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PDB: 78 results

7UBK
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BU of 7ubk by Molmil
Transcription antitermination factor Qlambda, type-II crystal
Descriptor: 1,2-ETHANEDIOL, Antitermination protein Q, CHLORIDE ION, ...
Authors:Yin, Z, Ebright, R.H.
Deposit date:2022-03-15
Release date:2022-09-28
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.97 Å)
Cite:In transcription antitermination by Q lambda , NusA induces refolding of Q lambda to form a nozzle that extends the RNA polymerase RNA-exit channel.
Proc.Natl.Acad.Sci.USA, 119, 2022
7UBM
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BU of 7ubm by Molmil
Transcription antitermination complex: "pre-engaged" Qlambda-loading complex
Descriptor: Antitermination protein Q, DNA (52-MER), DNA (53-MER), ...
Authors:Yin, Z, Ebright, R.H.
Deposit date:2022-03-15
Release date:2022-09-28
Last modified:2024-06-12
Method:ELECTRON MICROSCOPY (3.13 Å)
Cite:In transcription antitermination by Q lambda , NusA induces refolding of Q lambda to form a nozzle that extends the RNA polymerase RNA-exit channel.
Proc.Natl.Acad.Sci.USA, 119, 2022
7UBN
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BU of 7ubn by Molmil
Transcription antitermination complex: NusA-containing "engaged" Qlambda-loading complex
Descriptor: Antitermination protein, DNA (52-MER), DNA (53-MER), ...
Authors:Yin, Z, Ebright, R.H.
Deposit date:2022-03-15
Release date:2022-09-28
Last modified:2024-06-12
Method:ELECTRON MICROSCOPY (3.36 Å)
Cite:In transcription antitermination by Q lambda , NusA induces refolding of Q lambda to form a nozzle that extends the RNA polymerase RNA-exit channel.
Proc.Natl.Acad.Sci.USA, 119, 2022
5VPD
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BU of 5vpd by Molmil
Transcription factor FosB/JunD bZIP domain in its oxidized form, type-III crystal
Descriptor: CHLORIDE ION, Protein fosB, SODIUM ION, ...
Authors:Yin, Z, Machius, M, Rudenko, G.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.79 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
5VPE
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BU of 5vpe by Molmil
Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-I crystal
Descriptor: 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ...
Authors:Yin, Z, Machius, M, Rudenko, G.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.053 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
4K3M
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BU of 4k3m by Molmil
E.coli sliding clamp in complex with AcALDLF peptide
Descriptor: ALDLF, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3R
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BU of 4k3r by Molmil
E. coli sliding clamp in complex with AcQLDLA
Descriptor: (ACE)QLDLA, CALCIUM ION, CHLORIDE ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.86 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3L
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BU of 4k3l by Molmil
E. coli sliding clamp in complex with AcLF dipeptide
Descriptor: 1,2-ETHANEDIOL, ACETYL GROUP, CALCIUM ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-10
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.5 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
5VPB
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BU of 5vpb by Molmil
Transcription factor FosB/JunD bZIP domain in its oxidized form, type-I crystal
Descriptor: CHLORIDE ION, Protein fosB, Transcription factor jun-D
Authors:Yin, Z, Machius, M, Rudenko, G.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.691 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
5VPC
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BU of 5vpc by Molmil
Transcription factor FosB/JunD bZIP domain in its oxidized form, type-II crystal
Descriptor: CHLORIDE ION, Protein fosB, SODIUM ION, ...
Authors:Yin, Z, Machius, M.C, Rudenko, G.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.498 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
5VPA
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BU of 5vpa by Molmil
Transcription factor FosB/JunD bZIP domain
Descriptor: CHLORIDE ION, Protein fosB, SODIUM ION, ...
Authors:Yin, Z, Machius, M, Rudenko, G.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.83 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
5VPF
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BU of 5vpf by Molmil
Transcription factor FosB/JunD bZIP domain in complex with cognate DNA, type-II crystal
Descriptor: 1,2-ETHANEDIOL, CHLORIDE ION, DNA (5'-D(*CP*GP*TP*CP*GP*GP*TP*GP*AP*CP*TP*CP*AP*CP*CP*GP*AP*CP*G)-3'), ...
Authors:Yin, Z, Rudenko, G, Machius, M.
Deposit date:2017-05-04
Release date:2017-09-06
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (2.694 Å)
Cite:Activator Protein-1: redox switch controlling structure and DNA-binding.
Nucleic Acids Res., 45, 2017
4K3Q
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BU of 4k3q by Molmil
E. coli sliding clamp in complex with AcQLDAF
Descriptor: (ACE)QLDAF, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3S
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BU of 4k3s by Molmil
E. coli sliding clamp in P1 crystal space group
Descriptor: CALCIUM ION, DNA polymerase III subunit beta, O-ACETALDEHYDYL-HEXAETHYLENE GLYCOL, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.75 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3O
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BU of 4k3o by Molmil
E. coli sliding clamp in complex with AcQADLF
Descriptor: (ACE)QADLF, 1,2-ETHANEDIOL, CALCIUM ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3K
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BU of 4k3k by Molmil
E. Coli sliding clamp in complex with (S)-2-(4-methylpentanamido)-3-phenylpropanoic acid
Descriptor: CALCIUM ION, CHLORIDE ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-10
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (1.85 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
4K3P
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BU of 4k3p by Molmil
E. coli sliding clamp in complex with AcQLALF
Descriptor: (ACE)QLALF, 1,2-ETHANEDIOL, CALCIUM ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-04-11
Release date:2013-05-01
Last modified:2023-11-08
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Structural and Thermodynamic Dissection of Linear Motif Recognition by the E. coli Sliding Clamp
J.Med.Chem., 56, 2013
5EJK
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BU of 5ejk by Molmil
Crystal structure of the Rous sarcoma virus intasome
Descriptor: DNA (5'-D(*AP*AP*TP*GP*TP*TP*GP*TP*CP*TP*TP*AP*TP*GP*CP*AP*AP*TP*AP*CP*TP*C)-3'), DNA (5'-D(*AP*GP*TP*GP*TP*CP*TP*T)-3'), DNA (5'-D(*CP*TP*TP*CP*TP*CP*TP*C)-3'), ...
Authors:Yin, Z, Shi, K, Banerjee, S, Aihara, H.
Deposit date:2015-11-02
Release date:2016-02-17
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Crystal structure of the Rous sarcoma virus intasome.
Nature, 530, 2016
4N96
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BU of 4n96 by Molmil
E. coli sliding clamp in complex with 6-nitroindazole
Descriptor: 6-NITROINDAZOLE, CALCIUM ION, CHLORIDE ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-10-19
Release date:2013-11-06
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.7 Å)
Cite:Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4OVF
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BU of 4ovf by Molmil
E. coli sliding clamp in complex with (R)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid
Descriptor: (2R)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2014-02-21
Release date:2014-03-05
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.05 Å)
Cite:Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs.
J.Med.Chem., 58, 2015
4N94
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BU of 4n94 by Molmil
E. coli sliding clamp in complex with 3,4-difluorobenzamide
Descriptor: 1,2-ETHANEDIOL, 3,4-difluorobenzamide, CALCIUM ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-10-19
Release date:2013-11-06
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.73 Å)
Cite:Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4PNW
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BU of 4pnw by Molmil
E. coli sliding clamp in complex with (R)-6-bromo-9-(2-((S)-1-carboxy-2-phenylethylamino)-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid
Descriptor: (2R)-6-bromo-9-(2-{[(1S)-1-carboxy-2-phenylethyl]amino}-2-oxoethyl)-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, CALCIUM ION, CHLORIDE ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2014-02-21
Release date:2014-03-05
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2 Å)
Cite:Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs.
J.Med.Chem., 58, 2015
4N97
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BU of 4n97 by Molmil
E. coli sliding clamp in complex with 5-nitroindole
Descriptor: 5-nitro-1H-indole, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-10-19
Release date:2013-11-06
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (1.97 Å)
Cite:Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4N99
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BU of 4n99 by Molmil
E. coli sliding clamp in complex with 6-chloro-2,3,4,9-tetrahydro-1H-carbazole-7-carboxylic acid
Descriptor: 6-chloro-2,3,4,9-tetrahydro-1H-carbazole-7-carboxylic acid, CALCIUM ION, DI(HYDROXYETHYL)ETHER, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2013-10-19
Release date:2013-11-06
Last modified:2023-09-20
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Discovery of lead compounds targeting the bacterial sliding clamp using a fragment-based approach.
J.Med.Chem., 57, 2014
4OVG
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BU of 4ovg by Molmil
E. coli sliding clamp in complex with (R)-9-(2-amino-2-oxoethyl)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid
Descriptor: (2R)-9-(2-amino-2-oxoethyl)-6-chloro-2,3,4,9-tetrahydro-1H-carbazole-2-carboxylic acid, 1,2-ETHANEDIOL, CALCIUM ION, ...
Authors:Yin, Z, Oakley, A.J.
Deposit date:2014-02-21
Release date:2014-03-05
Last modified:2024-02-28
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Bacterial Sliding Clamp Inhibitors that Mimic the Sequential Binding Mechanism of Endogenous Linear Motifs.
J.Med.Chem., 58, 2015

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