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PDB: 7 件

1WBU
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BU of 1wbu by Molmil
Fragment based lead discovery using crystallography
分子名称: 5-AMINO-1H-PYRIMIDINE-2,4-DIONE, RIBONUCLEASE
著者Cleasby, A, Hartshorn, M.J, Murray, C.W, Jhoti, H, Tickle, I.J.
登録日2004-11-05
公開日2005-01-27
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1WBO
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BU of 1wbo by Molmil
fragment based p38 inhibitors
分子名称: 2-CHLOROPHENOL, MITOGEN-ACTIVATED PROTEIN KINASE 14
著者Cleasby, A, Devine, L, Gill, A, Jhoti, H.
登録日2004-11-04
公開日2005-01-27
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.16 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1WCC
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BU of 1wcc by Molmil
Screening for fragment binding by X-ray crystallography
分子名称: 2-AMINO-6-CHLOROPYRAZINE, CELL DIVISION PROTEIN KINASE 2
著者Cleasby, A, O'Reilly, M, Hartshorn, M.J, Murray, C.W, Tickle, I.J, Jhoti, H, Frederickson, M.
登録日2004-11-12
公開日2005-01-27
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1WAY
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BU of 1way by Molmil
Active site thrombin inhibitors
分子名称: 4-[3-(4-CHLOROPHENYL)-1H-PYRAZOL-5-YL]PIPERIDINE, DIMETHYL SULFOXIDE, HIRUGEN, ...
著者Hartshorn, M.J, Murray, C.W, Cleasby, A, Frederickson, M, Tickle, I.J, Jhoti, H.
登録日2004-10-28
公開日2005-01-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1WBG
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BU of 1wbg by Molmil
Active site thrombin inhibitors
分子名称: 3-(4-CHLOROPHENYL)-5-(METHYLTHIO)-4H-1,2,4-TRIAZOLE, DIMETHYL SULFOXIDE, HIRUGEN, ...
著者Hartshorn, M.J, Murray, C.W, Cleasby, A, Frederickson, M, Tickle, I.J, Jhoti, H.
登録日2004-11-01
公開日2005-01-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1WAX
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BU of 1wax by Molmil
Protein tyrosine phosphatase 1B with active site inhibitor
分子名称: MAGNESIUM ION, PROTEIN-TYROSINE PHOSPHATASE, [[4-(AMINOMETHYL)PHENYL]AMINO]OXO-ACETIC ACID,
著者Hartshorn, M.J, Murray, C.W, Cleasby, A, Frederickson, M, Tickle, I.J, Jhoti, H.
登録日2004-10-28
公開日2005-01-27
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005
1W7H
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BU of 1w7h by Molmil
p38 Kinase crystal structure in complex with small molecule inhibitor
分子名称: 3-(BENZYLOXY)PYRIDIN-2-AMINE, MITOGEN-ACTIVATED PROTEIN KINASE 14
著者Jhoti, H, Gill, A, Cleasby, A, Devine, L.
登録日2004-09-02
公開日2005-02-08
最終更新日2023-12-13
実験手法X-RAY DIFFRACTION (2.214 Å)
主引用文献Fragment-Based Lead Discovery Using X-Ray Crystallography
J.Med.Chem., 48, 2005

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件を2024-07-31に公開中

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