8IPY
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8IDY
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8IPD
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8INF
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8IDT
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8IR1
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6J1L
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![BU of 6j1l by Molmil](/molmil-images/mine/6j1l) | Crystal Structure Analysis of the ROR gamma(C455E) | 分子名称: | 2-[4-(ethylsulfonyl)phenyl]-N-[2'-fluoro-4'-(1,1,1,3,3,3-hexafluoro-2-hydroxypropan-2-yl)[1,1'-biphenyl]-4-yl]acetamide, Nuclear receptor ROR-gamma | 著者 | zhang, Y, Li, C.C, wu, X.S. | 登録日 | 2018-12-28 | 公開日 | 2019-05-01 | 最終更新日 | 2023-11-22 | 実験手法 | X-RAY DIFFRACTION (2.3 Å) | 主引用文献 | Discovery and Characterization of XY101, a Potent, Selective, and Orally Bioavailable ROR gamma Inverse Agonist for Treatment of Castration-Resistant Prostate Cancer. J.Med.Chem., 62, 2019
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8XNG
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8XS4
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8XW3
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8XW1
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8XVY
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8XW2
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8XRY
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8XS5
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8XW0
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![BU of 8xw0 by Molmil](/molmil-images/mine/8xw0) | Cryo-EM structure of OSCA3.1-GDN state | 分子名称: | CSC1-like protein ERD4, O-[(R)-{[(2R)-2,3-bis(octadecanoyloxy)propyl]oxy}(hydroxy)phosphoryl]-L-serine | 著者 | Zhang, Y, Han, Y. | 登録日 | 2024-01-15 | 公開日 | 2024-04-10 | 最終更新日 | 2024-05-08 | 実験手法 | ELECTRON MICROSCOPY (3.11 Å) | 主引用文献 | Mechanical activation opens a lipid-lined pore in OSCA ion channels. Nature, 628, 2024
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8XVZ
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8XW4
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8XAJ
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8XVX
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8XS0
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6VRJ
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6VYM
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![BU of 6vym by Molmil](/molmil-images/mine/6vym) | Cryo-EM structure of mechanosensitive channel MscS in PC-18:1 nanodiscs treated with beta-cyclodextran | 分子名称: | Mechanosensitive channel MscS | 著者 | Zhang, Y, Daday, C, Gu, R, Cox, C.D, Martinac, B, Groot, B, Walz, T. | 登録日 | 2020-02-27 | 公開日 | 2021-02-10 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.7 Å) | 主引用文献 | Visualization of the mechanosensitive ion channel MscS under membrane tension. Nature, 590, 2021
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6VYK
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![BU of 6vyk by Molmil](/molmil-images/mine/6vyk) | Cryo-EM structure of mechanosensitive channel MscS in PC-18:1 nanodiscs | 分子名称: | 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, Mechanosensitive channel MscS | 著者 | Zhang, Y, Daday, C, Gu, R, Cox, C.D, Martinac, B, Groot, B, Walz, T. | 登録日 | 2020-02-27 | 公開日 | 2021-02-10 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.2 Å) | 主引用文献 | Visualization of the mechanosensitive ion channel MscS under membrane tension. Nature, 590, 2021
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6VYL
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![BU of 6vyl by Molmil](/molmil-images/mine/6vyl) | Cryo-EM structure of mechanosensitive channel MscS in PC-10 nanodiscs | 分子名称: | Mechanosensitive channel MscS | 著者 | Zhang, Y, Daday, C, Gu, R, Cox, C.D, Martinac, B, Groot, B, Walz, T. | 登録日 | 2020-02-27 | 公開日 | 2021-02-10 | 最終更新日 | 2024-03-06 | 実験手法 | ELECTRON MICROSCOPY (3.4 Å) | 主引用文献 | Visualization of the mechanosensitive ion channel MscS under membrane tension. Nature, 590, 2021
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