3ZOT
| Structure of E.coli rhomboid protease GlpG in complex with monobactam L29 (data set 2) | 分子名称: | CHLORIDE ION, RHOMBOID PROTEASE GLPG, nonyl beta-D-glucopyranoside, ... | 著者 | Vinothkumar, K.R, Pierrat, O.A, Large, J.M, Freeman, M. | 登録日 | 2013-02-24 | 公開日 | 2013-05-22 | 最終更新日 | 2023-12-20 | 実験手法 | X-RAY DIFFRACTION (2.399 Å) | 主引用文献 | Structure of Rhomboid Protease in Complex with Beta-Lactam Inhibitors Defines the S2' Cavity. Structure, 21, 2013
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5F5J
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5F5K
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6PJR
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6PJ5
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6PJ8
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6XRP
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8AB5
| Structure of E. coli GlpG in complex with peptide derived inhibitor Ac-VRHA-conh-[4-(4-butyl)-phenoxy-1-phenyl-2-butyl] | 分子名称: | Ac-VRHA-conh-[4-(4-butyl)-phenoxy-1-phenyl-2-butyl], Rhomboid protease GlpG | 著者 | Skerlova, J, Polovinkin, V, Bach, K, Borshchevskiy, V, Strisovsky, K. | 登録日 | 2022-07-04 | 公開日 | 2023-10-25 | 最終更新日 | 2024-07-10 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Extensive targeting of chemical space at the prime side of ketoamide inhibitors of rhomboid proteases by branched substituents empowers their selectivity and potency. Eur.J.Med.Chem., 275, 2024
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4NJN
| Crystal Structure of E.coli GlpG at pH 4.5 | 分子名称: | Rhomboid protease GlpG | 著者 | Dickey, S.W, Baker, R.P, Cho, S, Urban, S. | 登録日 | 2013-11-11 | 公開日 | 2013-12-25 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity. Cell(Cambridge,Mass.), 155, 2013
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4NJP
| Proteolysis inside the membrane is a rate-governed reaction not Driven by substrate affinity | 分子名称: | Rhomboid protease GlpG | 著者 | Dickey, S.W, Baker, R.P, Cho, S, Urban, S. | 登録日 | 2013-11-11 | 公開日 | 2013-12-25 | 最終更新日 | 2023-09-20 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Proteolysis inside the Membrane Is a Rate-Governed Reaction Not Driven by Substrate Affinity. Cell(Cambridge,Mass.), 155, 2013
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6PJP
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5F5D
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6PJU
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6PJ9
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2O7L
| The open-cap conformation of GlpG | 分子名称: | Protein glpG, nonyl beta-D-glucopyranoside | 著者 | Ha, Y. | 登録日 | 2006-12-11 | 公開日 | 2006-12-26 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Open-cap conformation of intramembrane protease GlpG. Proc.Natl.Acad.Sci.Usa, 104, 2007
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6PJQ
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6PJA
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2NRF
| Crystal Structure of GlpG, a Rhomboid family intramembrane protease | 分子名称: | Protein GlpG | 著者 | Wu, Z, Yan, N, Feng, L, Yan, H, Gu, L, Shi, Y. | 登録日 | 2006-11-02 | 公開日 | 2006-11-14 | 最終更新日 | 2023-08-30 | 実験手法 | X-RAY DIFFRACTION (2.6 Å) | 主引用文献 | Structural analysis of a rhomboid family intramembrane protease reveals a gating mechanism for substrate entry. Nat.Struct.Mol.Biol., 13, 2006
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3UBB
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4H1D
| Cocrystal structure of GlpG and DFP | 分子名称: | DIISOPROPYL PHOSPHONATE, Rhomboid protease GlpG | 著者 | Xue, Y, Ha, Y. | 登録日 | 2012-09-10 | 公開日 | 2013-05-01 | 最終更新日 | 2013-06-26 | 実験手法 | X-RAY DIFFRACTION (2.8975 Å) | 主引用文献 | Large lateral movement of transmembrane helix s5 is not required for substrate access to the active site of rhomboid intramembrane protease. J.Biol.Chem., 288, 2013
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2LEP
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