirchner, T, Proschak, E, Chaikuad, A, Knapp, S, Structural Genomics Consortium (SGC) | 登録日 | 2020-08-28 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Combined Cardioprotective and Adipocyte Browning Effects Promoted by the Eutomer of Dual sEH/PPAR gamma Modulator. J.Med.Chem., 64, 2021
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6ZVV
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![BU of 6zvv by Molmil](/molmil-images/mine/6zvv) | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-P174W LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE | 分子名称: | CALCIUM ION, CHLORIDE ION, GLYCEROL, ... | 著者 | Tarnawski, M, Frei, M, Hiblot, J, Johnsson, K. | 登録日 | 2020-07-27 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-P174W LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE To Be Published
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6ZVW
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![BU of 6zvw by Molmil](/molmil-images/mine/6zvw) | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-Q165H LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE | 分子名称: | CHLORIDE ION, DI(HYDROXYETHYL)ETHER, GLYCEROL, ... | 著者 | Tarnawski, M, Frei, M, Hiblot, J, Johnsson, K. | 登録日 | 2020-07-27 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.6 Å) | 主引用文献 | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-Q165H LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE To Be Published
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6ZVU
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![BU of 6zvu by Molmil](/molmil-images/mine/6zvu) | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-P174L LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE | 分子名称: | CHLORIDE ION, GLYCEROL, Haloalkane dehalogenase, ... | 著者 | Tarnawski, M, Frei, M, Hiblot, J, Johnsson, K. | 登録日 | 2020-07-27 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-P174L LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE To Be Published
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6ZVX
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![BU of 6zvx by Molmil](/molmil-images/mine/6zvx) | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-Q165H-P174L LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE | 分子名称: | CHLORIDE ION, GLYCEROL, Haloalkane dehalogenase, ... | 著者 | Tarnawski, M, Frei, M, Hiblot, J, Johnsson, K. | 登録日 | 2020-07-27 | 公開日 | 2021-08-04 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.4 Å) | 主引用文献 | X-RAY STRUCTURE OF THE HALOALKANE DEHALOGENASE HALOTAG7-Q165H-P174L LABELED WITH A CHLOROALKANE-TETRAMETHYLRHODAMINE FLUOROPHORE SUBSTRATE To Be Published
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7AL5
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![BU of 7al5 by Molmil](/molmil-images/mine/7al5) | |
7AL6
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![BU of 7al6 by Molmil](/molmil-images/mine/7al6) | |
5IE6
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![BU of 5ie6 by Molmil](/molmil-images/mine/5ie6) | Crystal structure of a lactonase mutant in complex with substrate b | 分子名称: | (3S,7S,11E)-7,14,16-trihydroxy-3-methyl-3,4,5,6,7,8,9,10-octahydro-1H-2-benzoxacyclotetradecin-1-one, Zearalenone hydrolase | 著者 | Zheng, Y.Y, Xu, Z.X, Liu, W.D, Chen, C.C, Guo, R.T. | 登録日 | 2016-02-25 | 公開日 | 2017-01-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.67 Å) | 主引用文献 | Enhanced alph-Zearalenol Hydrolyzing Activity of a Mycoestrogen-Detoxifying Lactonase by Structure-Based Engineering Acs Catalysis, 6, 2016
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5IE5
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![BU of 5ie5 by Molmil](/molmil-images/mine/5ie5) | Crystal structure of a lactonase double mutant in complex with substrate a | 分子名称: | (3S,7R,11E)-7,14,16-trihydroxy-3-methyl-3,4,5,6,7,8,9,10-octahydro-1H-2-benzoxacyclotetradecin-1-one, Zearalenone hydrolase | 著者 | Zheng, Y.Y, Xu, Z.X, Liu, W.D, Chen, C.C, Guo, R.T. | 登録日 | 2016-02-25 | 公開日 | 2017-01-04 | 最終更新日 | 2024-04-03 | 実験手法 | X-RAY DIFFRACTION (2.39 Å) | 主引用文献 | Enhanced alph-Zearalenol Hydrolyzing Activity of a Mycoestrogen-Detoxifying Lactonase by Structure-Based Engineering Acs Catalysis, 6, 2016
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5IE4
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![BU of 5ie4 by Molmil](/molmil-images/mine/5ie4) | Crystal structure of a lactonase mutant in complex with substrate a | 分子名称: | (3S,7R,11E)-7,14,16-trihydroxy-3-methyl-3,4,5,6,7,8,9,10-octahydro-1H-2-benzoxacyclotetradecin-1-one, Zearalenone hydrolase | 著者 | Zheng, Y.Y, Xu, Z.X, Liu, W.D, Chen, C.C, Guo, R.T. | 登録日 | 2016-02-25 | 公開日 | 2017-01-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Enhanced alph-Zearalenol Hydrolyzing Activity of a Mycoestrogen-Detoxifying Lactonase by Structure-Based Engineering Acs Catalysis, 6, 2016
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5IE7
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![BU of 5ie7 by Molmil](/molmil-images/mine/5ie7) | Crystal structure of a lactonase double mutant in complex with substrate b | 分子名称: | (3S,7S,11E)-7,14,16-trihydroxy-3-methyl-3,4,5,6,7,8,9,10-octahydro-1H-2-benzoxacyclotetradecin-1-one, Zearalenone hydrolase | 著者 | Zheng, Y.Y, Xu, Z.X, Liu, W.D, Chen, C.C, Guo, R.T. | 登録日 | 2016-02-25 | 公開日 | 2017-01-04 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Enhanced alph-Zearalenol Hydrolyzing Activity of a Mycoestrogen-Detoxifying Lactonase by Structure-Based Engineering Acs Catalysis, 6, 2016
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5K3E
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![BU of 5k3e by Molmil](/molmil-images/mine/5k3e) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Asp110Asn/Glycolate - Cocrystallized | 分子名称: | CHLORIDE ION, Fluoroacetate dehalogenase, GLYCOLIC ACID | 著者 | Mehrabi, P, Kim, T.H, Prosser, S.R, Pai, E.F. | 登録日 | 2016-05-19 | 公開日 | 2017-02-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.54 Å) | 主引用文献 | The role of dimer asymmetry and protomer dynamics in enzyme catalysis. Science, 355, 2017
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5K3A
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![BU of 5k3a by Molmil](/molmil-images/mine/5k3a) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - His280Asn/Fluoroacetate - Cocrystallized - Both Protomers Reacted with Ligand | 分子名称: | CHLORIDE ION, Fluoroacetate dehalogenase | 著者 | Mehrabi, P, Kim, T.H, Prosser, S.R, Pai, E.F. | 登録日 | 2016-05-19 | 公開日 | 2017-02-01 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.511 Å) | 主引用文献 | The role of dimer asymmetry and protomer dynamics in enzyme catalysis. Science, 355, 2017
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5JZS
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![BU of 5jzs by Molmil](/molmil-images/mine/5jzs) | HsaD bound to 3,5-dichloro-4-hydroxybenzoic acid | 分子名称: | 2-hydroxy-6-oxo-6-phenylhexa-2,4-dienoate hydrolase BphD, 3,5-dichloro-4-hydroxybenzoic acid | 著者 | Ryan, A, Polycarpou, E, Lack, N, Evangelopoulos, D, Sieg, C, Halman, A, Bhakta, S, Sinclair, A, Eleftheriadou, O, McHugh, T.D, Keany, S, Lowe, E.D, Ballet, R, Abuhammad, A, Ciulli, A, Sim, E. | 登録日 | 2016-05-17 | 公開日 | 2017-04-05 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.27 Å) | 主引用文献 | Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. Br. J. Pharmacol., 174, 2017
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5K3B
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![BU of 5k3b by Molmil](/molmil-images/mine/5k3b) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - Asp110Asn/Chloroacetate - Cocrystallized | 分子名称: | CHLORIDE ION, Fluoroacetate dehalogenase, chloroacetic acid | 著者 | Mehrabi, P, Kim, T.H, Prosser, S.R, Pai, E.F. | 登録日 | 2016-05-19 | 公開日 | 2017-02-01 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.58 Å) | 主引用文献 | The role of dimer asymmetry and protomer dynamics in enzyme catalysis. Science, 355, 2017
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5JZB
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![BU of 5jzb by Molmil](/molmil-images/mine/5jzb) | Crystal structure of HsaD bound to 3,5-dichlorobenzene sulphonamide | 分子名称: | 3,5-dichlorobenzene-1-sulfonamide, 4,5:9,10-diseco-3-hydroxy-5,9,17-trioxoandrosta-1(10),2-diene-4-oate hydrolase, PHOSPHATE ION | 著者 | Ryan, A, Polycarpou, E, Lack, N.A, Evangelopoulos, D, Sieg, C, Halman, A, Bhakta, S, Sinclair, A, Eleftheriadou, O, McHugh, T.D, Keany, S, Lowe, E, Ballet, R, Abihammad, A, Ciulli, A, Sim, E. | 登録日 | 2016-05-16 | 公開日 | 2017-04-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.102 Å) | 主引用文献 | Investigation of the mycobacterial enzyme HsaD as a potential novel target for anti-tubercular agents using a fragment-based drug design approach. Br. J. Pharmacol., 174, 2017
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5K3C
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![BU of 5k3c by Molmil](/molmil-images/mine/5k3c) | Crystal Structure of the Fluoroacetate Dehalogenase RPA1163 - WT/5-Fluorotryptophan | 分子名称: | CHLORIDE ION, Fluoroacetate dehalogenase | 著者 | Mehrabi, P, Kim, T.H, Prosser, S.R, Pai, E.F. | 登録日 | 2016-05-19 | 公開日 | 2017-02-01 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.541 Å) | 主引用文献 | The role of dimer asymmetry and protomer dynamics in enzyme catalysis. Science, 355, 2017
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5K3D
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![BU of 5k3d by Molmil](/molmil-images/mine/5k3d) | |
8OOH
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![BU of 8ooh by Molmil](/molmil-images/mine/8ooh) | |