5K0M
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![BU of 5k0m by Molmil](/molmil-images/mine/5k0m) | Targeting the PRC2 complex through a novel protein-protein interaction inhibitor of EED | 分子名称: | (3R,4S)-1-[(1S)-7-fluoro-2,3-dihydro-1H-inden-1-yl]-N,N-dimethyl-4-{4-[4-(methylsulfonyl)piperazin-1-yl]phenyl}pyrrolidin-3-amine, Polycomb protein EED | 著者 | Jakob, C.G, Bigelow, L.J, Zhu, H, Sun, C. | 登録日 | 2016-05-17 | 公開日 | 2017-01-25 | 最終更新日 | 2023-09-27 | 実験手法 | X-RAY DIFFRACTION (1.83 Å) | 主引用文献 | The EED protein-protein interaction inhibitor A-395 inactivates the PRC2 complex. Nat. Chem. Biol., 13, 2017
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1LYW
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![BU of 1lyw by Molmil](/molmil-images/mine/1lyw) | CATHEPSIN D AT PH 7.5 | 分子名称: | 4-(2-HYDROXYETHYL)-1-PIPERAZINE ETHANESULFONIC ACID, CATHEPSIN D | 著者 | Lee, A.Y, Gulnik, S.V, Erickson, J.W. | 登録日 | 1998-06-30 | 公開日 | 1999-07-22 | 最終更新日 | 2023-08-09 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Conformational switching in an aspartic proteinase. Nat.Struct.Biol., 5, 1998
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4OD2
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![BU of 4od2 by Molmil](/molmil-images/mine/4od2) | |
7AZY
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7LQ6
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![BU of 7lq6 by Molmil](/molmil-images/mine/7lq6) | CryoEM structure of Escherichia coli PBP1b | 分子名称: | Penicillin-binding protein 1B | 著者 | Caveney, N.A, Workman, S.D, Yan, R, Atkinson, C.E, Yu, Z, Strynadka, N.C.J. | 登録日 | 2021-02-13 | 公開日 | 2021-05-26 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.28 Å) | 主引用文献 | CryoEM structure of the antibacterial target PBP1b at 3.3 angstrom resolution. Nat Commun, 12, 2021
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1VRL
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![BU of 1vrl by Molmil](/molmil-images/mine/1vrl) | MutY adenine glycosylase in complex with DNA and soaked adenine free base | 分子名称: | 5'-D(*AP*AP*GP*AP*CP*(8OG)P*TP*GP*GP*AP*C)-3', 5'-D(*TP*GP*TP*CP*CP*AP*(HPD)P*GP*TP*CP*T)-3', ADENINE, ... | 著者 | Fromme, J.C, Banerjee, A, Huang, S.J, Verdine, G.L. | 登録日 | 2005-03-08 | 公開日 | 2005-03-22 | 最終更新日 | 2023-12-27 | 実験手法 | X-RAY DIFFRACTION (2.5 Å) | 主引用文献 | Structural basis for removal of adenine mispaired with 8-oxoguanine by MutY adenine DNA glycosylase Nature, 427, 2004
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5UN6
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5UN5
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![BU of 5un5 by Molmil](/molmil-images/mine/5un5) | |
1RRQ
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![BU of 1rrq by Molmil](/molmil-images/mine/1rrq) | MutY adenine glycosylase in complex with DNA containing an A:oxoG pair | 分子名称: | 5'-D(*TP*GP*TP*CP*CP*AP*AP*GP*TP*CP*T)-3', 5'-D(AP*AP*GP*AP*CP*(8OG)P*TP*GP*GP*AP*C)-3', CALCIUM ION, ... | 著者 | Fromme, J.C, Banerjee, A, Huang, S.J, Verdine, G.L. | 登録日 | 2003-12-08 | 公開日 | 2004-02-17 | 最終更新日 | 2024-02-14 | 実験手法 | X-RAY DIFFRACTION (2.22 Å) | 主引用文献 | Structural basis for removal of adenine mispaired with 8-oxoguanine by MutY adenine DNA glycosylase Nature, 427, 2004
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1RRS
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![BU of 1rrs by Molmil](/molmil-images/mine/1rrs) | MutY adenine glycosylase in complex with DNA containing an abasic site | 分子名称: | 5'-D(*AP*AP*GP*AP*CP*(8OG)P*TP*GP*GP*AP*C)-3', 5'-D(*TP*GP*TP*CP*CP*AP*(HPD)P*GP*TP*CP*T)-3', CALCIUM ION, ... | 著者 | Fromme, J.C, Banerjee, A, Huang, S.J, Verdine, G.L. | 登録日 | 2003-12-08 | 公開日 | 2004-02-17 | 最終更新日 | 2023-08-23 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Structural basis for removal of adenine mispaired with 8-oxoguanine by MutY adenine DNA glycosylase Nature, 427, 2004
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1MA7
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![BU of 1ma7 by Molmil](/molmil-images/mine/1ma7) | |
1J3H
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![BU of 1j3h by Molmil](/molmil-images/mine/1j3h) | Crystal structure of apoenzyme cAMP-dependent protein kinase catalytic subunit | 分子名称: | (4S)-2-METHYL-2,4-PENTANEDIOL, cAMP-dependent protein kinase, alpha-catalytic subunit | 著者 | Akamine, P, Madhusudan, Wu, J, Xuong, N.H, Ten Eyck, L.F, Taylor, S.S. | 登録日 | 2003-01-31 | 公開日 | 2003-03-04 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (2.9 Å) | 主引用文献 | Dynamic Features of cAMP-dependent Protein Kinase Revealed by Apoenzyme Crystal Structure J.Mol.Biol., 327, 2003
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