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PDB: 5 件
4TND
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BU of 4tnd by Molmil
Crystal Structure of G Protein-Coupled Receptor Kinase 5 in Complex with AMP-PNP
分子名称: G protein-coupled receptor kinase 5, MAGNESIUM ION, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER
著者Bhardwaj, A, Komolov, K.E, Benovic, J.L.
登録日2014-06-04
公開日2015-06-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (1.802 Å)
主引用文献Atomic Structure of G Protein-Coupled Receptor Kinase 5 (GRK5) Reveals Distinct Structural Features Novel for GRKs.
J.Biol.Chem., 2015
6PJX
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BU of 6pjx by Molmil
Crystal Structure of G Protein-Coupled Receptor Kinase 5 (GRK5) in Complex with Calmodulin (CaM)
分子名称: CALCIUM ION, Calmodulin, G protein-coupled receptor kinase 5, ...
著者Bhardwaj, A, Komolov, K.E, Sulon, S, Benovic, J.L.
登録日2019-06-28
公開日2020-12-09
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.96 Å)
主引用文献Structure of a GRK5-Calmodulin Complex Reveals Molecular Mechanism of GRK Activation and Substrate Targeting.
Mol.Cell, 81, 2021
4TNB
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BU of 4tnb by Molmil
Crystal Structure of G Protein-Coupled Receptor Kinase 5 in Complex with Sangivamycin
分子名称: G protein-coupled receptor kinase 5, SANGIVAMYCIN
著者Bhardwaj, A, Komolov, K.E, Benovic, J.L.
登録日2014-06-03
公開日2015-06-10
最終更新日2023-09-27
実験手法X-RAY DIFFRACTION (2.113 Å)
主引用文献Atomic Structure of G Protein-Coupled Receptor Kinase 5 (GRK5) Reveals Distinct Structural Features Novel for GRKs.
J.Biol.Chem., 2015
8UAP
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BU of 8uap by Molmil
Crystal Structure of Human G Protein-Coupled Receptor Kinase 5 D311N in Complex with CCG273441
分子名称: (3Z)-3-{[4-(2-chloroacetamido)-3,5-dimethyl-1H-pyrrol-2-yl]methylidene}-N-[(1R)-1-(4-fluorophenyl)ethyl]-2-oxo-2,3-dihydro-1H-indole-5-carboxamide, G protein-coupled receptor kinase 5
著者Chen, Y, Tesmer, J.J.G.
登録日2023-09-21
公開日2023-12-13
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Development of a new class of potent and highly selective G protein-coupled receptor kinase 5 inhibitors and structural insight from crystal structures of inhibitor complexes.
Eur.J.Med.Chem., 264, 2023
8UAQ
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BU of 8uaq by Molmil
Crystal Structure of Human G Protein-Coupled Receptor Kinase 5 in Complex with GRL018-21
分子名称: (3Z)-N-[(1R)-1-(4-fluorophenyl)ethyl]-3-[(4-{[(2S)-2-(furan-2-yl)-2-hydroxyacetyl]amino}-3,5-dimethyl-1H-pyrrol-2-yl)methylidene]-2-oxo-2,3-dihydro-1H-indole-5-carboxamide, G protein-coupled receptor kinase 5
著者Chen, Y, Tesmer, J.J.G.
登録日2023-09-21
公開日2023-12-13
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Development of a new class of potent and highly selective G protein-coupled receptor kinase 5 inhibitors and structural insight from crystal structures of inhibitor complexes.
Eur.J.Med.Chem., 264, 2023

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件を2024-08-07に公開中

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