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PDB: 3 件

9BWT
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BU of 9bwt by Molmil
human sodium chloride cotransporter NCC S344E in the phosphorylation state and in complex with hydrochlorothiazide
分子名称: 6-chloro-3,4-dihydro-2H-1,2,4-benzothiadiazine-7-sulfonamide 1,1-dioxide, ADENOSINE-5'-TRIPHOSPHATE, Solute carrier family 12 member 3
著者Cao, E.H, Zhao, Y.X.
登録日2024-05-21
公開日2024-09-04
実験手法ELECTRON MICROSCOPY (2.5 Å)
主引用文献Structural bases for Na + -Cl - cotransporter inhibition by thiazide diuretic drugs and activation by kinases.
Nat Commun, 15, 2024
8VPP
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BU of 8vpp by Molmil
Phosphorylated human NCC in complex with chlorthalidone
分子名称: 2-chloro-5-[(1S)-1-hydroxy-3-oxo-2H-isoindol-1-yl]benzenesulfonamide, Solute carrier family 12 member 3
著者Zhao, Y.X, Cao, E.H.
登録日2024-01-16
公開日2024-09-04
実験手法ELECTRON MICROSCOPY (2.9 Å)
主引用文献Structural bases for Na + -Cl - cotransporter inhibition by thiazide diuretic drugs and activation by kinases.
Nat Commun, 15, 2024
8VPN
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BU of 8vpn by Molmil
Phosphorylated human NCC in complex with indapamide
分子名称: 4-chloro-N-[(2S)-2-methyl-2,3-dihydro-1H-indol-1-yl]-3-sulfamoylbenzamide, ADENOSINE-5'-TRIPHOSPHATE, Solute carrier family 12 member 3
著者Zhao, Y.X, Cao, E.H.
登録日2024-01-16
公開日2024-09-04
実験手法ELECTRON MICROSCOPY (2.7 Å)
主引用文献Structural bases for Na + -Cl - cotransporter inhibition by thiazide diuretic drugs and activation by kinases.
Nat Commun, 15, 2024

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件を2024-09-04に公開中

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