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PDB: 2 件

6FYM
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BU of 6fym by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK1
分子名称: 7,8-dimethyl-2-(pyrimidin-2-ylsulfanylmethyl)-3~{H}-quinazolin-4-one, NITRATE ION, Poly [ADP-ribose] polymerase 14
著者Karlberg, T, Thorsell, A.G, Kirby, I.T, Sreenivasan, R, Cohen, M.S, Schuler, H.
登録日2018-03-12
公開日2019-02-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献A Potent and Selective PARP11 Inhibitor Suggests Coupling between Cellular Localization and Catalytic Activity.
Cell Chem Biol, 25, 2018
6FZM
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BU of 6fzm by Molmil
Human PARP14 (ARTD8), catalytic fragment in complex with inhibitor ITK6
分子名称: 4-[(8-methyl-4-oxidanylidene-7-prop-1-ynyl-3~{H}-quinazolin-2-yl)methylsulfanyl]benzoic acid, Poly [ADP-ribose] polymerase 14
著者Karlberg, T, Thorsell, A.G, Kirby, I.T, Sreenivasan, R, Cohen, M.S, Schuler, H.
登録日2018-03-15
公開日2019-02-20
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (2.67 Å)
主引用文献A Potent and Selective PARP11 Inhibitor Suggests Coupling between Cellular Localization and Catalytic Activity.
Cell Chem Biol, 25, 2018

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件を2024-10-09に公開中

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