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PDB: 55 件

7FSG
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BU of 7fsg by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z56772132
分子名称: (5R)-5-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione, 1,2-ETHANEDIOL, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FTA
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BU of 7fta by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z228589380
分子名称: 1,2-ETHANEDIOL, 3-[(pyrimidin-2-yl)amino]benzoic acid, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT2
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BU of 7ft2 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z235449082
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.04 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSZ
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BU of 7fsz by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z3006151474
分子名称: (5S)-5-(difluoromethoxy)pyridin-2(5H)-one, 1,2-ETHANEDIOL, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT3
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BU of 7ft3 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z291279160
分子名称: 1,2-ETHANEDIOL, 1-[2-(trifluoromethyloxy)phenyl]thiourea, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSQ
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BU of 7fsq by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1429867185
分子名称: 1,2-ETHANEDIOL, 4-methoxy-1H-indole, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.07 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSM
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BU of 7fsm by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z763030030
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSH
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BU of 7fsh by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z32367954
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT1
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BU of 7ft1 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z2204875953
分子名称: (3P)-3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazole, 1,2-ETHANEDIOL, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSS
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BU of 7fss by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z839706072
分子名称: 1,2-ETHANEDIOL, 2-(4-bromanylpyrazol-1-yl)-~{N}-cyclopropyl-~{N}-methyl-ethanamide, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.11 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSW
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BU of 7fsw by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z169675004
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.14 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT4
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BU of 7ft4 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z48847594
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
8AAP
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BU of 8aap by Molmil
Crystal structure of the PDZ tandem of syntenin in complex with compound SYNTi
分子名称: (2S)-2-[[(2S)-2-(6-bromanyl-3-oxidanylidene-1H-isoindol-2-yl)-3-[4-(5-ethanoyl-2-fluoranyl-phenyl)phenyl]propanoyl]amino]propanoic acid, Syntenin-1
著者Feracci, M, Barral, K.
登録日2022-07-01
公開日2023-04-26
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (2.174 Å)
主引用文献Discovery of a PDZ Domain Inhibitor Targeting the Syndecan/Syntenin Protein-Protein Interaction: A Semi-Automated "Hit Identification-to-Optimization" Approach.
J.Med.Chem., 66, 2023
6RLC
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BU of 6rlc by Molmil
Crystal structure of the PDZ tandem of syntenin in complex with fragment F13
分子名称: (2~{S})-2-[3-(4-chlorophenyl)sulfanylpropanoylamino]-3-methyl-butanoic acid, ACETATE ION, Syntenin-1
著者Feracci, M, Barral, K.
登録日2019-05-02
公開日2021-02-03
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Pharmacological inhibition of syntenin PDZ2 domain impairs breast cancer cell activities and exosome loadifing with syndecan and EpCAM cargo.
J Extracell Vesicles, 10, 2020
7FTB
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BU of 7ftb by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1198269757
分子名称: 1,2-ETHANEDIOL, D-GLUTAMIC ACID, GLYCINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.22 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSV
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BU of 7fsv by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1454310449
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
1W9O
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BU of 1w9o by Molmil
Crystal structure of the PDZ tandem of human syntenin in complex with TNEYYV peptide
分子名称: BENZOIC ACID, SYNTENIN 1, TNEYYV PEPTIDE
著者Grembecka, J, Cierpicki, T, Devedjiev, Y, Cooper, D.R, Derewenda, U, Derewenda, Z.S.
登録日2004-10-15
公開日2006-03-22
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.25 Å)
主引用文献The Binding of the Pdz Tandem of Syntenin to Target Proteins.
Biochemistry, 45, 2006
7FSR
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BU of 7fsr by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z54615640
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.29 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
1YBO
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BU of 1ybo by Molmil
Crystal structure of the PDZ tandem of human syntenin with syndecan peptide
分子名称: Syndecan-4, Syntenin 1
著者Grembecka, J, Cooper, D.R, Cierpicki, T, Kang, B.S, Devedjiev, Y, Derewenda, Z.
登録日2004-12-21
公開日2006-01-10
最終更新日2023-08-23
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The binding of the PDZ tandem of syntenin to target proteins
Biochemistry, 45, 2006
7FSI
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BU of 7fsi by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z18197050
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.31 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSL
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BU of 7fsl by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z730649594
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSK
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BU of 7fsk by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z1954800564
分子名称: 1,2-ETHANEDIOL, 5-methoxy-1,3-benzothiazol-2-amine, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FSN
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BU of 7fsn by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z254580486
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT8
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BU of 7ft8 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with NCL-00024671
分子名称: 1,2-ETHANEDIOL, 2-(4-bromo-1H-pyrazol-1-yl)ethan-1-ol, ALANINE, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published
7FT0
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BU of 7ft0 by Molmil
SDCBP PanDDA analysis group deposition -- The PDZ domans of SDCBP in complex with Z56767614
分子名称: 1,2-ETHANEDIOL, ALANINE, D-GLUTAMIC ACID, ...
著者Bradshaw, W.J, Katis, V.L, Bountra, C, von Delft, F, Brennan, P.E.
登録日2023-01-24
公開日2023-02-15
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.45 Å)
主引用文献SDCBP PanDDA analysis group deposition
To Be Published

223532

件を2024-08-07に公開中

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