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4TND

Crystal Structure of G Protein-Coupled Receptor Kinase 5 in Complex with AMP-PNP

Summary for 4TND
Entry DOI10.2210/pdb4tnd/pdb
Related4TNB
DescriptorG protein-coupled receptor kinase 5, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, MAGNESIUM ION, ... (4 entities in total)
Functional Keywordsgrk5-(5-adenylylimidodiphosphate) complex, grk5-(amp-pnp) complex, gpcr kinase, kinase, gpcr kinase 5, signaling protein
Biological sourceHomo sapiens (Human)
Cellular locationCytoplasm: P34947
Total number of polymer chains1
Total formula weight68473.17
Authors
Bhardwaj, A.,Komolov, K.E.,Benovic, J.L. (deposition date: 2014-06-04, release date: 2015-06-10, Last modification date: 2023-09-27)
Primary citationKomolov, K.E.,Bhardwaj, A.,Benovic, J.L.
Atomic Structure of G Protein-Coupled Receptor Kinase 5 (GRK5) Reveals Distinct Structural Features Novel for GRKs.
J.Biol.Chem., 2015
Cited by
PubMed: 26032409
DOI: 10.1074/jbc.M115.647297
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.802 Å)
Structure validation

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