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PDB: 2 件

5NOB
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BU of 5nob by Molmil
Crystal structure of human tankyrase 2 in complex with OD336
分子名称: 1-[3-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]cyclobutyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, Tankyrase-2, ZINC ION
著者Ignatev, A, Lehtio, L.
登録日2017-04-11
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach.
J. Med. Chem., 60, 2017
5NSP
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BU of 5nsp by Molmil
Crystal structure of TNKS2 in complex with OD334
分子名称: 1-[4-[4-(2-chlorophenyl)-5-pyrimidin-4-yl-1,2,4-triazol-3-yl]phenyl]-2-oxidanylidene-3~{H}-benzimidazole-5-carbonitrile, BICARBONATE ION, GLYCEROL, ...
著者Nkizinkiko, Y, Haikarainen, T, Lehtio, L.
登録日2017-04-26
公開日2017-11-29
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Discovery of a Novel Series of Tankyrase Inhibitors by a Hybridization Approach.
J. Med. Chem., 60, 2017

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件を2024-10-09に公開中

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