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PDB: 4 件

4XI2
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BU of 4xi2 by Molmil
Crystal Structure of an auto-inhibited form of Bruton's Tryrosine Kinase
分子名称: GOLD ION, Tyrosine-protein kinase BTK
著者Vogan, E.M, Harrison, S.C.
登録日2015-01-06
公開日2015-02-25
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Autoinhibition of Bruton's tyrosine kinase (Btk) and activation by soluble inositol hexakisphosphate.
Elife, 4, 2015
4Y95
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BU of 4y95 by Molmil
Crystal structure of the kinase domain of Bruton's tyrosine kinase with mutations in the activation loop
分子名称: 2-{2-[2-(2-{2-[2-(2-ETHOXY-ETHOXY)-ETHOXY]-ETHOXY}-ETHOXY)-ETHOXY]-ETHOXY}-ETHANOL, 4-tert-butyl-N-[2-methyl-3-(4-methyl-6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-5-oxo-4,5-dihydropyrazin-2-yl)phenyl]benzamide, BETA-MERCAPTOETHANOL, ...
著者Wang, Q, Rosen, C.E, Kuriyan, J.
登録日2015-02-16
公開日2015-03-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.599 Å)
主引用文献Autoinhibition of Bruton's tyrosine kinase (Btk) and activation by soluble inositol hexakisphosphate.
Elife, 4, 2015
4Y94
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BU of 4y94 by Molmil
Crystal structure of the PH-TH module of Bruton's tyrosine kinase bound to inositol hexakisphosphate
分子名称: INOSITOL HEXAKISPHOSPHATE, Non-specific protein-tyrosine kinase, ZINC ION
著者Wang, Q, Kuriyan, J.
登録日2015-02-16
公開日2015-03-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Autoinhibition of Bruton's tyrosine kinase (Btk) and activation by soluble inositol hexakisphosphate.
Elife, 4, 2015
4Y93
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BU of 4y93 by Molmil
Crystal structure of the PH-TH-kinase construct of Bruton's tyrosine kinase (Btk)
分子名称: 4-tert-butyl-N-[2-methyl-3-(4-methyl-6-{[4-(morpholin-4-ylcarbonyl)phenyl]amino}-5-oxo-4,5-dihydropyrazin-2-yl)phenyl]benzamide, CALCIUM ION, Non-specific protein-tyrosine kinase,Non-specific protein-tyrosine kinase, ...
著者Wang, Q, Kuriyan, J.
登録日2015-02-16
公開日2015-03-18
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.695 Å)
主引用文献Autoinhibition of Bruton's tyrosine kinase (Btk) and activation by soluble inositol hexakisphosphate.
Elife, 4, 2015

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件を2024-05-29に公開中

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