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PDB: 145 件

8QVO
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L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris
分子名称: CALCIUM ION, Carboxypeptidase T, SULFATE ION, ...
著者Timofeev, V.I, Dorovatovskii, P.V, Lazarenko, V.A, Akparov, V.K, Kuranova, I.P.
登録日2023-10-18
公開日2024-01-17
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献L211Q, L254N, T262G mutant of carboxypeptidase T from Thermoactinomyces vulgaris
To Be Published
8CPA
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COMPARISON OF THE STRUCTURES OF THREE CARBOXYPEPTIDASE A-PHOSPHONATE COMPLEXES DETERMINED BY X-RAY CRYSTALLOGRAPHY
分子名称: CARBOXYPEPTIDASE A, O-(((1R)-((N-(PHENYL-METHOXY-CARBONYL)-ALANYL)-AMINO)METHYL)HYDROXYPHOSPHINYL)3-L-PHENYLLACTATE, ZINC ION
著者Kim, H, Lipscomb, W.N.
登録日1991-05-21
公開日1994-01-31
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Comparison of the structures of three carboxypeptidase A-phosphonate complexes determined by X-ray crystallography.
Biochemistry, 30, 1991
2RFH
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BU of 2rfh by Molmil
Crystal Structure Analysis of CPA-2-benzyl-3-nitropropanoic acid complex
分子名称: (2R)-2-benzyl-3-nitropropanoic acid, Carboxypeptidase A1, ZINC ION
著者Wang, S.-F, Zeng, Z.-H.
登録日2007-09-29
公開日2008-04-22
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Nitro as a novel zinc-binding group in the inhibition of carboxypeptidase A
Bioorg.Med.Chem., 16, 2008
4GM5
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BU of 4gm5 by Molmil
Carboxypeptidase T with Sulphamoil Arginine
分子名称: CALCIUM ION, Carboxypeptidase T, GLYCEROL, ...
著者Kuznetsov, S.A, Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2012-08-15
公開日2013-08-21
実験手法X-RAY DIFFRACTION (1.39 Å)
主引用文献Carboxypeptidase T with Sulphamoil Arginine
To be Published
7Q87
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Carboxypeptidase T with (S)-3-phenyllactic acid
分子名称: ALPHA-HYDROXY-BETA-PHENYL-PROPIONIC ACID, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Shevtsov, M.B, Kuranova, I.P.
登録日2021-11-10
公開日2022-01-26
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.73 Å)
主引用文献Carboxypeptidase T with (S)-3-phenyllactic acid
To Be Published
6Z28
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Carboxypeptidase T mutant L254N with N-sulfamoyl-L-glutamic acid
分子名称: CALCIUM ION, Carboxypeptidase T, N-sulfamoyl-L-glutamic acid, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-05-15
公開日2020-05-27
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献CARBOXYPEPTIDASE T MUTANT L254N WITH WITH N-SULFAMOYL-L-GLUT
To Be Published
5CPA
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REFINED CRYSTAL STRUCTURE OF CARBOXYPEPTIDASE A AT 1.54 ANGSTROMS RESOLUTION.
分子名称: CARBOXYPEPTIDASE A, ZINC ION
著者Lipscomb, W.N.
登録日1982-05-06
公開日1982-07-29
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (1.54 Å)
主引用文献Refined crystal structure of carboxypeptidase A at 1.54 A resolution.
J.Mol.Biol., 168, 1983
2V77
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Crystal Structure of Human Carboxypeptidase A1
分子名称: 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CARBOXYPEPTIDASE A1, OCTANE-1,3,5,7-TETRACARBOXYLIC ACID, ...
著者Pallares, I, Fernandez, D, Comellas-Bigler, M, Fernandez-Recio, J, Ventura, S, Aviles, F.X, Vendrell, J.
登録日2007-07-27
公開日2008-07-01
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.603 Å)
主引用文献Direct interaction between a human digestive protease and the mucoadhesive poly(acrylic acid).
Acta Crystallogr. D Biol. Crystallogr., D64, 2008
5ZEQ
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Carboxypeptidase B in complex with DD28
分子名称: (2~{S})-2-[(6-azanyl-5-chloranyl-pyridin-3-yl)methyl]-3-selanyl-propanoic acid, CACODYLATE ION, Carboxypeptidase B, ...
著者Itoh, T, Yoshimoto, N, Yamamoto, K.
登録日2018-02-27
公開日2018-06-20
最終更新日2018-07-04
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Structural basis for the selective inhibition of activated thrombin-activatable fibrinolysis inhibitor (TAFIa) by a selenium-containing inhibitor with chloro-aminopyridine as a basic group
Bioorg. Med. Chem. Lett., 28, 2018
6CPA
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CRYSTAL STRUCTURE OF THE COMPLEX OF CARBOXYPEPTIDASE A WITH A STRONGLY BOUND PHOSPHONATE IN A NEW CRYSTALLINE FORM: COMPARISON WITH STRUCTURES OF OTHER COMPLEXES
分子名称: CARBOXYPEPTIDASE A, O-(((1R)-((N-PHENYLMETHOXYCARBONYL-L-ALANYL)AMINO)ETHYL)HYDROXYPHOSPHONO)-L-BENZYLACETIC ACID, ZINC ION
著者Kim, H, Lipscomb, W.N.
登録日1990-02-15
公開日1991-10-15
最終更新日2024-06-05
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Crystal structure of the complex of carboxypeptidase A with a strongly bound phosphonate in a new crystalline form: comparison with structures of other complexes.
Biochemistry, 29, 1990
4Z65
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Carboxypeptidase B with Sulphamoil Arginine
分子名称: Carboxypeptidase B, N~2~-sulfamoyl-L-arginine, ZINC ION
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2015-04-03
公開日2015-10-14
最終更新日2015-10-28
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Structure of the complex of carboxypeptidase B and N-sulfamoyl-L-arginine.
Acta Crystallogr.,Sect.F, 71, 2015
6I6Z
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Crystal structure of the human CARBOXYPEPTIDASE A1 in complex with the PHOSPHINIC INHIBITOR Acetyl-Tyr-Ala-Y(PO2CH2)-homoPhe-OH
分子名称: (2S)-2-{[(S)-{(1R)-1-[(N-acetyl-L-tyrosyl)amino]ethyl}(hydroxy)phosphoryl]methyl}-4-phenylbutanoic acid, Carboxypeptidase A1, ZINC ION
著者Gallego, P, Reverter, D.
登録日2018-11-15
公開日2018-12-12
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.72 Å)
主引用文献Synthesis and Structural/Functional Characterization of Selective M14 Metallocarboxypeptidase Inhibitors Based on Phosphinic Pseudopeptide Scaffold: Implications on the Design of Specific Optical Probes.
J. Med. Chem., 62, 2019
2JEW
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BU of 2jew by Molmil
Crystal structure of ((2S)-5-amino-2-((1-n-propyl-1H-imidazol-4-yl) methyl)pentanoic acid) UK396,082 a TAFIa inhibitor, Bound to Activated Porcine Pancreatic carboxypeptidaseB
分子名称: (2S)-5-AMINO-2-[(1-PROPYL-1H-IMIDAZOL-4-YL)METHYL]PENTANOIC ACID, CARBOXYPEPTIDASE B, ZINC ION
著者Brown, D.G, Moore, R.S.
登録日2007-01-24
公開日2007-11-20
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Discovery of potent & selective inhibitors of activated thrombin-activatable fibrinolysis inhibitor for the treatment of thrombosis.
J. Med. Chem., 50, 2007
3QNV
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Carboxypeptidase T
分子名称: Carboxypeptidase T, GLYCEROL, SULFATE ION, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2011-02-09
公開日2012-02-15
実験手法X-RAY DIFFRACTION (1.69 Å)
主引用文献Three-dimensional structure of recombinant carboxypeptidase T from Thermoactinomyces vulgaris without calcium ions
Crystallography Reports, 56, 2011
5JC6
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Carboxypeptidase B with 2-nd zinc and acetate ion
分子名称: ACETATE ION, Carboxypeptidase B, ZINC ION
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2016-04-14
公開日2017-05-24
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Structure of the carboxypeptidase B complex with N-sulfamoyl-L-phenylalanine - a transition state analog of non-specific substrate.
J. Biomol. Struct. Dyn., 36, 2018
5J1Q
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Carboxypeptidase B with Sulphamoil Phenylalanine
分子名称: Carboxypeptidase B, PHENYLALANINE-N-SULFONAMIDE, ZINC ION
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2016-03-29
公開日2017-04-19
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.74 Å)
主引用文献Carboxypeptidase B with Sulphamoil Phenylalanine
To Be Published
4OKO
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BU of 4oko by Molmil
Crystal structure of Francisella tularensis REP34 (Rapid Encystment Phenotype Protein 34 KDa)
分子名称: ACETATE ION, Rapid Encystment Phenotype Protein 34 KDa, ZINC ION
著者Feld, G.K, Segelke, B.W, Corzett, M.H, Hunter, M.S, Frank, M, Rasley, A.
登録日2014-01-22
公開日2014-09-24
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.053 Å)
主引用文献Structure and Function of REP34 Implicates Carboxypeptidase Activity in Francisella tularensis Host Cell Invasion.
J.Biol.Chem., 289, 2014
3CPA
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X-RAY CRYSTALLOGRAPHIC INVESTIGATION OF SUBSTRATE BINDING TO CARBOXYPEPTIDASE A AT SUBZERO TEMPERATURE
分子名称: CARBOXYPEPTIDASE A, GLYCINE, TYROSINE, ...
著者Lipscomb, W.N.
登録日1982-03-24
公開日1982-07-29
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献X-ray crystallographic investigation of substrate binding to carboxypeptidase A at subzero temperature.
Proc.Natl.Acad.Sci.USA, 83, 1986
3V38
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Carboxypeptidase T mutant L254N
分子名称: Carboxypeptidase T, GLYCEROL, SULFATE ION, ...
著者Timofeev, V.I, Kuznetsov, S.A, Akparov, V.K, Kuranova, I.P.
登録日2011-12-13
公開日2012-12-19
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献Carboxypeptidase T mutant L254N
TO BE PUBLISHED
5HXD
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Crystal structure of murein-tripeptide amidase MpaA from Escherichia coli O157
分子名称: CACODYLATE ION, Protein MpaA, ZINC ION
著者Ma, Y, Bai, G, Zhang, X, Zhao, J, Yuan, Z, Kang, X, Li, Z, Mu, S, Liu, X.
登録日2016-01-30
公開日2017-02-08
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal Structure of Murein-Tripeptide Amidase MpaA from Escherichia coli O157 at 2.6 angstrom Resolution
Protein Pept.Lett., 24, 2017
6SN6
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CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-GLUTAMIC ACID
分子名称: CALCIUM ION, Carboxypeptidase T, N-sulfamoyl-L-glutamic acid, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-08-23
公開日2019-10-09
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-GLUTAMIC ACID
To Be Published
6T9Y
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BU of 6t9y by Molmil
CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-LYSIN
分子名称: (2~{S})-6-azanyl-2-(sulfamoylamino)hexanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-10-29
公開日2019-12-11
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.92 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-LYSIN
To Be Published
6TNK
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CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-VALINE
分子名称: (2~{S})-3-methyl-2-(sulfamoylamino)butanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2019-12-09
公開日2019-12-18
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献CARBOXYPEPTIDASE T WITH N-SULFAMOYL-L-VALINE
To Be Published
7ARU
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BU of 7aru by Molmil
L254N mutant of carboxypeptidase T from Thermoactinomyces vulgaris N-sulfamoyl-L-valine
分子名称: (2~{S})-3-methyl-2-(sulfamoylamino)butanoic acid, CALCIUM ION, Carboxypeptidase T, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-10-26
公開日2020-11-11
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献L254N mutant of carboxypeptidase T from Thermoactinomyces vulgaris N-sulfamoyl-L-valine
To Be Published
7AQP
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T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris
分子名称: CALCIUM ION, Carboxypeptidase T, SULFATE ION, ...
著者Timofeev, V.I, Akparov, V.K, Kuranova, I.P.
登録日2020-10-22
公開日2020-12-02
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献T262S, A251S, L254S, L211Q mutant of carboxypeptidase T from Thermoactinomyces vulgaris
To Be Published

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件を2024-07-17に公開中

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